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Page 1
Roles of conformational and positional adaptability in structure-based design of TMC125-R165335 (etravirine) and related non-nucleoside reverse transcriptase inhibitors that are highly potent and effective against wild-type and drug-resistant HIV-1 variants.
Das K, Clark AD Jr, Lewi PJ, Heeres J, De Jonge MR, Koymans LM, Vinkers HM, Daeyaert F, Ludovici DW, Kukla MJ, De Corte B, Kavash RW, Ho CY, Ye H, Lichtenstein MA, Andries K, Pauwels R, De Béthune MP, Boyer PL, Clark P, Hughes SH, Janssen PA, Arnold E. Das K, et al. Among authors: de jonge mr, de bethune mp, de corte b. J Med Chem. 2004 May 6;47(10):2550-60. doi: 10.1021/jm030558s. J Med Chem. 2004. PMID: 15115397
Evolution of anti-HIV drug candidates. Part 2: Diaryltriazine (DATA) analogues.
Ludovici DW, Kavash RW, Kukla MJ, Ho CY, Ye H, De Corte BL, Andries K, de Béthune MP, Azijn H, Pauwels R, Moereels HE, Heeres J, Koymans LM, de Jonge MR, Van Aken KJ, Daeyaert FF, Lewi PJ, Das K, Arnold E, Janssen PA. Ludovici DW, et al. Among authors: de bethune mp, de jonge mr, de corte bl. Bioorg Med Chem Lett. 2001 Sep 3;11(17):2229-34. doi: 10.1016/s0960-894x(01)00411-5. Bioorg Med Chem Lett. 2001. PMID: 11527704
Evolution of anti-HIV drug candidates. Part 3: Diarylpyrimidine (DAPY) analogues.
Ludovici DW, De Corte BL, Kukla MJ, Ye H, Ho CY, Lichtenstein MA, Kavash RW, Andries K, de Béthune MP, Azijn H, Pauwels R, Lewi PJ, Heeres J, Koymans LM, de Jonge MR, Van Aken KJ, Daeyaert FF, Das K, Arnold E, Janssen PA. Ludovici DW, et al. Among authors: de bethune mp, de jonge mr, de corte bl. Bioorg Med Chem Lett. 2001 Sep 3;11(17):2235-9. doi: 10.1016/s0960-894x(01)00412-7. Bioorg Med Chem Lett. 2001. PMID: 11527705
On the detection of multiple-binding modes of ligands to proteins, from biological, structural, and modeling data.
Lewi PJ, de Jonge M, Daeyaert F, Koymans L, Vinkers M, Heeres J, Janssen PA, Arnold E, Das K, Clark AD Jr, Hughes SH, Boyer PL, de Béthune MP, Pauwels R, Andries K, Kukla M, Ludovici D, De Corte B, Kavash R, Ho C. Lewi PJ, et al. Among authors: de bethune mp, de jonge m, de corte b. J Comput Aided Mol Des. 2003 Feb-Apr;17(2-4):129-34. doi: 10.1023/a:1025313705564. J Comput Aided Mol Des. 2003. PMID: 13677481
TMC125, a novel next-generation nonnucleoside reverse transcriptase inhibitor active against nonnucleoside reverse transcriptase inhibitor-resistant human immunodeficiency virus type 1.
Andries K, Azijn H, Thielemans T, Ludovici D, Kukla M, Heeres J, Janssen P, De Corte B, Vingerhoets J, Pauwels R, de Béthune MP. Andries K, et al. Among authors: de bethune mp, de corte b. Antimicrob Agents Chemother. 2004 Dec;48(12):4680-6. doi: 10.1128/AAC.48.12.4680-4686.2004. Antimicrob Agents Chemother. 2004. PMID: 15561844 Free PMC article.
Novel triazole based inhibitors of Ras farnesyl transferase.
Saha AK, Liu L, Simoneaux R, DeCorte B, Meyer C, Skrzat S, Breslin HJ, Kukla MJ, End DW. Saha AK, et al. Bioorg Med Chem Lett. 2005 Dec 15;15(24):5407-11. doi: 10.1016/j.bmcl.2005.09.007. Epub 2005 Oct 10. Bioorg Med Chem Lett. 2005. PMID: 16216509
33 results