The adenosine-triphosphate-sensitive potassium-channel opener pinacidil is effective in blood cardioplegia

Ann Thorac Surg. 1998 Sep;66(3):768-73. doi: 10.1016/s0003-4975(98)00471-8.

Abstract

Background: This study was designed to evaluate the adenosine-triphosphate-sensitive potassium channel opener pinacidil as a blood cardioplegic agent.

Methods: Using a blood-perfused, parabiotic, Langendorff rabbit model, hearts underwent 30 minutes of normothermic ischemia protected with blood cardioplegia (St. Thomas' solution [n = 8] or Krebs-Henseleit solution with pinacidil [50 micromol/L, n = 81) and 30 minutes of reperfusion. Percent recovery of developed pressure, mechanical arrest, electrical arrest, reperfusion ventricular fibrillation, percent tissue water, and myocardial oxygen consumption were compared.

Results: The percent recovery of developed pressure was not different between the groups (52.3 +/- 5.9 and 52.8 +/- 6.9 for hyperkalemic and pinacidil cardioplegia, respectively). Pinacidil cardioplegia was associated with prolonged electrical and mechanical activity (14.4 +/- 8.7 and 6.1 +/- 3.9 minutes), compared with hyperkalemic cardioplegia (1.1 +/- 0.6 and 1.1 +/- 0.6 minutes, respectively; p < 0.05). Pinacidil cardioplegia was associated with a higher reperfusion myocardial oxygen consumption (0.6 +/- 0.1 versus 0.2 +/- 0.0 mL/100 g myocardium/beat; p < 0.05) and a higher percent of tissue water (79.6% +/- 0.7% versus 78.6% +/- 1.2%; p < 0.05).

Conclusions: Systolic recovery was not different between groups, demonstrating comparable effectiveness of pinacidil and hyperkalemic warm blood cardioplegia.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Cardioplegic Solutions*
  • Electrophysiology
  • Female
  • Guanidines / pharmacology*
  • Heart / physiology
  • Heart Arrest, Induced*
  • In Vitro Techniques
  • Male
  • Myocardial Reperfusion
  • Myocardium / metabolism
  • Oxygen Consumption
  • Pinacidil
  • Potassium Channels* / drug effects
  • Rabbits
  • Random Allocation
  • Vasodilator Agents / pharmacology*

Substances

  • Cardioplegic Solutions
  • Guanidines
  • Potassium Channels
  • Vasodilator Agents
  • Pinacidil