Goulet MT - Search Results

1

2-Arylindoles as gonadotropin releasing hormone (GnRH) antagonists: optimization of the tryptamine side chain.

Young JR, Huang SX, Walsh TF, Wyvratt MJ, Yang YT, Yudkovitz JB, Cui J, Mount GR, Ren RN, Wu TJ, Shen X, Lyons KA, Mao AH, Carlin JR, Karanam BV, Vincent SH, Cheng K, Goulet MT. Young JR, et al. Among authors: goulet mt. Bioorg Med Chem Lett. 2002 Mar 11;12(5):827-32. doi: 10.1016/s0960-894x(02)00026-4. Bioorg Med Chem Lett. 2002. PMID: 11859012

2

Modification of the pyridine moiety of non-peptidyl indole GnRH receptor antagonists.

Simeone JP, Bugianesi RL, Ponpipom MM, Yang YT, Lo JL, Yudkovitz JB, Cui J, Mount GR, Ren RN, Creighton M, Mao AH, Vincent SH, Cheng K, Goulet MT. Simeone JP, et al. Among authors: goulet mt. Bioorg Med Chem Lett. 2002 Nov 18;12(22):3329-32. doi: 10.1016/s0960-894x(02)00751-5. Bioorg Med Chem Lett. 2002. PMID: 12392744

3

Design and syntheses of melanocortin subtype-4 receptor agonists: evolution of the pyridazinone archetype.

Ujjainwalla F, Warner D, Walsh TF, Wyvratt MJ, Zhou C, Yang L, Kalyani RN, MacNeil T, Van der Ploeg LH, Rosenblum CI, Tang R, Vongs A, Weinberg DH, Goulet MT. Ujjainwalla F, et al. Among authors: goulet mt. Bioorg Med Chem Lett. 2003 Dec 15;13(24):4431-5. doi: 10.1016/j.bmcl.2003.09.026. Bioorg Med Chem Lett. 2003. PMID: 14643340

4

Syntheses and structure-activity relationship studies of piperidine-substituted quinolones as nonpeptide gonadotropin releasing hormone antagonists.

Jiang J, DeVita RJ, Goulet MT, Wyvratt MJ, Lo JL, Ren N, Yudkovitz JB, Cui J, Yang YT, Cheng K, Rohrer SP. Jiang J, et al. Among authors: goulet mt. Bioorg Med Chem Lett. 2004 Apr 5;14(7):1795-8. doi: 10.1016/j.bmcl.2003.12.101. Bioorg Med Chem Lett. 2004. PMID: 15026074

5

Identification of neutral 4-O-alkyl quinolone nonpeptide GnRH receptor antagonists.

DeVita RJ, Parikh M, Jiang J, Fair JA, Young JR, Walsh TF, Goulet MT, Lo JL, Ren N, Yudkovitz JB, Cui J, Yang YT, Cheng K, Rohrer SP, Wyvratt MJ. DeVita RJ, et al. Among authors: goulet mt. Bioorg Med Chem Lett. 2004 Nov 15;14(22):5599-603. doi: 10.1016/j.bmcl.2004.08.056. Bioorg Med Chem Lett. 2004. PMID: 15482932

6

Identification and initial structure-activity relationships of a novel non-peptide quinolone GnRH receptor antagonist.

DeVita RJ, Hollings DD, Goulet MT, Wyvratt MJ, Fisher MH, Lo JL, Yang YT, Cheng K, Smith RG. DeVita RJ, et al. Among authors: goulet mt. Bioorg Med Chem Lett. 1999 Sep 6;9(17):2615-20. doi: 10.1016/s0960-894x(99)00446-1. Bioorg Med Chem Lett. 1999. PMID: 10498220

7

Investigation of the 4-O-alkylamine substituent of non-peptide quinolone GnRH receptor antagonists.

DeVita RJ, Goulet MT, Wyvratt MJ, Fisher MH, Lo JL, Yang YT, Cheng K, Smith RG. DeVita RJ, et al. Among authors: goulet mt. Bioorg Med Chem Lett. 1999 Sep 6;9(17):2621-4. doi: 10.1016/s0960-894x(99)00447-3. Bioorg Med Chem Lett. 1999. PMID: 10498221

8

Potent antagonists of gonadotropin releasing hormone receptors derived from quinolone-6-carboxamides.

Walsh TF, Toupence RB, Young JR, Huang SX, Ujjainwalla F, DeVita RJ, Goulet MT, Wyvratt MJ Jr, Fisher MH, Lo JL, Ren N, Yudkovitz JB, Yang YT, Cheng K, Smith RG. Walsh TF, et al. Among authors: goulet mt. Bioorg Med Chem Lett. 2000 Mar 6;10(5):443-7. doi: 10.1016/s0960-894x(00)00024-x. Bioorg Med Chem Lett. 2000. PMID: 10743944

9

Identification of Phe313 of the gonadotropin-releasing hormone (GnRH) receptor as a site critical for the binding of nonpeptide GnRH antagonists.

Cui J, Smith RG, Mount GR, Lo JL, Yu J, Walsh TF, Singh SB, DeVita RJ, Goulet MT, Schaeffer JM, Cheng K. Cui J, et al. Among authors: goulet mt. Mol Endocrinol. 2000 May;14(5):671-81. doi: 10.1210/mend.14.5.0464. Mol Endocrinol. 2000. PMID: 10809231

10

Quinolones as gonadotropin releasing hormone (GnRH) antagonists: simultaneous optimization of the C(3)-aryl and C(6)-substituents.

Young JR, Huang SX, Chen I, Walsh TF, DeVita RJ, Wyvratt MJ Jr, Goulet MT, Ren N, Lo J, Yang YT, Yudkovitz JB, Cheng K, Smith RG. Young JR, et al. Among authors: goulet mt. Bioorg Med Chem Lett. 2000 Aug 7;10(15):1723-7. doi: 10.1016/s0960-894x(00)00318-8. Bioorg Med Chem Lett. 2000. PMID: 10937733

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