Classon B - Search Results

1

P1/P1' modified HIV protease inhibitors as tools in two new sensitive surface plasmon resonance biosensor screening assays.

Alterman M, Sjöbom H, Säfsten P, Markgren PO, Danielson UH, Hämäläinen M, Löfås S, Hultén J, Classon B, Samuelsson B, Hallberg A. Alterman M, et al. Among authors: classon b. Eur J Pharm Sci. 2001 May;13(2):203-12. doi: 10.1016/s0928-0987(01)00109-9. Eur J Pharm Sci. 2001. PMID: 11297905

2

Optimization of P1-P3 groups in symmetric and asymmetric HIV-1 protease inhibitors.

Andersson HO, Fridborg K, Löwgren S, Alterman M, Mühlman A, Björsne M, Garg N, Kvarnström I, Schaal W, Classon B, Karlén A, Danielsson UH, Ahlsén G, Nillroth U, Vrang L, Oberg B, Samuelsson B, Hallberg A, Unge T. Andersson HO, et al. Among authors: classon b. Eur J Biochem. 2003 Apr;270(8):1746-58. doi: 10.1046/j.1432-1033.2003.03533.x. Eur J Biochem. 2003. PMID: 12694187 Free article.

3

Cyclic HIV-1 protease inhibitors derived from mannitol: synthesis, inhibitory potencies, and computational predictions of binding affinities.

Hultén J, Bonham NM, Nillroth U, Hansson T, Zuccarello G, Bouzide A, Aqvist J, Classon B, Danielson UH, Karlén A, Kvarnström I, Samuelsson B, Hallberg A. Hultén J, et al. Among authors: classon b. J Med Chem. 1997 Mar 14;40(6):885-97. doi: 10.1021/jm960728j. J Med Chem. 1997. PMID: 9083477

4

Design and synthesis of new potent C2-symmetric HIV-1 protease inhibitors. Use of L-mannaric acid as a peptidomimetic scaffold.

Alterman M, Björsne M, Mühlman A, Classon B, Kvarnström I, Danielson H, Markgren PO, Nillroth U, Unge T, Hallberg A, Samuelsson B. Alterman M, et al. Among authors: classon b. J Med Chem. 1998 Sep 24;41(20):3782-92. doi: 10.1021/jm970777b. J Med Chem. 1998. PMID: 9748353

5

Design and fast synthesis of C-terminal duplicated potent C(2)-symmetric P1/P1'-modified HIV-1 protease inhibitors.

Alterman M, Andersson HO, Garg N, Ahlsén G, Lövgren S, Classon B, Danielson UH, Kvarnström I, Vrang L, Unge T, Samuelsson B, Hallberg A. Alterman M, et al. Among authors: classon b. J Med Chem. 1999 Sep 23;42(19):3835-44. doi: 10.1021/jm9910371. J Med Chem. 1999. PMID: 10508432

6

Characterization of a set of HIV-1 protease inhibitors using binding kinetics data from a biosensor-based screen.

Hämäläinen MD, Markgren PO, Schaal W, Karlén A, Classon B, Vrang L, Samuelsson B, Hallberg A, Danielson UH. Hämäläinen MD, et al. Among authors: classon b. J Biomol Screen. 2000 Oct;5(5):353-60. doi: 10.1177/108705710000500507. J Biomol Screen. 2000. PMID: 11080694

7

Synthesis and comparative molecular field analysis (CoMFA) of symmetric and nonsymmetric cyclic sulfamide HIV-1 protease inhibitors.

Schaal W, Karlsson A, Ahlsén G, Lindberg J, Andersson HO, Danielson UH, Classon B, Unge T, Samuelsson B, Hultén J, Hallberg A, Karlén A. Schaal W, et al. Among authors: classon b. J Med Chem. 2001 Jan 18;44(2):155-69. doi: 10.1021/jm001024j. J Med Chem. 2001. PMID: 11170625

8

Synthesis of potent C(2)-symmetric, diol-based hiv-1 protease inhibitors. Investigation of thioalkyl and thioaryl P1/P1' substituents.

Mühlman A, Classon B, Hallberg A, Samuelsson B. Mühlman A, et al. Among authors: classon b. J Med Chem. 2001 Oct 11;44(21):3402-6. doi: 10.1021/jm0011169. J Med Chem. 2001. PMID: 11585445

9

Symmetric fluoro-substituted diol-based HIV protease inhibitors. Ortho-fluorinated and meta-fluorinated P1/P1'-benzyloxy side groups significantly improve the antiviral activity and preserve binding efficacy.

Lindberg J, Pyring D, Löwgren S, Rosenquist A, Zuccarello G, Kvarnström I, Zhang H, Vrang L, Classon B, Hallberg A, Samuelsson B, Unge T. Lindberg J, et al. Among authors: classon b. Eur J Biochem. 2004 Nov;271(22):4594-602. doi: 10.1111/j.1432-1033.2004.04431.x. Eur J Biochem. 2004. PMID: 15560801 Free article.

10

Inhibitors of the C(2)-symmetric HIV-1 protease: nonsymmetric binding of a symmetric cyclic sulfamide with ketoxime groups in the P2/P2' side chains.

Hultén J, Andersson HO, Schaal W, Danielson HU, Classon B, Kvarnström I, Karlén A, Unge T, Samuelsson B, Hallberg A. Hultén J, et al. Among authors: classon b. J Med Chem. 1999 Oct 7;42(20):4054-61. doi: 10.1021/jm991054q. J Med Chem. 1999. PMID: 10514275

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