Einsiedel J - Search Results

1

3,4,6-Tri-O-acetyl-2-deoxy-2-[18F]fluoroglucopyranosyl phenylthiosulfonate: a thiol-reactive agent for the chemoselective 18F-glycosylation of peptides.

Prante O, Einsiedel J, Haubner R, Gmeiner P, Wester HJ, Kuwert T, Maschauer S. Prante O, et al. Among authors: einsiedel j. Bioconjug Chem. 2007 Jan-Feb;18(1):254-62. doi: 10.1021/bc060340v. Bioconjug Chem. 2007. PMID: 17226980

2

Cyclic amidines as benzamide bioisosteres: EPC synthesis and SAR studies leading to the selective dopamine D4 receptor agonist FAUC 312.

Einsiedel J, Hübner H, Gmeiner P. Einsiedel J, et al. Bioorg Med Chem Lett. 2003 Mar 10;13(5):851-4. doi: 10.1016/s0960-894x(03)00004-0. Bioorg Med Chem Lett. 2003. PMID: 12617906

3

Stereocontrolled dopamine receptor binding and subtype selectivity of clebopride analogues synthesized from aspartic acid.

Einsiedel J, Weber K, Thomas C, Lehmann T, Hübner H, Gmeiner P. Einsiedel J, et al. Bioorg Med Chem Lett. 2003 Oct 6;13(19):3293-6. doi: 10.1016/s0960-894x(03)00678-4. Bioorg Med Chem Lett. 2003. PMID: 12951112

4

Evaluation of lactam-bridged neurotensin analogues adjusting psi(Pro10) close to the experimentally derived bioactive conformation of NT(8-13).

Bittermann H, Einsiedel J, Hübner H, Gmeiner P. Bittermann H, et al. Among authors: einsiedel j. J Med Chem. 2004 Oct 21;47(22):5587-90. doi: 10.1021/jm049644y. J Med Chem. 2004. PMID: 15481995

5

A highly practical RCM approach towards a molecular building kit of spirocyclic reverse turn mimics.

Bittermann H, Böckler F, Einsiedel J, Gmeiner P. Bittermann H, et al. Among authors: einsiedel j. Chemistry. 2006 Aug 16;12(24):6315-22. doi: 10.1002/chem.200600432. Chemistry. 2006. PMID: 16729342

6

Peptide backbone modifications on the C-terminal hexapeptide of neurotensin.

Einsiedel J, Hübner H, Hervet M, Härterich S, Koschatzky S, Gmeiner P. Einsiedel J, et al. Bioorg Med Chem Lett. 2008 Mar 15;18(6):2013-8. doi: 10.1016/j.bmcl.2008.01.110. Epub 2008 Feb 2. Bioorg Med Chem Lett. 2008. PMID: 18276136

7

Novel insights into GPCR-peptide interactions: mutations in extracellular loop 1, ligand backbone methylations and molecular modeling of neurotensin receptor 1.

Härterich S, Koschatzky S, Einsiedel J, Gmeiner P. Härterich S, et al. Among authors: einsiedel j. Bioorg Med Chem. 2008 Oct 15;16(20):9359-68. doi: 10.1016/j.bmc.2008.08.051. Epub 2008 Aug 27. Bioorg Med Chem. 2008. PMID: 18809332

8

Labeling and glycosylation of peptides using click chemistry: a general approach to (18)F-glycopeptides as effective imaging probes for positron emission tomography.

Maschauer S, Einsiedel J, Haubner R, Hocke C, Ocker M, Hübner H, Kuwert T, Gmeiner P, Prante O. Maschauer S, et al. Among authors: einsiedel j. Angew Chem Int Ed Engl. 2010;49(5):976-9. doi: 10.1002/anie.200904137. Angew Chem Int Ed Engl. 2010. PMID: 20029856 No abstract available.

9

Functional characterization of a partial loss-of-function mutation of the epithelial sodium channel (ENaC) associated with atypical cystic fibrosis.

Huber R, Krueger B, Diakov A, Korbmacher J, Haerteis S, Einsiedel J, Gmeiner P, Azad AK, Cuppens H, Cassiman JJ, Korbmacher C, Rauh R. Huber R, et al. Among authors: einsiedel j. Cell Physiol Biochem. 2010;25(1):145-58. doi: 10.1159/000272059. Epub 2009 Dec 22. Cell Physiol Biochem. 2010. PMID: 20054153

10

Click-chemistry-derived tetracycline-amino acid conjugates exhibiting exceptional potency and exclusive recognition of the reverse tet repressor.

Usai I, Krueger M, Einsiedel J, Hillen W, Gmeiner P. Usai I, et al. Among authors: einsiedel j. Chembiochem. 2010 Mar 22;11(5):703-12. doi: 10.1002/cbic.200900710. Chembiochem. 2010. PMID: 20148427

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