Leonardi A - Search Results

1

Design, synthesis, and biological evaluation of prazosin-related derivatives as multipotent compounds.

Antonello A, Hrelia P, Leonardi A, Marucci G, Rosini M, Tarozzi A, Tumiatti V, Melchiorre C. Antonello A, et al. Among authors: leonardi a. J Med Chem. 2005 Jan 13;48(1):28-31. doi: 10.1021/jm049153d. J Med Chem. 2005. PMID: 15633998

2

Structure-activity relationships in 1,4-benzodioxan-related compounds. 7. Selectivity of 4-phenylchroman analogues for alpha(1)-adrenoreceptor subtypes.

Quaglia W, Pigini M, Piergentili A, Giannella M, Gentili F, Marucci G, Carrieri A, Carotti A, Poggesi E, Leonardi A, Melchiorre C. Quaglia W, et al. Among authors: leonardi a. J Med Chem. 2002 Apr 11;45(8):1633-43. doi: 10.1021/jm011066n. J Med Chem. 2002. PMID: 11931617

3

Rosini M, Antonello A, Cavalli A, Bolognesi ML, Minarini A, Marucci G, Poggesi E, Leonardi A, Melchiorre C. Rosini M, et al. Among authors: leonardi a. J Med Chem. 2003 Nov 6;46(23):4895-903. doi: 10.1021/jm030952q. J Med Chem. 2003. PMID: 14584940

4

Synthesis and alpha(1)-adrenoceptor antagonist activity of derivatives and isosters of the furan portion of (+)-cyclazosin.

Sagratini G, Angeli P, Buccioni M, Gulini U, Marucci G, Melchiorre C, Leonardi A, Poggesi E, Giardinà D. Sagratini G, et al. Among authors: leonardi a. Bioorg Med Chem. 2007 Mar 15;15(6):2334-45. doi: 10.1016/j.bmc.2007.01.028. Epub 2007 Jan 19. Bioorg Med Chem. 2007. PMID: 17276073

5

Design, synthesis, and biological activity of prazosin-related antagonists. Role of the piperazine and furan units of prazosin on the selectivity for alpha1-adrenoreceptor subtypes.

Bolognesi ML, Budriesi R, Chiarini A, Poggesi E, Leonardi A, Melchiorre C. Bolognesi ML, et al. Among authors: leonardi a. J Med Chem. 1998 Nov 19;41(24):4844-53. doi: 10.1021/jm9810654. J Med Chem. 1998. PMID: 9822553

6

Search for alpha 1-adrenoceptor subtypes selective antagonists: design, synthesis and biological activity of cystazosin, an alpha 1D-adrenoceptor antagonist.

Minarini A, Budriesi R, Chiarini A, Leonardi A, Melchiorre C. Minarini A, et al. Among authors: leonardi a. Bioorg Med Chem Lett. 1998 Jun 2;8(11):1353-8. doi: 10.1016/s0960-894x(98)00217-0. Bioorg Med Chem Lett. 1998. PMID: 9871765

7

Structure-activity relationships in 1,4-benzodioxan-related compounds. 6. Role of the dioxane unit on selectivity for alpha(1)-adrenoreceptor subtypes.

Quaglia W, Pigini M, Piergentili A, Giannella M, Marucci G, Poggesi E, Leonardi A, Melchiorre C. Quaglia W, et al. Among authors: leonardi a. J Med Chem. 1999 Jul 29;42(15):2961-8. doi: 10.1021/jm9910324. J Med Chem. 1999. PMID: 10425105

8

Bolognesi ML, Budriesi R, Cavalli A, Chiarini A, Gotti R, Leonardi A, Minarini A, Poggesi E, Recanatini M, Rosini M, Tumiatti V, Melchiorre C. Bolognesi ML, et al. Among authors: leonardi a. J Med Chem. 1999 Oct 7;42(20):4214-24. doi: 10.1021/jm991065j. J Med Chem. 1999. PMID: 10514291

9

1,3-dioxolane-based ligands as a novel class of alpha1-adrenoceptor antagonists.

Brasili L, Sorbi C, Franchini S, Manicardi M, Angeli P, Marucci G, Leonardi A, Poggesi E. Brasili L, et al. Among authors: leonardi a. J Med Chem. 2003 Apr 10;46(8):1504-11. doi: 10.1021/jm021078o. J Med Chem. 2003. PMID: 12672251

10

Synthesis, absolute configuration, and biological profile of the enantiomers of trans-[2-(2,6-dimethoxyphenoxy)ethyl] [(3-p-tolyl-2,3-dihydro-1,4-benzodioxin-2-yl)methyl]amine (mephendioxan), a potent competitive alpha 1A-adrenoreceptor antagonist.

Quaglia W, Pigini M, Tayebati SK, Piergentili A, Giannella M, Leonardi A, Taddei C, Melchiorre C. Quaglia W, et al. Among authors: leonardi a. J Med Chem. 1996 May 24;39(11):2253-8. doi: 10.1021/jm960069a. J Med Chem. 1996. PMID: 8667368

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