Bousquet P - Search Results

1

Alpha2-adrenoreceptors profile modulation and high antinociceptive activity of (S)-(-)-2-[1-(biphenyl-2-yloxy)ethyl]-4,5-dihydro-1H-imidazole.

Gentili F, Bousquet P, Brasili L, Caretto M, Carrieri A, Dontenwill M, Giannella M, Marucci G, Perfumi M, Piergentili A, Quaglia W, Rascente C, Pigini M. Gentili F, et al. Among authors: bousquet p. J Med Chem. 2002 Jan 3;45(1):32-40. doi: 10.1021/jm0110082. J Med Chem. 2002. PMID: 11754577

2

Imidazoline binding sites (IBS) profile modulation: key role of the bridge in determining I1-IBS or I2-IBS selectivity within a series of 2-phenoxymethylimidazoline analogues.

Gentili F, Bousquet P, Brasili L, Dontenwill M, Feldman J, Ghelfi F, Giannella M, Piergentili A, Quaglia W, Pigini M. Gentili F, et al. Among authors: bousquet p. J Med Chem. 2003 May 22;46(11):2169-76. doi: 10.1021/jm021113r. J Med Chem. 2003. PMID: 12747788

3

Imidazoline receptors: qualitative structure-activity relationships and discovery of tracizoline and benazoline. Two ligands with high affinity and unprecedented selectivity.

Pigini M, Bousquet P, Carotti A, Dontenwill M, Giannella M, Moriconi R, Piergentili A, Quaglia W, Tayebati SK, Brasili L. Pigini M, et al. Among authors: bousquet p. Bioorg Med Chem. 1997 May;5(5):833-41. doi: 10.1016/s0968-0896(97)00009-6. Bioorg Med Chem. 1997. PMID: 9208095

4

2-D and 3-D modeling of imidazoline receptor ligands: insights into pharmacophore.

Carrieri A, Brasili L, Leonetti F, Pigini M, Giannella M, Bousquet P, Carotti A. Carrieri A, et al. Among authors: bousquet p. Bioorg Med Chem. 1997 May;5(5):843-56. doi: 10.1016/s0968-0896(97)00023-0. Bioorg Med Chem. 1997. PMID: 9208096

5

Ligand binding to I2 imidazoline receptor: the role of lipophilicity in quantitative structure-activity relationship models.

Pigini M, Bousquet P, Brasili L, Carrieri A, Cavagna R, Dontenwill M, Gentili F, Giannella M, Leonetti F, Piergentili A, Quaglia W, Carotti A. Pigini M, et al. Among authors: bousquet p. Bioorg Med Chem. 1998 Dec;6(12):2245-60. doi: 10.1016/s0968-0896(98)80005-9. Bioorg Med Chem. 1998. PMID: 9925287

6

2-(2-Phenylcyclopropyl)imidazolines: reversed enantioselective interaction at I(1) and I(2) imidazoline receptors.

Quaglia W, Bousquet P, Pigini M, Carotti A, Carrieri A, Dontenwill M, Gentili F, Giannella M, Maranca F, Piergentili A, Brasili L. Quaglia W, et al. Among authors: bousquet p. J Med Chem. 1999 Jul 29;42(15):2737-40. doi: 10.1021/jm991049m. J Med Chem. 1999. PMID: 10425083 No abstract available.

7

Methylation of imidazoline related compounds leads to loss of α₂-adrenoceptor affinity. Synthesis and biological evaluation of selective I₁ imidazoline receptor ligands.

Schann S, Greney H, Gasparik V, Dontenwill M, Rascente C, Lacroix G, Monassier L, Bruban V, Feldman J, Ehrhardt JD, Bousquet P. Schann S, et al. Among authors: bousquet p. Bioorg Med Chem. 2012 Aug 1;20(15):4710-5. doi: 10.1016/j.bmc.2012.06.008. Epub 2012 Jun 9. Bioorg Med Chem. 2012. PMID: 22750139

8

Structure-affinity relationship of cirazoline derivatives for idazoxan imidazoline-specific sites in the human cerebral cortex and the rabbit kidney.

Brasili L, Pigini M, Ehrhardt JD, Molines A, Greney H, Bousquet P, Dontenwill M. Brasili L, et al. Among authors: bousquet p. Ann N Y Acad Sci. 1995 Jul 12;763:149-52. doi: 10.1111/j.1749-6632.1995.tb32399.x. Ann N Y Acad Sci. 1995. PMID: 7677323 No abstract available.

9

Binding of tracizolines to the imidazoline receptor. Role of lipophilicity in quantitative structure-activity relationship models.

Pigini M, Bousquet P, Brasili L, Carrieri A, Dontenwill M, Gentili F, Giannella M, Leonetti F, Piergentili A, Quaglia W, Carotti A. Pigini M, et al. Among authors: bousquet p. Ann N Y Acad Sci. 1999 Jun 21;881:118-22. doi: 10.1111/j.1749-6632.1999.tb09351.x. Ann N Y Acad Sci. 1999. PMID: 10415907 No abstract available.

10

Coupling of I(1) imidazoline receptors to the cAMP pathway: studies with a highly selective ligand, benazoline.

Greney H, Ronde P, Magnier C, Maranca F, Rascente C, Quaglia W, Giannella M, Pigini M, Brasili L, Lugnier C, Bousquet P, Dontenwill M. Greney H, et al. Among authors: bousquet p. Mol Pharmacol. 2000 Jun;57(6):1142-51. Mol Pharmacol. 2000. PMID: 10825384

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

465 results

Search Page

Filters