Ijzerman AP - Search Results

1

Ligand binding and subtype selectivity of the human A(2A) adenosine receptor: identification and characterization of essential amino acid residues.

Jaakola VP, Lane JR, Lin JY, Katritch V, Ijzerman AP, Stevens RC. Jaakola VP, et al. Among authors: ijzerman ap. J Biol Chem. 2010 Apr 23;285(17):13032-44. doi: 10.1074/jbc.M109.096974. Epub 2010 Feb 10. J Biol Chem. 2010. PMID: 20147292 Free PMC article.

2

Identification of the adenine binding site of the human A1 adenosine receptor.

Rivkees SA, Barbhaiya H, IJzerman AP. Rivkees SA, et al. Among authors: ijzerman ap. J Biol Chem. 1999 Feb 5;274(6):3617-21. doi: 10.1074/jbc.274.6.3617. J Biol Chem. 1999. PMID: 9920910 Free article.

3

2-Nitro analogues of adenosine and 1-deazaadenosine: synthesis and binding studies at the adenosine A1, A2A and A3 receptor subtypes.

Wanner MJ, Von Frijtag Drabbe Künzel JK, Ijzerman AP, Koomen GJ. Wanner MJ, et al. Among authors: ijzerman ap. Bioorg Med Chem Lett. 2000 Sep 18;10(18):2141-4. doi: 10.1016/s0960-894x(00)00415-7. Bioorg Med Chem Lett. 2000. PMID: 10999489

4

The 2.6 angstrom crystal structure of a human A2A adenosine receptor bound to an antagonist.

Jaakola VP, Griffith MT, Hanson MA, Cherezov V, Chien EY, Lane JR, Ijzerman AP, Stevens RC. Jaakola VP, et al. Among authors: ijzerman ap. Science. 2008 Nov 21;322(5905):1211-7. doi: 10.1126/science.1164772. Epub 2008 Oct 2. Science. 2008. PMID: 18832607 Free PMC article.

5

Structure-based discovery of novel chemotypes for adenosine A(2A) receptor antagonists.

Katritch V, Jaakola VP, Lane JR, Lin J, Ijzerman AP, Yeager M, Kufareva I, Stevens RC, Abagyan R. Katritch V, et al. Among authors: ijzerman ap. J Med Chem. 2010 Feb 25;53(4):1799-809. doi: 10.1021/jm901647p. J Med Chem. 2010. PMID: 20095623 Free PMC article.

6

Hybrid ortho/allosteric ligands for the adenosine A(1) receptor.

Narlawar R, Lane JR, Doddareddy M, Lin J, Brussee J, Ijzerman AP. Narlawar R, et al. Among authors: ijzerman ap. J Med Chem. 2010 Apr 22;53(8):3028-37. doi: 10.1021/jm901252a. J Med Chem. 2010. PMID: 20345101

7

A novel chemogenomics analysis of G protein-coupled receptors (GPCRs) and their ligands: a potential strategy for receptor de-orphanization.

van der Horst E, Peironcely JE, Ijzerman AP, Beukers MW, Lane JR, van Vlijmen HW, Emmerich MT, Okuno Y, Bender A. van der Horst E, et al. Among authors: ijzerman ap. BMC Bioinformatics. 2010 Jun 10;11:316. doi: 10.1186/1471-2105-11-316. BMC Bioinformatics. 2010. PMID: 20537162 Free PMC article.

8

The crystallographic structure of the human adenosine A2A receptor in a high-affinity antagonist-bound state: implications for GPCR drug screening and design.

Jaakola VP, Ijzerman AP. Jaakola VP, et al. Among authors: ijzerman ap. Curr Opin Struct Biol. 2010 Aug;20(4):401-14. doi: 10.1016/j.sbi.2010.05.002. Epub 2010 Jun 9. Curr Opin Struct Biol. 2010. PMID: 20538452 Review.

9

Characterization of [3H]LUF5834: A novel non-ribose high-affinity agonist radioligand for the adenosine A1 receptor.

Lane JR, Klaasse E, Lin J, van Bruchem J, Beukers MW, Ijzerman AP. Lane JR, et al. Among authors: ijzerman ap. Biochem Pharmacol. 2010 Oct 15;80(8):1180-9. doi: 10.1016/j.bcp.2010.06.041. Epub 2010 Jun 30. Biochem Pharmacol. 2010. PMID: 20599769

10

Structure-activity relationships of trans-substituted-propenoic acid derivatives on the nicotinic acid receptor HCA2 (GPR109A).

van Veldhoven JP, Blad CC, Artsen CM, Klopman C, Wolfram DR, Abdelkadir MJ, Lane JR, Brussee J, Ijzerman AP. van Veldhoven JP, et al. Among authors: ijzerman ap. Bioorg Med Chem Lett. 2011 May 1;21(9):2736-9. doi: 10.1016/j.bmcl.2010.11.091. Epub 2010 Nov 25. Bioorg Med Chem Lett. 2011. PMID: 21167710

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

437 results

Search Page

Filters