Scaglione F - Search Results

1

Toward the definition of stereochemical requirements for MT2-selective antagonists and partial agonists by studying 4-phenyl-2-propionamidotetralin derivatives.

Bedini A, Lucarini S, Spadoni G, Tarzia G, Scaglione F, Dugnani S, Pannacci M, Lucini V, Carmi C, Pala D, Rivara S, Mor M. Bedini A, et al. Among authors: scaglione f. J Med Chem. 2011 Dec 22;54(24):8362-72. doi: 10.1021/jm200790v. Epub 2011 Nov 18. J Med Chem. 2011. PMID: 22047556

2

Design and synthesis of N-(3,3-diphenylpropenyl)alkanamides as a novel class of high-affinity MT2-selective melatonin receptor ligands.

Bedini A, Spadoni G, Gatti G, Lucarini S, Tarzia G, Rivara S, Lorenzi S, Lodola A, Mor M, Lucini V, Pannacci M, Scaglione F. Bedini A, et al. Among authors: scaglione f. J Med Chem. 2006 Dec 14;49(25):7393-403. doi: 10.1021/jm060850a. J Med Chem. 2006. PMID: 17149869

3

N-(substituted-anilinoethyl)amides: design, synthesis, and pharmacological characterization of a new class of melatonin receptor ligands.

Rivara S, Lodola A, Mor M, Bedini A, Spadoni G, Lucini V, Pannacci M, Fraschini F, Scaglione F, Sanchez RO, Gobbi G, Tarzia G. Rivara S, et al. Among authors: scaglione f. J Med Chem. 2007 Dec 27;50(26):6618-26. doi: 10.1021/jm700957j. Epub 2007 Dec 6. J Med Chem. 2007. PMID: 18052314

4

Design, synthesis, and pharmacological effects of structurally simple ligands for MT(1) and MT(2) melatonin receptors.

Carocci A, Catalano A, Lovece A, Lentini G, Duranti A, Lucini V, Pannacci M, Scaglione F, Franchini C. Carocci A, et al. Among authors: scaglione f. Bioorg Med Chem. 2010 Sep 1;18(17):6496-511. doi: 10.1016/j.bmc.2010.06.100. Epub 2010 Jul 3. Bioorg Med Chem. 2010. PMID: 20674373

5

Bivalent ligand approach on N-{2-[(3-methoxyphenyl)methylamino]ethyl}acetamide: synthesis, binding affinity and intrinsic activity for MT(1) and MT(2) melatonin receptors.

Spadoni G, Bedini A, Orlando P, Lucarini S, Tarzia G, Mor M, Rivara S, Lucini V, Pannacci M, Scaglione F. Spadoni G, et al. Among authors: scaglione f. Bioorg Med Chem. 2011 Aug 15;19(16):4910-6. doi: 10.1016/j.bmc.2011.06.063. Epub 2011 Jun 28. Bioorg Med Chem. 2011. PMID: 21775151

6

MT1-selective melatonin receptor ligands: synthesis, pharmacological evaluation, and molecular dynamics investigation of N-{[(3-O-substituted)anilino]alkyl}amides.

Rivara S, Pala D, Lodola A, Mor M, Lucini V, Dugnani S, Scaglione F, Bedini A, Lucarini S, Tarzia G, Spadoni G. Rivara S, et al. Among authors: scaglione f. ChemMedChem. 2012 Nov;7(11):1954-64. doi: 10.1002/cmdc.201200303. Epub 2012 Aug 27. ChemMedChem. 2012. PMID: 22927210

7

Synthesis and characterization of new bivalent agents as melatonin- and histamine H3-ligands.

Pala D, Scalvini L, Lodola A, Mor M, Flammini L, Barocelli E, Lucini V, Scaglione F, Bartolucci S, Bedini A, Rivara S, Spadoni G. Pala D, et al. Among authors: scaglione f. Int J Mol Sci. 2014 Sep 12;15(9):16114-33. doi: 10.3390/ijms150916114. Int J Mol Sci. 2014. PMID: 25222552 Free PMC article.

8

Highly Potent and Selective MT2 Melatonin Receptor Full Agonists from Conformational Analysis of 1-Benzyl-2-acylaminomethyl-tetrahydroquinolines.

Spadoni G, Bedini A, Lucarini S, Mari M, Caignard DH, Boutin JA, Delagrange P, Lucini V, Scaglione F, Lodola A, Zanardi F, Pala D, Mor M, Rivara S. Spadoni G, et al. Among authors: scaglione f. J Med Chem. 2015 Sep 24;58(18):7512-25. doi: 10.1021/acs.jmedchem.5b01066. J Med Chem. 2015. PMID: 26334942

9

Tetrahydroquinoline Ring as a Versatile Bioisostere of Tetralin for Melatonin Receptor Ligands.

Rivara S, Scalvini L, Lodola A, Mor M, Caignard DH, Delagrange P, Collina S, Lucini V, Scaglione F, Furiassi L, Mari M, Lucarini S, Bedini A, Spadoni G. Rivara S, et al. Among authors: scaglione f. J Med Chem. 2018 Apr 26;61(8):3726-3737. doi: 10.1021/acs.jmedchem.8b00359. Epub 2018 Apr 4. J Med Chem. 2018. PMID: 29595267

10

Chiral Recognition of Flexible Melatonin Receptor Ligands Induced by Conformational Equilibria.

Elisi GM, Bedini A, Scalvini L, Carmi C, Bartolucci S, Lucini V, Scaglione F, Mor M, Rivara S, Spadoni G. Elisi GM, et al. Among authors: scaglione f. Molecules. 2020 Sep 4;25(18):4057. doi: 10.3390/molecules25184057. Molecules. 2020. PMID: 32899888 Free PMC article.

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