Gratteri P - Search Results

1

Synthesis, SAR and in vitro evaluation of new cyclic Arg-Gly-Asp pseudopentapeptides containing a s-cis peptide bond as integrin alphavbeta3 and alphavbeta5 ligands.

Salvati M, Cordero FM, Pisaneschi F, Melani F, Gratteri P, Cini N, Bottoncetti A, Brandi A. Salvati M, et al. Among authors: gratteri p. Bioorg Med Chem. 2008 Apr 15;16(8):4262-71. doi: 10.1016/j.bmc.2008.02.080. Epub 2008 Feb 29. Bioorg Med Chem. 2008. PMID: 18343671

2

FILO (field interaction ligand optimization): a simplex strategy for searching the optimal ligand interaction field in drug design.

Melani F, Gratteri P, Adamo M, Bonaccini C. Melani F, et al. Among authors: gratteri p. J Comput Aided Mol Des. 2001 Jan;15(1):57-66. doi: 10.1023/a:1011178027463. J Comput Aided Mol Des. 2001. PMID: 11217919

3

Synthesis and benzodiazepine receptor affinity of pyrazolo[1,5-a]pyrimidine derivatives. 3. New 6-(3-thienyl) series as alpha 1 selective ligands.

Selleri S, Bruni F, Costagli C, Costanzo A, Guerrini G, Ciciani G, Gratteri P, Bonaccini C, Malmberg Aiello P, Besnard F, Renard S, Costa B, Martini C. Selleri S, et al. Among authors: gratteri p. J Med Chem. 2003 Jan 16;46(2):310-3. doi: 10.1021/jm020999w. J Med Chem. 2003. PMID: 12519068

4

Field interaction and geometrical overlap: a new simplex and experimental design based computational procedure for superposing small ligand molecules.

Melani F, Gratteri P, Adamo M, Bonaccini C. Melani F, et al. Among authors: gratteri p. J Med Chem. 2003 Apr 10;46(8):1359-71. doi: 10.1021/jm0210616. J Med Chem. 2003. PMID: 12672236

5

Searching for a reliable orientation of ligands in their binding site: comparison between a structure-based (Glide) and a ligand-based (FIGO) approach in the case study of PDE4 inhibitors.

Gratteri P, Bonaccini C, Melani F. Gratteri P, et al. J Med Chem. 2005 Mar 10;48(5):1657-65. doi: 10.1021/jm049289b. J Med Chem. 2005. PMID: 15743207

6

Insight into 2-phenylpyrazolo[1,5-a]pyrimidin-3-yl acetamides as peripheral benzodiazepine receptor ligands: synthesis, biological evaluation and 3D-QSAR investigation.

Selleri S, Gratteri P, Costagli C, Bonaccini C, Costanzo A, Melani F, Guerrini G, Ciciani G, Costa B, Spinetti F, Martini C, Bruni F. Selleri S, et al. Among authors: gratteri p. Bioorg Med Chem. 2005 Aug 15;13(16):4821-34. doi: 10.1016/j.bmc.2005.05.015. Bioorg Med Chem. 2005. PMID: 15975799

7

A novel selective GABA(A) alpha1 receptor agonist displaying sedative and anxiolytic-like properties in rodents.

Selleri S, Bruni F, Costagli C, Costanzo A, Guerrini G, Ciciani G, Gratteri P, Besnard F, Costa B, Montali M, Martini C, Fohlin J, De Siena G, Aiello PM. Selleri S, et al. Among authors: gratteri p. J Med Chem. 2005 Oct 20;48(21):6756-60. doi: 10.1021/jm058002n. J Med Chem. 2005. PMID: 16220991

8

Structural investigation of the 7-chloro-3-hydroxy-1H-quinazoline-2,4-dione scaffold to obtain AMPA and kainate receptor selective antagonists. Synthesis, pharmacological, and molecular modeling studies.

Colotta V, Catarzi D, Varano F, Lenzi O, Filacchioni G, Costagli C, Galli A, Ghelardini C, Galeotti N, Gratteri P, Sgrignani J, Deflorian F, Moro S. Colotta V, et al. Among authors: gratteri p. J Med Chem. 2006 Oct 5;49(20):6015-26. doi: 10.1021/jm0604880. J Med Chem. 2006. PMID: 17004715

9

Modeling and biological investigations of an unusual behavior of novel synthesized acridine-based polyamine ligands in the binding of double helix and G-quadruplex DNA.

Bazzicalupi C, Chioccioli M, Sissi C, Porcù E, Bonaccini C, Pivetta C, Bencini A, Giorgi C, Valtancoli B, Melani F, Gratteri P. Bazzicalupi C, et al. Among authors: gratteri p. ChemMedChem. 2010 Dec 3;5(12):1995-2005. doi: 10.1002/cmdc.201000332. ChemMedChem. 2010. PMID: 20957717

10

Benzenesulfonamides Incorporating Flexible Triazole Moieties Are Highly Effective Carbonic Anhydrase Inhibitors: Synthesis and Kinetic, Crystallographic, Computational, and Intraocular Pressure Lowering Investigations.

Nocentini A, Ferraroni M, Carta F, Ceruso M, Gratteri P, Lanzi C, Masini E, Supuran CT. Nocentini A, et al. Among authors: gratteri p. J Med Chem. 2016 Dec 8;59(23):10692-10704. doi: 10.1021/acs.jmedchem.6b01389. Epub 2016 Nov 21. J Med Chem. 2016. PMID: 27933963

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