Hauser D - Search Results

1

Tri- and tetrasubstituted imidazoles as p38α mitogen-activated protein kinase inhibitors.

Laufer S, Hauser D, Stegmiller T, Bracht C, Ruff K, Schattel V, Albrecht W, Koch P. Laufer S, et al. Among authors: hauser d. Bioorg Med Chem Lett. 2010 Nov 15;20(22):6671-5. doi: 10.1016/j.bmcl.2010.09.012. Epub 2010 Sep 9. Bioorg Med Chem Lett. 2010. PMID: 20934337

2

3,4-Diaryl-isoxazoles and -imidazoles as potent dual inhibitors of p38alpha mitogen activated protein kinase and casein kinase 1delta.

Peifer C, Abadleh M, Bischof J, Hauser D, Schattel V, Hirner H, Knippschild U, Laufer S. Peifer C, et al. Among authors: hauser d. J Med Chem. 2009 Dec 10;52(23):7618-30. doi: 10.1021/jm9005127. J Med Chem. 2009. PMID: 19591487

3

Synthesis and biological testing of purine derivatives as potential ATP-competitive kinase inhibitors.

Laufer SA, Domeyer DM, Scior TR, Albrecht W, Hauser DR. Laufer SA, et al. J Med Chem. 2005 Feb 10;48(3):710-22. doi: 10.1021/jm0408767. J Med Chem. 2005. PMID: 15689155

4

Synthesis, biological testing, and binding mode prediction of 6,9-diarylpurin-8-ones as p38 MAP kinase inhibitors.

Hauser DR, Scior T, Domeyer DM, Kammerer B, Laufer SA. Hauser DR, et al. J Med Chem. 2007 May 3;50(9):2060-6. doi: 10.1021/jm061061w. Epub 2007 Apr 6. J Med Chem. 2007. PMID: 17411025

5

Design, synthesis, and biological evaluation of novel Tri- and tetrasubstituted imidazoles as highly potent and specific ATP-mimetic inhibitors of p38 MAP kinase: focus on optimized interactions with the enzyme's surface-exposed front region.

Laufer SA, Hauser DR, Domeyer DM, Kinkel K, Liedtke AJ. Laufer SA, et al. J Med Chem. 2008 Jul 24;51(14):4122-49. doi: 10.1021/jm701529q. Epub 2008 Jun 26. J Med Chem. 2008. PMID: 18578517

6

2-Acylaminopyridin-4-ylimidazoles as p38 MAP kinase inhibitors: Design, synthesis, and biological and metabolic evaluations.

Ziegler K, Hauser DR, Unger A, Albrecht W, Laufer SA. Ziegler K, et al. ChemMedChem. 2009 Nov;4(11):1939-48. doi: 10.1002/cmdc.200900242. ChemMedChem. 2009. PMID: 19731280

7

Synthesis and biological testing of N-aminoimidazole-based p38alpha MAP kinase inhibitors.

Bracht C, Hauser DR, Schattel V, Albrecht W, Laufer SA. Bracht C, et al. ChemMedChem. 2010 Jul 5;5(7):1134-42. doi: 10.1002/cmdc.201000114. ChemMedChem. 2010. PMID: 20473979

8

Design, synthesis and characterization of N9/N7-substituted 6-aminopurines as VEGF-R and EGF-R inhibitors.

Peifer C, Bühler S, Hauser D, Kinkel K, Totzke F, Schächtele C, Laufer S. Peifer C, et al. Among authors: hauser d. Eur J Med Chem. 2009 Apr;44(4):1788-93. doi: 10.1016/j.ejmech.2008.04.012. Epub 2008 Apr 30. Eur J Med Chem. 2009. PMID: 18524423

9

Fluorescence polarization binding assay to develop inhibitors of inactive p38alpha mitogen-activated protein kinase.

Munoz L, Selig R, Yeung YT, Peifer C, Hauser D, Laufer S. Munoz L, et al. Among authors: hauser d. Anal Biochem. 2010 Jun 1;401(1):125-33. doi: 10.1016/j.ab.2010.02.016. Epub 2010 Feb 20. Anal Biochem. 2010. PMID: 20175985

10

N-{4-[4-(4-Fluoro-phen-yl)-1-methyl-2-[(R)-methyl-sulfin-yl]-1H-imidazol-5-yl]-2-pyridyl}acetamide dihydrate.

Bühler S, Schollmeyer D, Hauser D, Albrecht W, Laufer S. Bühler S, et al. Among authors: hauser d. Acta Crystallogr Sect E Struct Rep Online. 2009 Dec 12;66(Pt 1):o121. doi: 10.1107/S1600536809051873. Acta Crystallogr Sect E Struct Rep Online. 2009. PMID: 21580011 Free PMC article.

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