Tagari P - Search Results

1

(4-Piperidinylphenyl)aminoethyl amides as a novel class of non-covalent cathepsin K inhibitors.

Kim TS, Hague AB, Lee TI, Lian B, Tegley CM, Wang X, Burgess TL, Qian YX, Ross S, Tagari P, Lin CH, Mayeda C, Dao J, Jordan S, Mohr C, Cheetham J, Viswanadhan V, Tasker AS. Kim TS, et al. Among authors: tagari p. Bioorg Med Chem Lett. 2004 Jan 5;14(1):87-90. doi: 10.1016/j.bmcl.2003.10.009. Bioorg Med Chem Lett. 2004. PMID: 14684304

2

Discovery of novel hydroxy-thiazoles as HIF-alpha prolyl hydroxylase inhibitors: SAR, synthesis, and modeling evaluation.

Tegley CM, Viswanadhan VN, Biswas K, Frohn MJ, Peterkin TA, Chang C, Bürli RW, Dao JH, Veith H, Rogers N, Yoder SC, Biddlecome G, Tagari P, Allen JR, Hungate RW. Tegley CM, et al. Among authors: tagari p. Bioorg Med Chem Lett. 2008 Jul 15;18(14):3925-8. doi: 10.1016/j.bmcl.2008.06.031. Epub 2008 Jun 13. Bioorg Med Chem Lett. 2008. PMID: 18579373

3

Potent hFPRL1 (ALXR) agonists as potential anti-inflammatory agents.

Bürli RW, Xu H, Zou X, Muller K, Golden J, Frohn M, Adlam M, Plant MH, Wong M, McElvain M, Regal K, Viswanadhan VN, Tagari P, Hungate R. Bürli RW, et al. Among authors: tagari p. Bioorg Med Chem Lett. 2006 Jul 15;16(14):3713-8. doi: 10.1016/j.bmcl.2006.04.068. Epub 2006 May 11. Bioorg Med Chem Lett. 2006. PMID: 16697190

4

Kinetic characterization and identification of a novel inhibitor of hypoxia-inducible factor prolyl hydroxylase 2 using a time-resolved fluorescence resonance energy transfer-based assay technology.

Dao JH, Kurzeja RJ, Morachis JM, Veith H, Lewis J, Yu V, Tegley CM, Tagari P. Dao JH, et al. Among authors: tagari p. Anal Biochem. 2009 Jan 15;384(2):213-23. doi: 10.1016/j.ab.2008.09.052. Epub 2008 Oct 14. Anal Biochem. 2009. PMID: 18952043

5

Structure-guided Discovery of Dual-recognition Chemibodies.

Cheng AC, Doherty EM, Johnstone S, DiMauro EF, Dao J, Luthra A, Ye J, Tang J, Nixey T, Min X, Tagari P, Miranda LP, Wang Z. Cheng AC, et al. Among authors: tagari p. Sci Rep. 2018 May 15;8(1):7570. doi: 10.1038/s41598-018-25848-0. Sci Rep. 2018. PMID: 29765112 Free PMC article.

6

Substituted 2,2-bisaryl-bicycloheptanes as novel and potent inhibitors of 5-lipoxygenase activating protein.

Macdonald D, Brideau C, Chan CC, Falgueyret JP, Frenette R, Guay J, Hutchinson JH, Perrier H, Prasit P, Riendeau D, Tagari P, Thérien M, Young RN, Girard Y. Macdonald D, et al. Among authors: tagari p. Bioorg Med Chem Lett. 2008 Mar 15;18(6):2023-7. doi: 10.1016/j.bmcl.2008.01.105. Epub 2008 Feb 2. Bioorg Med Chem Lett. 2008. PMID: 18276139

7

New 'chemical probes' to examine the role of the hFPRL1 (or ALXR) receptor in inflammation.

Frohn M, Xu H, Zou X, Chang C, McElvaine M, Plant MH, Wong M, Tagari P, Hungate R, Bürli RW. Frohn M, et al. Among authors: tagari p. Bioorg Med Chem Lett. 2007 Dec 1;17(23):6633-7. doi: 10.1016/j.bmcl.2007.09.043. Epub 2007 Sep 15. Bioorg Med Chem Lett. 2007. PMID: 17920884

8

Substituted coumarins as potent 5-lipoxygenase inhibitors.

Grimm EL, Brideau C, Chauret N, Chan CC, Delorme D, Ducharme Y, Ethier D, Falgueyret JP, Friesen RW, Guay J, Hamel P, Riendeau D, Soucy-Breau C, Tagari P, Girard Y. Grimm EL, et al. Among authors: tagari p. Bioorg Med Chem Lett. 2006 May 1;16(9):2528-31. doi: 10.1016/j.bmcl.2006.01.085. Epub 2006 Feb 7. Bioorg Med Chem Lett. 2006. PMID: 16464579

9

Quinolines as potent 5-lipoxygenase inhibitors: synthesis and biological profile of L-746,530.

Dubé D, Blouin M, Brideau C, Chan CC, Desmarais S, Ethier D, Falgueyret JP, Friesen RW, Girard M, Girard Y, Guay J, Riendeau D, Tagari P, Young RN. Dubé D, et al. Among authors: tagari p. Bioorg Med Chem Lett. 1998 May 19;8(10):1255-60. doi: 10.1016/s0960-894x(98)00201-7. Bioorg Med Chem Lett. 1998. PMID: 9871745

10

Substituted indoles as potent and orally active 5-lipoxygenase activating protein (FLAP) inhibitors.

Frenette R, Hutchinson JH, Léger S, Thérien M, Brideau C, Chan CC, Charleson S, Ethier D, Guay J, Jones TR, McAuliffe M, Piechuta H, Riendeau D, Tagari P, Girard Y. Frenette R, et al. Among authors: tagari p. Bioorg Med Chem Lett. 1999 Aug 16;9(16):2391-6. doi: 10.1016/s0960-894x(99)00399-6. Bioorg Med Chem Lett. 1999. PMID: 10476875

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

71 results

Search Page

Filters