Yager KM - Search Results

1

Structure-based design, synthesis, and study of potent inhibitors of beta-ketoacyl-acyl carrier protein synthase III as potential antimicrobial agents.

Nie Z, Perretta C, Lu J, Su Y, Margosiak S, Gajiwala KS, Cortez J, Nikulin V, Yager KM, Appelt K, Chu S. Nie Z, et al. Among authors: yager km. J Med Chem. 2005 Mar 10;48(5):1596-609. doi: 10.1021/jm049141s. J Med Chem. 2005. PMID: 15743201

2

Structure-based design, synthesis, and antimicrobial activity of indazole-derived SAH/MTA nucleosidase inhibitors.

Li X, Chu S, Feher VA, Khalili M, Nie Z, Margosiak S, Nikulin V, Levin J, Sprankle KG, Tedder ME, Almassy R, Appelt K, Yager KM. Li X, et al. Among authors: yager km. J Med Chem. 2003 Dec 18;46(26):5663-73. doi: 10.1021/jm0302039. J Med Chem. 2003. PMID: 14667220

3

Structure-based design, synthesis, and antimicrobial activity of purine derived SAH/MTA nucleosidase inhibitors.

Tedder ME, Nie Z, Margosiak S, Chu S, Feher VA, Almassy R, Appelt K, Yager KM. Tedder ME, et al. Among authors: yager km. Bioorg Med Chem Lett. 2004 Jun 21;14(12):3165-8. doi: 10.1016/j.bmcl.2004.04.006. Bioorg Med Chem Lett. 2004. PMID: 15149667

4

Structure-based design, synthesis, and study of pyrazolo[1,5-a][1,3,5]triazine derivatives as potent inhibitors of protein kinase CK2.

Nie Z, Perretta C, Erickson P, Margosiak S, Almassy R, Lu J, Averill A, Yager KM, Chu S. Nie Z, et al. Among authors: yager km. Bioorg Med Chem Lett. 2007 Aug 1;17(15):4191-5. doi: 10.1016/j.bmcl.2007.05.041. Epub 2007 May 18. Bioorg Med Chem Lett. 2007. PMID: 17540560

5

Novel Mps1 kinase inhibitors: from purine to pyrrolopyrimidine and quinazoline leads.

Bursavich MG, Dastrup D, Shenderovich M, Yager KM, Cimbora DM, Williams B, Kumar DV. Bursavich MG, et al. Among authors: yager km. Bioorg Med Chem Lett. 2013 Dec 15;23(24):6829-33. doi: 10.1016/j.bmcl.2013.10.008. Epub 2013 Oct 11. Bioorg Med Chem Lett. 2013. PMID: 24183538

6

Triterpene based compounds with potent anti-maturation activity against HIV-1.

Gerrish D, Kim IC, Kumar DV, Austin H, Garrus JE, Baichwal V, Saunders M, McKinnon RS, Anderson MB, Carlson R, Arranz-Plaza E, Yager KM. Gerrish D, et al. Among authors: yager km. Bioorg Med Chem Lett. 2008 Dec 15;18(24):6377-80. doi: 10.1016/j.bmcl.2008.10.098. Epub 2008 Oct 25. Bioorg Med Chem Lett. 2008. PMID: 18996008

7

Lead optimization of purine based orally bioavailable Mps1 (TTK) inhibitors.

Vijay Kumar D, Hoarau C, Bursavich M, Slattum P, Gerrish D, Yager K, Saunders M, Shenderovich M, Roth BL, McKinnon R, Chan A, Cimbora DM, Bradford C, Reeves L, Patton S, Papac DI, Williams BL, Carlson RO. Vijay Kumar D, et al. Bioorg Med Chem Lett. 2012 Jul 1;22(13):4377-85. doi: 10.1016/j.bmcl.2012.04.131. Epub 2012 May 5. Bioorg Med Chem Lett. 2012. PMID: 22632936

8

Discovery of (2S)-1-[4-(2-{6-amino-8-[(6-bromo-1,3-benzodioxol-5-yl)sulfanyl]-9H-purin-9-yl}ethyl)piperidin-1-yl]-2-hydroxypropan-1-one (MPC-3100), a purine-based Hsp90 inhibitor.

Kim SH, Bajji A, Tangallapally R, Markovitz B, Trovato R, Shenderovich M, Baichwal V, Bartel P, Cimbora D, McKinnon R, Robinson R, Papac D, Wettstein D, Carlson R, Yager KM. Kim SH, et al. Among authors: yager km. J Med Chem. 2012 Sep 13;55(17):7480-501. doi: 10.1021/jm3004619. Epub 2012 Aug 31. J Med Chem. 2012. PMID: 22913511

9

Discovery of an L-alanine ester prodrug of the Hsp90 inhibitor, MPC-3100.

Kim SH, Tangallapally R, Kim IC, Trovato R, Parker D, Patton JS, Reeves L, Bradford C, Wettstein D, Baichwal V, Papac D, Bajji A, Carlson R, Yager KM. Kim SH, et al. Among authors: yager km. Bioorg Med Chem Lett. 2015 Nov 15;25(22):5254-7. doi: 10.1016/j.bmcl.2015.09.053. Epub 2015 Sep 28. Bioorg Med Chem Lett. 2015. PMID: 26483201

10

Cell cycle progression score is a marker for five-year lung cancer-specific mortality risk in patients with resected stage I lung adenocarcinoma.

Eguchi T, Kadota K, Chaft J, Evans B, Kidd J, Tan KS, Dycoco J, Kolquist K, Davis T, Hamilton SA, Yager K, Jones JT, Travis WD, Jones DR, Hartman AR, Adusumilli PS. Eguchi T, et al. Oncotarget. 2016 Jun 7;7(23):35241-56. doi: 10.18632/oncotarget.9129. Oncotarget. 2016. PMID: 27153551 Free PMC article.

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