March DR - Search Results

1

Conformational selection of inhibitors and substrates by proteolytic enzymes: implications for drug design and polypeptide processing.

Fairlie DP, Tyndall JD, Reid RC, Wong AK, Abbenante G, Scanlon MJ, March DR, Bergman DA, Chai CL, Burkett BA. Fairlie DP, et al. Among authors: march dr. J Med Chem. 2000 Apr 6;43(7):1271-81. doi: 10.1021/jm990315t. J Med Chem. 2000. PMID: 10753465

2

Molecular recognition of macrocyclic peptidomimetic inhibitors by HIV-1 protease.

Martin JL, Begun J, Schindeler A, Wickramasinghe WA, Alewood D, Alewood PF, Bergman DA, Brinkworth RI, Abbenante G, March DR, Reid RC, Fairlie DP. Martin JL, et al. Among authors: march dr. Biochemistry. 1999 Jun 22;38(25):7978-88. doi: 10.1021/bi990174x. Biochemistry. 1999. PMID: 10387041

3

Synthesis, stability, antiviral activity, and protease-bound structures of substrate-mimicking constrained macrocyclic inhibitors of HIV-1 protease.

Tyndall JD, Reid RC, Tyssen DP, Jardine DK, Todd B, Passmore M, March DR, Pattenden LK, Bergman DA, Alewood D, Hu SH, Alewood PF, Birch CJ, Martin JL, Fairlie DP. Tyndall JD, et al. Among authors: march dr. J Med Chem. 2000 Sep 21;43(19):3495-504. doi: 10.1021/jm000013n. J Med Chem. 2000. PMID: 11000004

4

Potent cyclic antagonists of the complement C5a receptor on human polymorphonuclear leukocytes. Relationships between structures and activity.

March DR, Proctor LM, Stoermer MJ, Sbaglia R, Abbenante G, Reid RC, Woodruff TM, Wadi K, Paczkowski N, Tyndall JD, Taylor SM, Fairlie DP. March DR, et al. Mol Pharmacol. 2004 Apr;65(4):868-79. doi: 10.1124/mol.65.4.868. Mol Pharmacol. 2004. PMID: 15044616

5

A cyclic metallopeptide induces alpha helicity in short peptide fragments of thermolysin.

Kelso MJ, Hoang HN, Oliver W, Sokolenko N, March DR, Appleton TG, Fairlie DP. Kelso MJ, et al. Among authors: march dr. Angew Chem Int Ed Engl. 2003 Jan 27;42(4):421-4. doi: 10.1002/anie.200390128. Angew Chem Int Ed Engl. 2003. PMID: 12569506 No abstract available.

6

Analogues of SB-203207 as inhibitors of tRNA synthetases.

Banwell MG, Crasto CF, Easton CJ, Forrest AK, Karoli T, March DR, Mensah L, Nairn MR, O'Hanlon PJ, Oldham MD, Yue W. Banwell MG, et al. Among authors: march dr. Bioorg Med Chem Lett. 2000 Oct 16;10(20):2263-6. doi: 10.1016/s0960-894x(00)00456-x. Bioorg Med Chem Lett. 2000. PMID: 11055334

7

Synthesis and activity of analogues of the isoleucyl tRNA synthetase inhibitor SB-203207.

Crasto CF, Forrest AK, Karoli T, March DR, Mensah L, O'Hanlon PJ, Nairn MR, Oldham MD, Yue W, Banwell MG, Easton CJ. Crasto CF, et al. Among authors: march dr. Bioorg Med Chem. 2003 Jul 3;11(13):2687-94. doi: 10.1016/s0968-0896(03)00237-2. Bioorg Med Chem. 2003. PMID: 12788342

8

Multi-component assembly of the bicyclic core associated with the tRNA synthetase inhibitors SB-203207 and SB-203208. Application to the synthesis of biologically active analogues.

Banwell MG, Crasto CF, Easton CJ, Karoli T, March DR, Nairn MR, O'Hanlon PJ, Oldham MD, Willis AC, Yue W. Banwell MG, et al. Among authors: march dr. Chem Commun (Camb). 2001 Nov 7;(21):2210-1. Chem Commun (Camb). 2001. PMID: 12240115

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

8 results

Search Page

Filters