Boschelli DH - Search Results

1

C-5 Substituted heteroaryl 3-pyridinecarbonitriles as PKCtheta inhibitors: Part I.

Subrath J, Wang D, Wu B, Niu C, Boschelli DH, Lee J, Yang X, Brennan A, Chaudhary D. Subrath J, et al. Among authors: boschelli dh. Bioorg Med Chem Lett. 2009 Sep 15;19(18):5423-5. doi: 10.1016/j.bmcl.2009.07.109. Epub 2009 Jul 26. Bioorg Med Chem Lett. 2009. PMID: 19682896

2

Further studies on ethenyl and ethynyl-4-phenylamino-3-quinolinecarbonitriles: identification of a subnanomolar Src kinase inhibitor.

Barrios Sosa AC, Boschelli DH, Wu B, Wang Y, Golas JM. Barrios Sosa AC, et al. Among authors: boschelli dh. Bioorg Med Chem Lett. 2005 Mar 15;15(6):1743-7. doi: 10.1016/j.bmcl.2005.01.004. Bioorg Med Chem Lett. 2005. PMID: 15745832

3

Inhibition of Src kinase activity by 7-[(2,4-dichloro-5-methoxyphenyl)amino]-2-heteroaryl-thieno[3,2-b]pyridine-6-carbonitriles.

Boschelli DH, Wu B, Barrios Sosa AC, Chen JJ, Golas JM, Boschelli F. Boschelli DH, et al. Among authors: boschelli f. Bioorg Med Chem Lett. 2005 Nov 1;15(21):4681-4. doi: 10.1016/j.bmcl.2005.07.061. Bioorg Med Chem Lett. 2005. PMID: 16125383

4

7-(aryl/heteroaryl-2-ylethynyl)-4-phenylamino-3-quinolinecarbonitriles as new Src kinase inhibitors: addition of water solubilizing groups.

Wu B, Barrios Sosa AC, Boschelli DH, Boschelli F, Honores EE, Golas JM, Powell DW, Wang YD. Wu B, et al. Among authors: boschelli dh, boschelli f. Bioorg Med Chem Lett. 2006 Aug 1;16(15):3993-7. doi: 10.1016/j.bmcl.2006.05.015. Epub 2006 Jun 2. Bioorg Med Chem Lett. 2006. PMID: 16735116

5

Synthesis and PKCtheta inhibitory activity of a series of 4-(indol-5-ylamino)thieno[2,3-b]pyridine-5-carbonitriles.

Boschelli DH, Wu B, Barrios Sosa AC, Chen J, Asselin M, Cole DC, Lee J, Yang X, Chaudhary D. Boschelli DH, et al. Bioorg Med Chem Lett. 2008 May 1;18(9):2850-3. doi: 10.1016/j.bmcl.2008.03.077. Epub 2008 Apr 8. Bioorg Med Chem Lett. 2008. PMID: 18434148

6

2-Alkenylthieno[2,3-b]pyridine-5-carbonitriles: Potent and selective inhibitors of PKCtheta.

Nathan Tumey L, Boschelli DH, Lee J, Chaudhary D. Nathan Tumey L, et al. Among authors: boschelli dh. Bioorg Med Chem Lett. 2008 Aug 1;18(15):4420-3. doi: 10.1016/j.bmcl.2008.06.040. Epub 2008 Jun 18. Bioorg Med Chem Lett. 2008. PMID: 18606543

7

Second generation 4-(4-methyl-1H-indol-5-ylamino)-2-phenylthieno[2,3-b]pyridine-5-carbonitrile PKCtheta inhibitors.

Wu B, Boschelli DH, Lee J, Yang X, Chaudhary D. Wu B, et al. Among authors: boschelli dh. Bioorg Med Chem Lett. 2009 Feb 1;19(3):766-9. doi: 10.1016/j.bmcl.2008.12.021. Epub 2008 Dec 10. Bioorg Med Chem Lett. 2009. PMID: 19111463

8

Synthesis and PKCtheta inhibitory activity of a series of 4-indolylamino-5-phenyl-3-pyridinecarbonitriles.

Dushin RG, Nittoli T, Ingalls C, Boschelli DH, Cole DC, Wissner A, Lee J, Yang X, Morgan P, Brennan A, Chaudhary D. Dushin RG, et al. Among authors: boschelli dh. Bioorg Med Chem Lett. 2009 May 1;19(9):2461-3. doi: 10.1016/j.bmcl.2009.03.053. Epub 2009 Mar 18. Bioorg Med Chem Lett. 2009. PMID: 19345579

9

Optimization of 5-phenyl-3-pyridinecarbonitriles as PKCtheta inhibitors.

Boschelli DH, Wang D, Prashad AS, Subrath J, Wu B, Niu C, Lee J, Yang X, Brennan A, Chaudhary D. Boschelli DH, et al. Bioorg Med Chem Lett. 2009 Jul 1;19(13):3623-6. doi: 10.1016/j.bmcl.2009.04.126. Epub 2009 May 3. Bioorg Med Chem Lett. 2009. PMID: 19447612

10

4-Anilino-7-pyridyl-3-quinolinecarbonitriles as Src kinase inhibitors.

Zhang N, Wu B, Boschelli DH, Golas JM, Boschelli F. Zhang N, et al. Among authors: boschelli dh, boschelli f. Bioorg Med Chem Lett. 2009 Sep 1;19(17):5071-4. doi: 10.1016/j.bmcl.2009.07.043. Epub 2009 Jul 10. Bioorg Med Chem Lett. 2009. PMID: 19632113

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

55 results

Search Page

Filters