Baell JB - Search Results

1

Discovery of 2-iminobenzimidazoles as a new class of trypanothione reductase inhibitor by high-throughput screening.

Holloway GA, Baell JB, Fairlamb AH, Novello PM, Parisot JP, Richardson J, Watson KG, Street IP. Holloway GA, et al. Among authors: baell jb. Bioorg Med Chem Lett. 2007 Mar 1;17(5):1422-7. doi: 10.1016/j.bmcl.2006.11.090. Epub 2006 Dec 3. Bioorg Med Chem Lett. 2007. PMID: 17194585 Free PMC article.

2

Khellinone derivatives as blockers of the voltage-gated potassium channel Kv1.3: synthesis and immunosuppressive activity.

Baell JB, Gable RW, Harvey AJ, Toovey N, Herzog T, Hänsel W, Wulff H. Baell JB, et al. J Med Chem. 2004 Apr 22;47(9):2326-36. doi: 10.1021/jm030523s. J Med Chem. 2004. PMID: 15084131

3

A three-residue, continuous binding epitope peptidomimetic of ShK toxin as a Kv1.3 inhibitor.

Harvey AJ, Gable RW, Baell JB. Harvey AJ, et al. Among authors: baell jb. Bioorg Med Chem Lett. 2005 Jul 1;15(13):3193-6. doi: 10.1016/j.bmcl.2005.05.014. Bioorg Med Chem Lett. 2005. PMID: 15935664

4

Phosphate isosteres in medicinal chemistry.

Rye CS, Baell JB. Rye CS, et al. Among authors: baell jb. Curr Med Chem. 2005;12(26):3127-41. doi: 10.2174/092986705774933452. Curr Med Chem. 2005. PMID: 16375706 Review.

5

A new class of blockers of the voltage-gated potassium channel Kv1.3 via modification of the 4- or 7-position of khellinone.

Harvey AJ, Baell JB, Toovey N, Homerick D, Wulff H. Harvey AJ, et al. Among authors: baell jb. J Med Chem. 2006 Feb 23;49(4):1433-41. doi: 10.1021/jm050839v. J Med Chem. 2006. PMID: 16480279

6

Synthesis and biological evaluation of chalcones as inhibitors of the voltage-gated potassium channel Kv1.3.

Cianci J, Baell JB, Flynn BL, Gable RW, Mould JA, Paul D, Harvey AJ. Cianci J, et al. Among authors: baell jb. Bioorg Med Chem Lett. 2008 Mar 15;18(6):2055-61. doi: 10.1016/j.bmcl.2008.01.099. Epub 2008 Jan 31. Bioorg Med Chem Lett. 2008. PMID: 18289849

7

Trypanothione reductase high-throughput screening campaign identifies novel classes of inhibitors with antiparasitic activity.

Holloway GA, Charman WN, Fairlamb AH, Brun R, Kaiser M, Kostewicz E, Novello PM, Parisot JP, Richardson J, Street IP, Watson KG, Baell JB. Holloway GA, et al. Among authors: baell jb. Antimicrob Agents Chemother. 2009 Jul;53(7):2824-33. doi: 10.1128/AAC.01568-08. Epub 2009 Apr 13. Antimicrob Agents Chemother. 2009. PMID: 19364854 Free PMC article.

8

New substructure filters for removal of pan assay interference compounds (PAINS) from screening libraries and for their exclusion in bioassays.

Baell JB, Holloway GA. Baell JB, et al. J Med Chem. 2010 Apr 8;53(7):2719-40. doi: 10.1021/jm901137j. J Med Chem. 2010. PMID: 20131845

9

Inhibitors of Leishmania GDP-mannose pyrophosphorylase identified by high-throughput screening of small-molecule chemical library.

Lackovic K, Parisot JP, Sleebs N, Baell JB, Debien L, Watson KG, Curtis JM, Handman E, Street IP, Kedzierski L. Lackovic K, et al. Among authors: baell jb. Antimicrob Agents Chemother. 2010 May;54(5):1712-9. doi: 10.1128/AAC.01634-09. Epub 2010 Feb 16. Antimicrob Agents Chemother. 2010. PMID: 20160053 Free PMC article.

10

Discovery of novel and potent benzhydryl-tropane trypanocides highly selective for Trypanosoma cruzi.

Holloway GA, Parisot JP, Novello PM, Watson KG, Armstrong T, Thompson RC, Street IP, Baell JB. Holloway GA, et al. Among authors: baell jb. Bioorg Med Chem Lett. 2010 Mar 15;20(6):1816-8. doi: 10.1016/j.bmcl.2010.02.022. Epub 2010 Feb 8. Bioorg Med Chem Lett. 2010. PMID: 20185305 Free article.

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