Link A - Search Results

1

5'-Deoxy congeners of 9-(3-amido-3-deoxy-beta-D-xylofuranosyl)-N(6)-cyclopentyladenine: new adenosine A(1) receptor antagonists and inverse agonists.

Van Calenbergh S, Link A, Fujikawa S, de Ligt RA, Vanheusden V, Golisade A, Blaton NM, Rozenski J, IJzerman AP, Herdewijn P. Van Calenbergh S, et al. Among authors: link a. J Med Chem. 2002 Apr 25;45(9):1845-52. doi: 10.1021/jm0110439. J Med Chem. 2002. PMID: 11960496

2

Exploration of the effect of sterically demanding 3'-amido substitution of 3'-deoxyadenosines towards inhibition of cyclin-dependent kinase 1.

Van Calenbergh S, Link A, Kunick C, Herdewijn P. Van Calenbergh S, et al. Among authors: link a. Pharmazie. 1999 Oct;54(10):727-9. Pharmazie. 1999. PMID: 10563371

3

Polymer-assisted solution-phase synthesis of 2'-amido-2'-deoxyadenosine derivatives targeted at the NAD(+)-binding sites of parasite enzymes.

Golisade A, Bressi JC, Van Calenbergh S, Gelb MH, Link A. Golisade A, et al. Among authors: link a. J Comb Chem. 2000 Sep-Oct;2(5):537-44. doi: 10.1021/cc0000343. J Comb Chem. 2000. PMID: 11029179

4

Biotin labelling of amines by polymer-assisted solution-phase synthesis.

Golisade A, Herforth C, Wieking K, Kunick C, Link A. Golisade A, et al. Among authors: link a. Bioorg Med Chem Lett. 2001 Jul 9;11(13):1783-6. doi: 10.1016/s0960-894x(01)00296-7. Bioorg Med Chem Lett. 2001. PMID: 11425560

5

Neoceptor concept based on molecular complementarity in GPCRs: a mutant adenosine A(3) receptor with selectively enhanced affinity for amine-modified nucleosides.

Jacobson KA, Gao ZG, Chen A, Barak D, Kim SA, Lee K, Link A, Rompaey PV, van Calenbergh S, Liang BT. Jacobson KA, et al. Among authors: link a. J Med Chem. 2001 Nov 22;44(24):4125-36. doi: 10.1021/jm010232o. J Med Chem. 2001. PMID: 11708915 Free PMC article.

6

Improving an antitrypanosomal lead applying nucleophilic substitution on a safety catch linker.

Golisade A, Herforth C, Quirijnen L, Maes L, Link A. Golisade A, et al. Among authors: link a. Bioorg Med Chem. 2002 Jan;10(1):159-65. doi: 10.1016/s0968-0896(01)00253-x. Bioorg Med Chem. 2002. PMID: 11738617

7

Anti-malarial activity of N(6)-substituted adenosine derivatives. Part I.

Golisade A, Wiesner J, Herforth C, Jomaa H, Link A. Golisade A, et al. Among authors: link a. Bioorg Med Chem. 2002 Mar;10(3):769-77. doi: 10.1016/s0968-0896(01)00331-5. Bioorg Med Chem. 2002. PMID: 11814867

8

Antimalarial activity of n(6)-substituted adenosine derivatives (part 2).

Herforth C, Wiesner J, Franke S, Golisade A, Jomaa H, Link A. Herforth C, et al. Among authors: link a. J Comb Chem. 2002 Jul-Aug;4(4):302-14. doi: 10.1021/cc0100823. J Comb Chem. 2002. PMID: 12099848

9

Antimalarial activity of N(6)-substituted adenosine derivatives. Part 3.

Herforth C, Wiesner J, Heidler P, Sanderbrand S, Van Calenbergh S, Jomaa H, Link A. Herforth C, et al. Among authors: link a. Bioorg Med Chem. 2004 Feb 15;12(4):755-62. doi: 10.1016/j.bmc.2003.11.008. Bioorg Med Chem. 2004. PMID: 14759735

10

Synthesis of beta- and gamma-oxa isosteres of fosmidomycin and FR900098 as antimalarial candidates.

Haemers T, Wiesner J, Giessmann D, Verbrugghen T, Hillaert U, Ortmann R, Jomaa H, Link A, Schlitzer M, Van Calenbergh S. Haemers T, et al. Among authors: link a. Bioorg Med Chem. 2008 Mar 15;16(6):3361-71. doi: 10.1016/j.bmc.2007.12.001. Epub 2007 Dec 8. Bioorg Med Chem. 2008. PMID: 18158249

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