Segarra V - Search Results

1

1-, 3- and 8-substituted-9-deazaxanthines as potent and selective antagonists at the human A2B adenosine receptor.

Stefanachi A, Brea JM, Cadavid MI, Centeno NB, Esteve C, Loza MI, Martinez A, Nieto R, Raviña E, Sanz F, Segarra V, Sotelo E, Vidal B, Carotti A. Stefanachi A, et al. Among authors: segarra v. Bioorg Med Chem. 2008 Mar 15;16(6):2852-69. doi: 10.1016/j.bmc.2008.01.002. Epub 2008 Jan 10. Bioorg Med Chem. 2008. PMID: 18226909

2

Synthesis, adenosine receptor binding and 3D-QSAR of 4-substituted 2-(2'-furyl)-1,2,4-triazolo[1,5-a]quinoxalines.

Martínez A, Gutiérrez-de-Terán H, Brea J, Raviña E, Loza MI, Cadavid MI, Sanz F, Vidal B, Segarra V, Sotelo E. Martínez A, et al. Among authors: segarra v. Bioorg Med Chem. 2008 Feb 15;16(4):2103-13. doi: 10.1016/j.bmc.2007.10.103. Epub 2008 Jan 24. Bioorg Med Chem. 2008. PMID: 18249548

3

1,3-dialkyl-8-N-substituted benzyloxycarbonylamino-9-deazaxanthines as potent adenosine receptor ligands: Design, synthesis, structure-affinity and structure-selectivity relationships.

Fernández F, Caamaño O, Isabel Nieto M, López C, García-Mera X, Stefanachi A, Nicolotti O, Isabel Loza M, Brea J, Esteve C, Segarra V, Vidal B, Carotti A. Fernández F, et al. Among authors: segarra v. Bioorg Med Chem. 2009 May 15;17(10):3618-29. doi: 10.1016/j.bmc.2009.03.062. Epub 2009 Apr 5. Bioorg Med Chem. 2009. PMID: 19398343

4

Design, synthesis, and structure-activity relationships of 1-,3-,8-, and 9-substituted-9-deazaxanthines at the human A2B adenosine receptor.

Carotti A, Cadavid MI, Centeno NB, Esteve C, Loza MI, Martinez A, Nieto R, Raviña E, Sanz F, Segarra V, Sotelo E, Stefanachi A, Vidal B. Carotti A, et al. Among authors: segarra v. J Med Chem. 2006 Jan 12;49(1):282-99. doi: 10.1021/jm0506221. J Med Chem. 2006. PMID: 16392813

5

1,7-Naphthyridine 1-oxides as novel potent and selective inhibitors of p38 mitogen activated protein kinase.

Lumeras W, Vidal L, Vidal B, Balagué C, Orellana A, Maldonado M, Domínguez M, Segarra V, Caturla F. Lumeras W, et al. Among authors: segarra v. J Med Chem. 2011 Nov 24;54(22):7899-910. doi: 10.1021/jm200975u. Epub 2011 Oct 31. J Med Chem. 2011. PMID: 21999461

6

Novel heterocyclic-fused pyridazinones as potent and selective phosphodiesterase IV inhibitors.

Dal Piaz V, Giovannoni MP, Castellana C, Palacios JM, Beleta J, Doménech T, Segarra V. Dal Piaz V, et al. Among authors: segarra v. J Med Chem. 1997 May 9;40(10):1417-21. doi: 10.1021/jm970105l. J Med Chem. 1997. PMID: 9154964

7

CoMFA of benzyl derivatives of 2,1,3-benzo and benzothieno[3,2-alpha]thiadiazine 2,2-dioxides: clues for the design of phosphodiesterase 7 inhibitors.

Castro A, Abasolo MI, Gil C, Segarra V, Martinez A. Castro A, et al. Among authors: segarra v. Eur J Med Chem. 2001 Apr;36(4):333-8. doi: 10.1016/s0223-5234(01)01227-2. Eur J Med Chem. 2001. PMID: 11461758

8

Phosphodiesterase inhibitory properties of losartan. Design and synthesis of new lead compounds.

Segarra V, Crespo MI, Pujol F, Beleta J, Doménech T, Miralpeix M, Palacios JM, Castro A, Martinez A. Segarra V, et al. Bioorg Med Chem Lett. 1998 Mar 3;8(5):505-10. doi: 10.1016/s0960-894x(98)00058-4. Bioorg Med Chem Lett. 1998. PMID: 9871607

9

Benzyl derivatives of 2,1,3-benzo- and benzothieno[3,2-a]thiadiazine 2,2-dioxides: first phosphodiesterase 7 inhibitors.

Martínez A, Castro A, Gil C, Miralpeix M, Segarra V, Doménech T, Beleta J, Palacios JM, Ryder H, Miró X, Bonet C, Casacuberta JM, Azorín F, Piña B, Puigdoménech P. Martínez A, et al. Among authors: segarra v. J Med Chem. 2000 Feb 24;43(4):683-9. doi: 10.1021/jm990382n. J Med Chem. 2000. PMID: 10691694

10

Discovery of novel quaternary ammonium derivatives of (3R)-quinuclidinyl amides as potent and long acting muscarinic antagonists.

Prat M, Buil MA, Fernández MD, Tort L, Monleón JM, Casals G, Ferrer M, Castro J, Gavaldà A, Miralpeix M, Ramos I, Vilella D, Huerta JM, Espinosa S, Hernández B, Segarra V, Córdoba M. Prat M, et al. Among authors: segarra v. Bioorg Med Chem Lett. 2015 Apr 15;25(8):1736-1741. doi: 10.1016/j.bmcl.2015.02.065. Epub 2015 Mar 5. Bioorg Med Chem Lett. 2015. PMID: 25800115

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