The orthosteric GABAA receptor ligand Thio-4-PIOL displays distinctly different functional properties at synaptic and extrasynaptic receptors.
Hoestgaard-Jensen K, O'Connor RM, Dalby NO, Simonsen C, Finger BC, Golubeva A, Hammer H, Bergmann ML, Kristiansen U, Krogsgaard-Larsen P, Bräuner-Osborne H, Ebert B, Frølund B, Cryan JF, Jensen AA.
Hoestgaard-Jensen K, et al. Among authors: kristiansen u.
Br J Pharmacol. 2013 Oct;170(4):919-32. doi: 10.1111/bph.12340.
Br J Pharmacol. 2013.
PMID: 23957253
Free PMC article.