Golas JM - Search Results

1

Further studies on ethenyl and ethynyl-4-phenylamino-3-quinolinecarbonitriles: identification of a subnanomolar Src kinase inhibitor.

Barrios Sosa AC, Boschelli DH, Wu B, Wang Y, Golas JM. Barrios Sosa AC, et al. Among authors: golas jm. Bioorg Med Chem Lett. 2005 Mar 15;15(6):1743-7. doi: 10.1016/j.bmcl.2005.01.004. Bioorg Med Chem Lett. 2005. PMID: 15745832

2

4-Anilino-7,8-dialkoxybenzo[g]quinoline-3-carbonitriles as potent Src kinase inhibitors.

Berger DM, Dutia M, Birnberg G, Powell D, Boschelli DH, Wang YD, Ravi M, Yaczko D, Golas J, Lucas J, Boschelli F. Berger DM, et al. J Med Chem. 2005 Sep 22;48(19):5909-20. doi: 10.1021/jm050512u. J Med Chem. 2005. PMID: 16161995

3

Optimization of 7-alkene-3-quinolinecarbonitriles as Src kinase inhibitors.

Boschelli DH, Wang D, Wang Y, Wu B, Honores EE, Barrios Sosa AC, Chaudhary I, Golas J, Lucas J, Boschelli F. Boschelli DH, et al. Bioorg Med Chem Lett. 2010 May 1;20(9):2924-7. doi: 10.1016/j.bmcl.2010.03.025. Epub 2010 Mar 7. Bioorg Med Chem Lett. 2010. PMID: 20363128

4

Inhibition of Src kinase activity by 4-anilino-5,10-dihydro-pyrimido[4,5-b]quinolines.

Boschelli DH, Powell D, Golas JM, Boschelli F. Boschelli DH, et al. Among authors: golas jm. Bioorg Med Chem Lett. 2003 Sep 15;13(18):2977-80. doi: 10.1016/s0960-894x(03)00628-0. Bioorg Med Chem Lett. 2003. PMID: 12941315

5

Investigation of the effect of varying the 4-anilino and 7-alkoxy groups of 3-quinolinecarbonitriles on the inhibition of Src kinase activity.

Boschelli DH, Ye F, Wu B, Wang YD, Barrios Sosa AC, Yaczko D, Powell D, Golas JM, Lucas J, Boschelli F. Boschelli DH, et al. Among authors: golas jm. Bioorg Med Chem Lett. 2003 Nov 3;13(21):3797-800. doi: 10.1016/j.bmcl.2003.07.001. Bioorg Med Chem Lett. 2003. PMID: 14552782

6

7-Alkoxy-4-phenylamino-3-quinolinecar-bonitriles as dual inhibitors of Src and Abl kinases.

Boschelli DH, Wang YD, Johnson S, Wu B, Ye F, Barrios Sosa AC, Golas JM, Boschelli F. Boschelli DH, et al. Among authors: golas jm. J Med Chem. 2004 Mar 25;47(7):1599-601. doi: 10.1021/jm0499458. J Med Chem. 2004. PMID: 15027848

7

Synthesis and inhibition of Src kinase activity by 7-ethenyl and 7-ethynyl-4-anilino-3-quinolinecarbonitriles.

Barrios Sosa AC, Boschelli DH, Ye F, Golas JM, Boschelli F. Barrios Sosa AC, et al. Among authors: golas jm. Bioorg Med Chem Lett. 2004 May 3;14(9):2155-8. doi: 10.1016/j.bmcl.2004.02.035. Bioorg Med Chem Lett. 2004. PMID: 15080999

8

Identification of 7-phenylaminothieno- [3,2-b]pyridine-6-carbonitriles as a new class of Src kinase inhibitors.

Boschelli DH, Wu B, Barrios Sosa AC, Durutlic H, Ye F, Raifeld Y, Golas JM, Boschelli F. Boschelli DH, et al. Among authors: golas jm. J Med Chem. 2004 Dec 30;47(27):6666-8. doi: 10.1021/jm049237m. J Med Chem. 2004. PMID: 15615514

9

Synthesis and Src kinase inhibitory activity of 2-phenyl- and 2-thienyl-7-phenylaminothieno[3,2-b]pyridine-6-carbonitriles.

Boschelli DH, Wu B, Barrios Sosa AC, Durutlic H, Chen JJ, Wang Y, Golas JM, Lucas J, Boschelli F. Boschelli DH, et al. Among authors: golas jm. J Med Chem. 2005 Jun 2;48(11):3891-902. doi: 10.1021/jm050175p. J Med Chem. 2005. PMID: 15916442

10

Inhibition of Src kinase activity by 7-[(2,4-dichloro-5-methoxyphenyl)amino]-2-heteroaryl-thieno[3,2-b]pyridine-6-carbonitriles.

Boschelli DH, Wu B, Barrios Sosa AC, Chen JJ, Golas JM, Boschelli F. Boschelli DH, et al. Among authors: golas jm. Bioorg Med Chem Lett. 2005 Nov 1;15(21):4681-4. doi: 10.1016/j.bmcl.2005.07.061. Bioorg Med Chem Lett. 2005. PMID: 16125383

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