Spampinato S - Search Results

1

The inverse type II β-turn on D-Trp-Phe, a pharmacophoric motif for MOR agonists.

Gentilucci L, Tolomelli A, De Marco R, Spampinato S, Bedini A, Artali R. Gentilucci L, et al. Among authors: spampinato s. ChemMedChem. 2011 Sep 5;6(9):1640-53. doi: 10.1002/cmdc.201100169. Epub 2011 Jun 30. ChemMedChem. 2011. PMID: 21721130

2

Synthesis and evaluation of the affinity toward mu-opioid receptors of atypical, lipophilic ligands based on the sequence c[-Tyr-Pro-Trp-Phe-Gly-].

Cardillo G, Gentilucci L, Tolomelli A, Spinosa R, Calienni M, Qasem AR, Spampinato S. Cardillo G, et al. Among authors: spampinato s. J Med Chem. 2004 Oct 7;47(21):5198-203. doi: 10.1021/jm0498811. J Med Chem. 2004. PMID: 15456262

3

Investigation of the interaction between the atypical agonist c[YpwFG] and MOR.

Gentilucci L, Squassabia F, De Marco R, Artali R, Cardillo G, Tolomelli A, Spampinato S, Bedini A. Gentilucci L, et al. Among authors: spampinato s. FEBS J. 2008 May;275(9):2315-37. doi: 10.1111/j.1742-4658.2008.06386.x. Epub 2008 Apr 3. FEBS J. 2008. PMID: 18397320 Free article.

4

Synthesis and conformational analysis of cyclotetrapeptide mimetic beta-turn templates and validation as 3D scaffolds.

Gentilucci L, Cardillo G, Tolomelli A, De Marco R, Garelli A, Spampinato S, Spartà A, Juaristi E. Gentilucci L, et al. Among authors: spampinato s. ChemMedChem. 2009 Apr;4(4):517-23. doi: 10.1002/cmdc.200800407. ChemMedChem. 2009. PMID: 19226499

5

Peripheral antinociceptive effects of the cyclic endomorphin-1 analog c[YpwFG] in a mouse visceral pain model.

Bedini A, Baiula M, Gentilucci L, Tolomelli A, De Marco R, Spampinato S. Bedini A, et al. Among authors: spampinato s. Peptides. 2010 Nov;31(11):2135-40. doi: 10.1016/j.peptides.2010.08.005. Epub 2010 Aug 14. Peptides. 2010. PMID: 20713109

6

Development of isoxazoline-containing peptidomimetics as dual αvβ3 and α5β1 integrin ligands.

Tolomelli A, Gentilucci L, Mosconi E, Viola A, Dattoli SD, Baiula M, Spampinato S, Belvisi L, Civera M. Tolomelli A, et al. Among authors: spampinato s. ChemMedChem. 2011 Dec 9;6(12):2264-72. doi: 10.1002/cmdc.201100372. Epub 2011 Sep 26. ChemMedChem. 2011. PMID: 21953988

7

Opioid activity profiles of oversimplified peptides lacking in the protonable N-terminus.

De Marco R, Tolomelli A, Spampinato S, Bedini A, Gentilucci L. De Marco R, et al. Among authors: spampinato s. J Med Chem. 2012 Nov 26;55(22):10292-6. doi: 10.1021/jm301213s. Epub 2012 Oct 19. J Med Chem. 2012. PMID: 22995061

8

Synthesis of tripeptides containing D-Trp substituted at the indole ring, assessment of opioid receptor binding and in vivo central antinociception.

De Marco R, Bedini A, Spampinato S, Gentilucci L. De Marco R, et al. Among authors: spampinato s. J Med Chem. 2014 Aug 14;57(15):6861-6. doi: 10.1021/jm5002925. Epub 2014 Jul 30. J Med Chem. 2014. PMID: 25051243

9

Versatile Picklocks To Access All Opioid Receptors: Tuning the Selectivity and Functional Profile of the Cyclotetrapeptide c[Phe-d-Pro-Phe-Trp] (CJ-15,208).

De Marco R, Bedini A, Spampinato S, Cavina L, Pirazzoli E, Gentilucci L. De Marco R, et al. Among authors: spampinato s. J Med Chem. 2016 Oct 13;59(19):9255-9261. doi: 10.1021/acs.jmedchem.6b00420. Epub 2016 Sep 22. J Med Chem. 2016. PMID: 27607020

10

Constraining Endomorphin-1 by β,α-Hybrid Dipeptide/Heterocycle Scaffolds: Identification of a Novel κ-Opioid Receptor Selective Partial Agonist.

De Marco R, Bedini A, Spampinato S, Comellini L, Zhao J, Artali R, Gentilucci L. De Marco R, et al. Among authors: spampinato s. J Med Chem. 2018 Jul 12;61(13):5751-5757. doi: 10.1021/acs.jmedchem.8b00296. Epub 2018 Jul 2. J Med Chem. 2018. PMID: 29901392

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