Comparative potencies of CGP 47654A and CGP 46165A as GABA(B) receptor antagonists in rat brain.
Ong J, Kerr DI, Froestl W.
Ong J, et al. Among authors: froestl w.
Eur J Pharmacol. 1999 Jun 25;374(3):351-4. doi: 10.1016/s0014-2999(99)00377-5.
Eur J Pharmacol. 1999.
PMID: 10422779
Although relatively potent on GABAB heteroreceptors studied here, CGP 47654A and CGP 46165A were 5 and 50 times weaker, respectively, as GABAB autoreceptor antagonists [Froestl, W., Mickel, S.J., Von Sprecher, G., Diel, P.J., Hall, R.G., Maier, L., Strub, D., Melill …
Although relatively potent on GABAB heteroreceptors studied here, CGP 47654A and CGP 46165A were 5 and 50 times weaker, respectively, as GAB …