Primofiore G - Search Results

1

Benzodiazepine receptor affinity and interaction of some N-(indol-3-ylglyoxylyl)amine derivatives.

Bianucci AM, Da Settimo A, Da Settimo F, Primofiore G, Martini C, Giannaccini G, Lucacchini A. Bianucci AM, et al. Among authors: primofiore g. J Med Chem. 1992 Jun 12;35(12):2214-20. doi: 10.1021/jm00090a011. J Med Chem. 1992. PMID: 1319492

2

Novel, highly potent aldose reductase inhibitors: cyano(2-oxo-2,3-dihydroindol-3-yl)acetic acid derivatives.

Da Settimo F, Primofiore G, Da Settimo A, La Motta C, Simorini F, Novellino E, Greco G, Lavecchia A, Boldrini E. Da Settimo F, et al. Among authors: primofiore g. J Med Chem. 2003 Apr 10;46(8):1419-28. doi: 10.1021/jm030762f. J Med Chem. 2003. PMID: 12672241

3

N,N-dialkyl-2-phenylindol-3-ylglyoxylamides. A new class of potent and selective ligands at the peripheral benzodiazepine receptor.

Primofiore G, Da Settimo F, Taliani S, Simorini F, Patrizi MP, Novellino E, Greco G, Abignente E, Costa B, Chelli B, Martini C. Primofiore G, et al. J Med Chem. 2004 Mar 25;47(7):1852-5. doi: 10.1021/jm030973k. J Med Chem. 2004. PMID: 15027878 Free article.

4

High affinity central benzodiazepine receptor ligands: synthesis and biological evaluation of a series of phenyltriazolobenzotriazindione derivatives.

Primofiore G, Da Settimo F, Taliani S, Salerno S, Novellino E, Greco G, Cosimelli B, Besnard F, Costa B, Montali M, Martini C. Primofiore G, et al. J Med Chem. 2005 Apr 21;48(8):2936-43. doi: 10.1021/jm0408722. J Med Chem. 2005. PMID: 15828832

5

Novel, highly potent adenosine deaminase inhibitors containing the pyrazolo[3,4-d]pyrimidine ring system. Synthesis, structure-activity relationships, and molecular modeling studies.

Da Settimo F, Primofiore G, La Motta C, Taliani S, Simorini F, Marini AM, Mugnaini L, Lavecchia A, Novellino E, Tuscano D, Martini C. Da Settimo F, et al. Among authors: primofiore g. J Med Chem. 2005 Aug 11;48(16):5162-74. doi: 10.1021/jm050136d. J Med Chem. 2005. PMID: 16078836

6

Refinement of the benzodiazepine receptor site topology by structure-activity relationships of new N-(heteroarylmethyl)indol-3-ylglyoxylamides.

Primofiore G, Da Settimo F, Marini AM, Taliani S, La Motta C, Simorini F, Novellino E, Greco G, Cosimelli B, Ehlardo M, Sala A, Besnard F, Montali M, Martini C. Primofiore G, et al. J Med Chem. 2006 Apr 20;49(8):2489-95. doi: 10.1021/jm0511841. J Med Chem. 2006. PMID: 16610792

7

Novel N-substituted indol-3-ylglyoxylamides probing the LDi and L1/L2 lipophilic regions of the benzodiazepine receptor site in search for subtype-selective ligands.

Primofiore G, Taliani S, Da Settimo F, Marini AM, La Motta C, Simorini F, Patrizi MP, Sergianni V, Novellino E, Greco G, Cosimelli B, Calderone V, Montali M, Besnard F, Martini C. Primofiore G, et al. J Med Chem. 2007 Apr 5;50(7):1627-34. doi: 10.1021/jm0607707. Epub 2007 Mar 3. J Med Chem. 2007. PMID: 17335185

8

5-amino-2-phenyl[1,2,3]triazolo[1,2-a][1,2,4]benzotriazin-1-one: a versatile scaffold to obtain potent and selective A3 adenosine receptor antagonists.

Da Settimo F, Primofiore G, Taliani S, Marini AM, La Motta C, Simorini F, Salerno S, Sergianni V, Tuccinardi T, Martinelli A, Cosimelli B, Greco G, Novellino E, Ciampi O, Trincavelli ML, Martini C. Da Settimo F, et al. Among authors: primofiore g. J Med Chem. 2007 Nov 15;50(23):5676-84. doi: 10.1021/jm0708376. Epub 2007 Oct 10. J Med Chem. 2007. PMID: 17927167

9

Specific inhibition of benzodiazepine receptor binding by some N-(2-methyl or 1,2-dimethylindol-3-ylglyoxylyl)amino acid derivatives.

Primofiore G, Marini AM, Da Settimo F, Salvadori C, Martini C, Lucacchini A, Giannaccini G. Primofiore G, et al. Farmaco. 1990 Mar;45(3):341-51. Farmaco. 1990. PMID: 2166528

10

Specific inhibition of benzodiazepine receptor binding by some N-(indol-3-ylglyoxylyl)amino acid derivatives: stereoselective interactions.

Primofiore G, Marini AM, Da Settimo F, Martini C, Bardellini A, Giannaccini G, Lucacchini A. Primofiore G, et al. J Med Chem. 1989 Dec;32(12):2514-8. doi: 10.1021/jm00132a004. J Med Chem. 1989. PMID: 2555510

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