Smits G - Search Results

1

Piperazine derivatives of [1,2,4]triazolo[1,5-a][1,3,5]triazine as potent and selective adenosine A2a receptor antagonists.

Vu CB, Peng B, Kumaravel G, Smits G, Jin X, Phadke D, Engber T, Huang C, Reilly J, Tam S, Grant D, Hetu G, Chen L, Zhang J, Petter RC. Vu CB, et al. Among authors: smits g. J Med Chem. 2004 Aug 12;47(17):4291-9. doi: 10.1021/jm0498405. J Med Chem. 2004. PMID: 15294001

2

Norbornyllactone-substituted xanthines as adenosine A(1) receptor antagonists.

Kiesman WF, Zhao J, Conlon PR, Petter RC, Jin X, Smits G, Lutterodt F, Sullivan GW, Linden J. Kiesman WF, et al. Among authors: smits g. Bioorg Med Chem. 2006 Jun 1;14(11):3654-61. doi: 10.1016/j.bmc.2006.01.021. Epub 2006 Feb 2. Bioorg Med Chem. 2006. PMID: 16458010

3

Potent and orally bioavailable 8-bicyclo[2.2.2]octylxanthines as adenosine A1 receptor antagonists.

Kiesman WF, Zhao J, Conlon PR, Dowling JE, Petter RC, Lutterodt F, Jin X, Smits G, Fure M, Jayaraj A, Kim J, Sullivan G, Linden J. Kiesman WF, et al. Among authors: smits g. J Med Chem. 2006 Nov 30;49(24):7119-31. doi: 10.1021/jm0605381. J Med Chem. 2006. PMID: 17125264

4

Tricyclic imidazoline derivatives as potent and selective adenosine A1 receptor antagonists.

Vu CB, Kiesman WF, Conlon PR, Lin KC, Tam M, Petter RC, Smits G, Lutterodt F, Jin X, Chen L, Zhang J. Vu CB, et al. Among authors: smits g. J Med Chem. 2006 Nov 30;49(24):7132-9. doi: 10.1021/jm060539t. J Med Chem. 2006. PMID: 17125265

5

Novel diamino derivatives of [1,2,4]triazolo[1,5-a][1,3,5]triazine as potent and selective adenosine A2a receptor antagonists.

Vu CB, Pan D, Peng B, Kumaravel G, Smits G, Jin X, Phadke D, Engber T, Huang C, Reilly J, Tam S, Grant D, Hetu G, Petter RC. Vu CB, et al. Among authors: smits g. J Med Chem. 2005 Mar 24;48(6):2009-18. doi: 10.1021/jm0498396. J Med Chem. 2005. PMID: 15771443

6

Synthesis and structure-activity relationships of nonpeptide, potent triazolone-based angiotensin II receptor antagonists.

Huang HC, Reitz DB, Chamberlain TS, Olins GM, Corpus VM, McMahon EG, Palomo MA, Koepke JP, Smits GJ, McGraw DE, et al. Huang HC, et al. Among authors: smits gj. J Med Chem. 1993 Jul 23;36(15):2172-81. doi: 10.1021/jm00067a015. J Med Chem. 1993. PMID: 8340920

7

Nonpeptide angiotensin II antagonists: N-phenyl-1H-pyrrole derivatives are angiotensin II receptor antagonists.

Bovy PR, Reitz DB, Collins JT, Chamberlain TS, Olins GM, Corpus VM, McMahon EG, Palomo MA, Koepke JP, Smits GJ, et al. Bovy PR, et al. Among authors: smits gj. J Med Chem. 1993 Jan 8;36(1):101-10. doi: 10.1021/jm00053a013. J Med Chem. 1993. PMID: 8421274

8

Comparison of three different A1 adenosine receptor antagonists on infarct size and multiple cycle ischemic preconditioning in anesthetized dogs.

Auchampach JA, Jin X, Moore J, Wan TC, Kreckler LM, Ge ZD, Narayanan J, Whalley E, Kiesman W, Ticho B, Smits G, Gross GJ. Auchampach JA, et al. Among authors: smits g. J Pharmacol Exp Ther. 2004 Mar;308(3):846-56. doi: 10.1124/jpet.103.057943. Epub 2003 Nov 21. J Pharmacol Exp Ther. 2004. PMID: 14634049

9

Dual A1/A2B Receptor Blockade Improves Cardiac and Renal Outcomes in a Rat Model of Heart Failure with Preserved Ejection Fraction.

Tofovic SP, Salah EM, Smits GJ, Whalley ET, Ticho B, Deykin A, Jackson EK. Tofovic SP, et al. J Pharmacol Exp Ther. 2016 Feb;356(2):333-40. doi: 10.1124/jpet.115.228841. Epub 2015 Nov 19. J Pharmacol Exp Ther. 2016. PMID: 26585572 Free PMC article.

10

Structure-activity relationships for the carboxy-terminus truncated analogues of angiotension II, a new class of angiotensin II antagonists.

Bovy PR, O'Neal JM, Olins GM, Patton DR, McMahon EG, Palomo M, Koepke JP, Salles KS, Trapani AJ, Smits GJ, et al. Bovy PR, et al. Among authors: smits gj. J Med Chem. 1990 May;33(5):1477-82. doi: 10.1021/jm00167a030. J Med Chem. 1990. PMID: 2329570

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