Kiso Y - Search Results

1

No auxiliary, no byproduct strategy for water-soluble prodrugs of taxoids: scope and limitation of O-N intramolecular acyl and acyloxy migration reactions.

Skwarczynski M, Sohma Y, Noguchi M, Kimura M, Hayashi Y, Hamada Y, Kimura T, Kiso Y. Skwarczynski M, et al. Among authors: kiso y. J Med Chem. 2005 Apr 7;48(7):2655-66. doi: 10.1021/jm049344g. J Med Chem. 2005. PMID: 15801856

2

New water-soluble prodrugs of HIV protease inhibitors based on O-->N intramolecular acyl migration.

Hamada Y, Ohtake J, Sohma Y, Kimura T, Hayashi Y, Kiso Y. Hamada Y, et al. Among authors: kiso y. Bioorg Med Chem. 2002 Dec;10(12):4155-67. doi: 10.1016/s0968-0896(02)00322-x. Bioorg Med Chem. 2002. PMID: 12413869

3

An expedient synthesis of N(alpha)-protected-L-tetrahydrofuranylglycine and its application in the synthesis of novel substrate based inhibitors of HIV-1 protease.

Rajesh S, Ami E, Kotake T, Kimura T, Hayashi Y, Kiso Y. Rajesh S, et al. Among authors: kiso y. Bioorg Med Chem Lett. 2002 Dec 16;12(24):3615-7. doi: 10.1016/s0960-894x(02)00781-3. Bioorg Med Chem Lett. 2002. PMID: 12443788

4

Design and synthesis of pseudo-symmetric HIV protease inhibitors containing a novel hydroxymethylcarbonyl (HMC)-hydrazide isostere.

Hidaka K, Kimura T, Hayashi Y, McDaniel KF, Dekhtyar T, Colletti L, Kiso Y. Hidaka K, et al. Among authors: kiso y. Bioorg Med Chem Lett. 2003 Jan 6;13(1):93-6. doi: 10.1016/s0960-894x(02)00848-x. Bioorg Med Chem Lett. 2003. PMID: 12467624

5

Effect of the acyl groups on O-->N acyl migration in the water-soluble prodrugs of HIV-1 protease inhibitor.

Hamada Y, Matsumoto H, Kimura T, Hayashi Y, Kiso Y. Hamada Y, et al. Among authors: kiso y. Bioorg Med Chem Lett. 2003 Aug 18;13(16):2727-30. doi: 10.1016/s0960-894x(03)00576-6. Bioorg Med Chem Lett. 2003. PMID: 12873502

6

A novel approach of water-soluble paclitaxel prodrug with no auxiliary and no byproduct: design and synthesis of isotaxel.

Hayashi Y, Skwarczynski M, Hamada Y, Sohma Y, Kimura T, Kiso Y. Hayashi Y, et al. Among authors: kiso y. J Med Chem. 2003 Aug 28;46(18):3782-4. doi: 10.1021/jm034112n. J Med Chem. 2003. PMID: 12930140

7

Development of water-soluble prodrugs of the HIV-1 protease inhibitor KNI-727: importance of the conversion time for higher gastrointestinal absorption of prodrugs based on spontaneous chemical cleavage.

Sohma Y, Hayashi Y, Ito T, Matsumoto H, Kimura T, Kiso Y. Sohma Y, et al. Among authors: kiso y. J Med Chem. 2003 Sep 11;46(19):4124-35. doi: 10.1021/jm030009m. J Med Chem. 2003. PMID: 12954064

8

O-N intramolecular acyl migration strategy in water-soluble prodrugs of taxoids.

Skwarczynski M, Sohma Y, Kimura M, Hayashi Y, Kimura T, Kiso Y. Skwarczynski M, et al. Among authors: kiso y. Bioorg Med Chem Lett. 2003 Dec 15;13(24):4441-4. doi: 10.1016/j.bmcl.2003.09.020. Bioorg Med Chem Lett. 2003. PMID: 14643342

9

Water-soluble prodrugs of dipeptide HIV protease inhibitors based on O-->N intramolecular acyl migration: Design, synthesis and kinetic study.

Hamada Y, Matsumoto H, Yamaguchi S, Kimura T, Hayashi Y, Kiso Y. Hamada Y, et al. Among authors: kiso y. Bioorg Med Chem. 2004 Jan 2;12(1):159-70. doi: 10.1016/j.bmc.2003.10.026. Bioorg Med Chem. 2004. PMID: 14697781

10

Novel and efficient synthesis of difficult sequence-containing peptides through O-N intramolecular acyl migration reaction of O-acyl isopeptides.

Sohma Y, Sasaki M, Hayashi Y, Kimura T, Kiso Y. Sohma Y, et al. Among authors: kiso y. Chem Commun (Camb). 2004 Jan 7;(1):124-5. doi: 10.1039/b312129a. Epub 2003 Nov 21. Chem Commun (Camb). 2004. PMID: 14737363

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