Bleasdale JE - Search Results

1

Modification of the N-terminus of peptidomimetic protein tyrosine phosphatase 1B (PTP1B) inhibitors: identification of analogues with cellular activity.

Larsen SD, Stevens FC, Lindberg TJ, Bodnar PM, O'Sullivan TJ, Schostarez HJ, Palazuk BJ, Bleasdale JE. Larsen SD, et al. Among authors: bleasdale je. Bioorg Med Chem Lett. 2003 Mar 10;13(5):971-5. doi: 10.1016/s0960-894x(02)01065-x. Bioorg Med Chem Lett. 2003. PMID: 12617932

2

Synthesis and biological activity of a novel class of small molecular weight peptidomimetic competitive inhibitors of protein tyrosine phosphatase 1B.

Larsen SD, Barf T, Liljebris C, May PD, Ogg D, O'Sullivan TJ, Palazuk BJ, Schostarez HJ, Stevens FC, Bleasdale JE. Larsen SD, et al. Among authors: bleasdale je. J Med Chem. 2002 Jan 31;45(3):598-622. doi: 10.1021/jm010393s. J Med Chem. 2002. PMID: 11806712

3

Investigation of potential bioisosteric replacements for the carboxyl groups of peptidomimetic inhibitors of protein tyrosine phosphatase 1B: identification of a tetrazole-containing inhibitor with cellular activity.

Liljebris C, Larsen SD, Ogg D, Palazuk BJ, Bleasdale JE. Liljebris C, et al. Among authors: bleasdale je. J Med Chem. 2002 Apr 25;45(9):1785-98. doi: 10.1021/jm011100y. J Med Chem. 2002. PMID: 11960490

4

Small molecule peptidomimetics containing a novel phosphotyrosine bioisostere inhibit protein tyrosine phosphatase 1B and augment insulin action.

Bleasdale JE, Ogg D, Palazuk BJ, Jacob CS, Swanson ML, Wang XY, Thompson DP, Conradi RA, Mathews WR, Laborde AL, Stuchly CW, Heijbel A, Bergdahl K, Bannow CA, Smith CW, Svensson C, Liljebris C, Schostarez HJ, May PD, Stevens FC, Larsen SD. Bleasdale JE, et al. Biochemistry. 2001 May 15;40(19):5642-54. doi: 10.1021/bi002865v. Biochemistry. 2001. PMID: 11341829

5

Analysis of in vitro interactions of protein tyrosine phosphatase 1B with insulin receptors.

Wang XY, Bergdahl K, Heijbel A, Liljebris C, Bleasdale JE. Wang XY, et al. Among authors: bleasdale je. Mol Cell Endocrinol. 2001 Feb 28;173(1-2):109-20. doi: 10.1016/s0303-7207(00)00402-0. Mol Cell Endocrinol. 2001. PMID: 11223182

6

Pioglitazone promotes insulin-induced activation of phosphoinositide 3-kinase in 3T3-L1 adipocytes by inhibiting a negative control mechanism.

Sizer KM, Smith CL, Jacob CS, Swanson ML, Bleasdale JE. Sizer KM, et al. Among authors: bleasdale je. Mol Cell Endocrinol. 1994 Jul;103(1-2):1-12. doi: 10.1016/0303-7207(94)90063-9. Mol Cell Endocrinol. 1994. PMID: 7525381

7

Pioglitazone promotes insulin-induced activation of phosphoinositide 3-kinase in 3T3-L1 adipocytes by inhibiting a negative control mechanism.

Sizer KM, Smith CL, Jacob CS, Swanson ML, Bleasdale JE. Sizer KM, et al. Among authors: bleasdale je. Mol Cell Endocrinol. 1994 Jun;102(1-2):119-29. doi: 10.1016/0303-7207(94)90105-8. Mol Cell Endocrinol. 1994. PMID: 7926264

8

Hepatic insulin resistance in KKA(y) mice and its amelioration by pioglitazone do not involve alterations in phospholipase C activity.

Bleasdale JE, Swanson ML. Bleasdale JE, et al. Biochim Biophys Acta. 1993 Jun 19;1181(3):240-8. doi: 10.1016/0925-4439(93)90027-x. Biochim Biophys Acta. 1993. PMID: 8391325

9

NPC 15669-modulated human polymorphonuclear neutrophil functional responsiveness: effects on receptor-coupled signal transduction.

Smith RJ, Justen JM, Bleasdale JE, Sly LM. Smith RJ, et al. Among authors: bleasdale je. Br J Pharmacol. 1995 Apr;114(8):1694-702. doi: 10.1111/j.1476-5381.1995.tb14959.x. Br J Pharmacol. 1995. PMID: 7599938 Free PMC article.

10

The aminosteroid U-73122 inhibits muscarinic receptor sequestration and phosphoinositide hydrolysis in SK-N-SH neuroblastoma cells. A role for Gp in receptor compartmentation.

Thompson AK, Mostafapour SP, Denlinger LC, Bleasdale JE, Fisher SK. Thompson AK, et al. Among authors: bleasdale je. J Biol Chem. 1991 Dec 15;266(35):23856-62. J Biol Chem. 1991. PMID: 1660886 Free article.

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