Rademann J - Search Results

1

Benzoylphosphonate-based photoactive phosphopeptide mimetics for modulation of protein tyrosine phosphatases and highly specific labeling of SH2 domains.

Horatscheck A, Wagner S, Ortwein J, Kim BG, Lisurek M, Beligny S, Schütz A, Rademann J. Horatscheck A, et al. Among authors: rademann j. Angew Chem Int Ed Engl. 2012 Sep 10;51(37):9441-7. doi: 10.1002/anie.201201475. Epub 2012 Aug 21. Angew Chem Int Ed Engl. 2012. PMID: 22907897 No abstract available.

2

Sensitized detection of inhibitory fragments and iterative development of non-peptidic protease inhibitors by dynamic ligation screening.

Schmidt MF, Isidro-Llobet A, Lisurek M, El-Dahshan A, Tan J, Hilgenfeld R, Rademann J. Schmidt MF, et al. Among authors: rademann j. Angew Chem Int Ed Engl. 2008;47(17):3275-8. doi: 10.1002/anie.200704594. Angew Chem Int Ed Engl. 2008. PMID: 18348134 Free PMC article.

3

Alzheimer's disease: identification and development of β-secretase (BACE-1) binding fragments and inhibitors by dynamic ligation screening (DLS).

Fernández-Bachiller MI, Horatscheck A, Lisurek M, Rademann J. Fernández-Bachiller MI, et al. Among authors: rademann j. ChemMedChem. 2013 Jul;8(7):1041-56. doi: 10.1002/cmdc.201300078. Epub 2013 Jun 11. ChemMedChem. 2013. PMID: 23757181

4

Fluorescent mimetics of CMP-Neu5Ac are highly potent, cell-permeable polarization probes of eukaryotic and bacterial sialyltransferases and inhibit cellular sialylation.

Preidl JJ, Gnanapragassam VS, Lisurek M, Saupe J, Horstkorte R, Rademann J. Preidl JJ, et al. Among authors: rademann j. Angew Chem Int Ed Engl. 2014 May 26;53(22):5700-5. doi: 10.1002/anie.201400394. Epub 2014 Apr 15. Angew Chem Int Ed Engl. 2014. PMID: 24737687

5

Light-switched inhibitors of protein tyrosine phosphatase PTP1B based on phosphonocarbonyl phenylalanine as photoactive phosphotyrosine mimetic.

Wagner S, Schütz A, Rademann J. Wagner S, et al. Among authors: rademann j. Bioorg Med Chem. 2015 Jun 15;23(12):2839-47. doi: 10.1016/j.bmc.2015.03.074. Epub 2015 Apr 4. Bioorg Med Chem. 2015. PMID: 25907367

6

Benzyl Mono-P-Fluorophosphonate and Benzyl Penta-P-Fluorophosphate Anions Are Physiologically Stable Phosphotyrosine Mimetics and Inhibitors of Protein Tyrosine Phosphatases.

Wagner S, Accorsi M, Rademann J. Wagner S, et al. Among authors: rademann j. Chemistry. 2017 Nov 2;23(61):15387-15395. doi: 10.1002/chem.201701204. Epub 2017 Oct 11. Chemistry. 2017. PMID: 29024172

7

The transcription factor STAT5 catalyzes Mannich ligation reactions yielding inhibitors of leukemic cell proliferation.

Wong EL, Nawrotzky E, Arkona C, Kim BG, Beligny S, Wang X, Wagner S, Lisurek M, Carstanjen D, Rademann J. Wong EL, et al. Among authors: rademann j. Nat Commun. 2019 Jan 8;10(1):66. doi: 10.1038/s41467-018-07923-2. Nat Commun. 2019. PMID: 30622248 Free PMC article.

8

Design of chemical libraries with potentially bioactive molecules applying a maximum common substructure concept.

Lisurek M, Rupp B, Wichard J, Neuenschwander M, von Kries JP, Frank R, Rademann J, Kühne R. Lisurek M, et al. Among authors: rademann j. Mol Divers. 2010 May;14(2):401-8. doi: 10.1007/s11030-009-9187-z. Epub 2009 Aug 15. Mol Divers. 2010. PMID: 19685275 Free PMC article.

9

Highly functionalized terpyridines as competitive inhibitors of AKAP-PKA interactions.

Schäfer G, Milić J, Eldahshan A, Götz F, Zühlke K, Schillinger C, Kreuchwig A, Elkins JM, Abdul Azeez KR, Oder A, Moutty MC, Masada N, Beerbaum M, Schlegel B, Niquet S, Schmieder P, Krause G, von Kries JP, Cooper DM, Knapp S, Rademann J, Rosenthal W, Klussmann E. Schäfer G, et al. Among authors: rademann j. Angew Chem Int Ed Engl. 2013 Nov 11;52(46):12187-91. doi: 10.1002/anie.201304686. Epub 2013 Sep 23. Angew Chem Int Ed Engl. 2013. PMID: 24115519 Free PMC article. No abstract available.

10

Selective identification of cooperatively binding fragments in a high-throughput ligation assay enables development of a picomolar caspase-3 inhibitor.

Schmidt MF, El-Dahshan A, Keller S, Rademann J. Schmidt MF, et al. Among authors: rademann j. Angew Chem Int Ed Engl. 2009;48(34):6346-9. doi: 10.1002/anie.200901647. Angew Chem Int Ed Engl. 2009. PMID: 19630042 No abstract available.

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