Jacobson KA - Search Results

1

Synthesis, biological properties, and molecular modeling investigation of the first potent, selective, and water-soluble human A(3) adenosine receptor antagonist.

Maconi A, Pastorin G, Da Ros T, Spalluto G, Gao ZG, Jacobson KA, Baraldi PG, Cacciari B, Varani K, Moro S, Borea PA. Maconi A, et al. Among authors: jacobson ka. J Med Chem. 2002 Aug 15;45(17):3579-82. doi: 10.1021/jm020974x. J Med Chem. 2002. PMID: 12166930 Free PMC article.

2

Synthesis and biological activity of N6-(p-sulfophenyl)alkyl and N6-sulfoalkyl derivatives of adenosine: water-soluble and peripherally selective adenosine agonists.

Jacobson KA, Nikodijevic O, Ji XD, Berkich DA, Eveleth D, Dean RL, Hiramatsu K, Kassell NF, van Galen PJ, Lee KS, et al. Jacobson KA, et al. J Med Chem. 1992 Oct 30;35(22):4143-9. doi: 10.1021/jm00100a020. J Med Chem. 1992. PMID: 1433217 Free PMC article.

3

Electrophilic derivatives of purines as irreversible inhibitors of A1 adenosine receptors.

Jacobson KA, Barone S, Kammula U, Stiles GL. Jacobson KA, et al. J Med Chem. 1989 May;32(5):1043-51. doi: 10.1021/jm00125a019. J Med Chem. 1989. PMID: 2709373 Free PMC article.

4

Sulfur-containing 1,3-dialkylxanthine derivatives as selective antagonists at A1-adenosine receptors.

Jacobson KA, Kiriasis L, Barone S, Bradbury BJ, Kammula U, Campagne JM, Secunda S, Daly JW, Neumeyer JL, Pfleiderer W. Jacobson KA, et al. J Med Chem. 1989 Aug;32(8):1873-9. doi: 10.1021/jm00128a031. J Med Chem. 1989. PMID: 2754711 Free PMC article.

5

Functionalized congeners of adenosine: preparation of analogues with high affinity for A1-adenosine receptors.

Jacobson KA, Kirk KL, Padgett WL, Daly JW. Jacobson KA, et al. J Med Chem. 1985 Sep;28(9):1341-6. doi: 10.1021/jm00147a039. J Med Chem. 1985. PMID: 2993623 Free PMC article.

6

Xanthine functionalized congeners as potent ligands at A2-adenosine receptors.

Jacobson KA, Ukena D, Padgett W, Daly JW, Kirk KL. Jacobson KA, et al. J Med Chem. 1987 Jan;30(1):211-4. doi: 10.1021/jm00384a037. J Med Chem. 1987. PMID: 3806597 Free PMC article.

7

Search for new purine- and ribose-modified adenosine analogues as selective agonists and antagonists at adenosine receptors.

Siddiqi SM, Jacobson KA, Esker JL, Olah ME, Ji XD, Melman N, Tiwari KN, Secrist JA 3rd, Schneller SW, Cristalli G, et al. Siddiqi SM, et al. Among authors: jacobson ka. J Med Chem. 1995 Mar 31;38(7):1174-88. doi: 10.1021/jm00007a014. J Med Chem. 1995. PMID: 7707320 Free PMC article.

8

Structure-activity relationships of 9-alkyladenine and ribose-modified adenosine derivatives at rat A3 adenosine receptors.

Jacobson KA, Siddiqi SM, Olah ME, Ji XD, Melman N, Bellamkonda K, Meshulam Y, Stiles GL, Kim HO. Jacobson KA, et al. J Med Chem. 1995 May 12;38(10):1720-35. doi: 10.1021/jm00010a017. J Med Chem. 1995. PMID: 7752196 Free PMC article.

9

Structure-activity relationships of 1,3-dialkylxanthine derivatives at rat A3 adenosine receptors.

Kim HO, Ji XD, Melman N, Olah ME, Stiles GL, Jacobson KA. Kim HO, et al. Among authors: jacobson ka. J Med Chem. 1994 Sep 30;37(20):3373-82. doi: 10.1021/jm00046a022. J Med Chem. 1994. PMID: 7932565 Free PMC article.

10

2-Substitution of N6-benzyladenosine-5'-uronamides enhances selectivity for A3 adenosine receptors.

Kim HO, Ji XD, Siddiqi SM, Olah ME, Stiles GL, Jacobson KA. Kim HO, et al. Among authors: jacobson ka. J Med Chem. 1994 Oct 14;37(21):3614-21. doi: 10.1021/jm00047a018. J Med Chem. 1994. PMID: 7932588 Free PMC article.

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