Stapelfeld A - Search Results

1

2,4-Disubstituted oxazoles and thiazoles as latent pharmacophores for diacylhydrazine of SC-51089, a potent PGE2 antagonist.

Hallinan EA, Hagen TJ, Tsymbalov S, Stapelfeld A, Savage MA. Hallinan EA, et al. Among authors: stapelfeld a. Bioorg Med Chem. 2001 Jan;9(1):1-6. doi: 10.1016/s0968-0896(00)00229-7. Bioorg Med Chem. 2001. PMID: 11197330

2

N-substituted dibenzoxazepines as analgesic PGE2 antagonists.

Hallinan EA, Hagen TJ, Husa RK, Tsymbalov S, Rao SN, vanHoeck JP, Rafferty MF, Stapelfeld A, Savage MA, Reichman M. Hallinan EA, et al. Among authors: stapelfeld a. J Med Chem. 1993 Oct 29;36(22):3293-9. doi: 10.1021/jm00074a010. J Med Chem. 1993. PMID: 7901416

3

Enkephalin analogs as systemically active antinociceptive agents: O- and N-alkylated derivatives of the dipeptide amide L-2,6-dimethyltyrosyl-N-(3-phenylpropyl)-D-alaninamide.

Pitzele BS, Hamilton RW, Kudla KD, Tsymbalov S, Stapelfeld A, Savage MA, Clare M, Hammond DL, Hansen DW Jr. Pitzele BS, et al. Among authors: stapelfeld a. J Med Chem. 1994 Apr 1;37(7):888-96. doi: 10.1021/jm00033a005. J Med Chem. 1994. PMID: 7908696

4

Aminoacetyl moiety as a potential surrogate for diacylhydrazine group of SC-51089, a potent PGE2 antagonist, and its analogs.

Hallinan EA, Hagen TJ, Tsymbalov S, Husa RK, Lee AC, Stapelfeld A, Savage MA. Hallinan EA, et al. Among authors: stapelfeld a. J Med Chem. 1996 Jan 19;39(2):609-13. doi: 10.1021/jm950454k. J Med Chem. 1996. PMID: 8558534

5

Systemic analgesic activity and delta-opioid selectivity in [2,6-dimethyl-Tyr1,D-Pen2,D-Pen5]enkephalin.

Hansen DW Jr, Stapelfeld A, Savage MA, Reichman M, Hammond DL, Haaseth RC, Mosberg HI. Hansen DW Jr, et al. Among authors: stapelfeld a. J Med Chem. 1992 Feb 21;35(4):684-7. doi: 10.1021/jm00082a008. J Med Chem. 1992. PMID: 1311764

6

Analogs of the delta opioid receptor selective cyclic peptide [2-D-penicillamine,5-D-penicillamine]-enkephalin: 2',6'-dimethyltyrosine and Gly3-Phe4 amide bond isostere substitutions.

Chandrakumar NS, Stapelfeld A, Beardsley PM, Lopez OT, Drury B, Anthony E, Savage MA, Williamson LN, Reichman M. Chandrakumar NS, et al. Among authors: stapelfeld a. J Med Chem. 1992 Aug 7;35(16):2928-38. doi: 10.1021/jm00094a002. J Med Chem. 1992. PMID: 1323677

7

Preparation and opioid activity of analogues of the analgesic dipeptide 2,6-dimethyl-L-tyrosyl-N-(3-phenylpropyl)-D-alaninamide.

Chandrakumar NS, Yonan PK, Stapelfeld A, Savage M, Rorbacher E, Contreras PC, Hammond D. Chandrakumar NS, et al. Among authors: stapelfeld a. J Med Chem. 1992 Jan 24;35(2):223-33. doi: 10.1021/jm00080a005. J Med Chem. 1992. PMID: 1346276

8

Antinociception produced by oral, subcutaneous or intrathecal administration of SC-39566, an opioid dipeptide arylalkylamide, in the rodent.

Hammond DL, Stapelfeld A, Drower EJ, Savage MA, Tam L, Mazur RH. Hammond DL, et al. Among authors: stapelfeld a. J Pharmacol Exp Ther. 1994 Feb;268(2):607-15. J Pharmacol Exp Ther. 1994. PMID: 8113971

9

Antinociception after intracerebroventricular administration of naltrindole in the mouse.

Stapelfeld A, Hammond DL, Rafferty MF. Stapelfeld A, et al. Eur J Pharmacol. 1992 Apr 22;214(2-3):273-6. doi: 10.1016/0014-2999(92)90129-r. Eur J Pharmacol. 1992. PMID: 1325358

10

Selective antagonism by naltrindole of the antinociceptive effects of the delta opioid agonist cyclic[D-penicillamine2-D-penicillamine5]enkephalin in the rat.

Drower EJ, Stapelfeld A, Rafferty MF, de Costa BR, Rice KC, Hammond DL. Drower EJ, et al. Among authors: stapelfeld a. J Pharmacol Exp Ther. 1991 Nov;259(2):725-31. J Pharmacol Exp Ther. 1991. PMID: 1658309

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

11 results

Search Page

Filters