Lucarini S - Search Results

1

MT1-selective melatonin receptor ligands: synthesis, pharmacological evaluation, and molecular dynamics investigation of N-{[(3-O-substituted)anilino]alkyl}amides.

Rivara S, Pala D, Lodola A, Mor M, Lucini V, Dugnani S, Scaglione F, Bedini A, Lucarini S, Tarzia G, Spadoni G. Rivara S, et al. Among authors: lucarini s. ChemMedChem. 2012 Nov;7(11):1954-64. doi: 10.1002/cmdc.201200303. Epub 2012 Aug 27. ChemMedChem. 2012. PMID: 22927210

2

Design and synthesis of N-(3,3-diphenylpropenyl)alkanamides as a novel class of high-affinity MT2-selective melatonin receptor ligands.

Bedini A, Spadoni G, Gatti G, Lucarini S, Tarzia G, Rivara S, Lorenzi S, Lodola A, Mor M, Lucini V, Pannacci M, Scaglione F. Bedini A, et al. Among authors: lucarini s. J Med Chem. 2006 Dec 14;49(25):7393-403. doi: 10.1021/jm060850a. J Med Chem. 2006. PMID: 17149869

3

N-(Anilinoethyl)amides: design and synthesis of metabolically stable, selective melatonin receptor ligands.

Rivara S, Vacondio F, Fioni A, Silva C, Carmi C, Mor M, Lucini V, Pannacci M, Caronno A, Scaglione F, Gobbi G, Spadoni G, Bedini A, Orlando P, Lucarini S, Tarzia G. Rivara S, et al. Among authors: lucarini s. ChemMedChem. 2009 Oct;4(10):1746-55. doi: 10.1002/cmdc.200900240. ChemMedChem. 2009. PMID: 19728346

4

Bivalent ligand approach on N-{2-[(3-methoxyphenyl)methylamino]ethyl}acetamide: synthesis, binding affinity and intrinsic activity for MT(1) and MT(2) melatonin receptors.

Spadoni G, Bedini A, Orlando P, Lucarini S, Tarzia G, Mor M, Rivara S, Lucini V, Pannacci M, Scaglione F. Spadoni G, et al. Among authors: lucarini s. Bioorg Med Chem. 2011 Aug 15;19(16):4910-6. doi: 10.1016/j.bmc.2011.06.063. Epub 2011 Jun 28. Bioorg Med Chem. 2011. PMID: 21775151

5

Toward the definition of stereochemical requirements for MT2-selective antagonists and partial agonists by studying 4-phenyl-2-propionamidotetralin derivatives.

Bedini A, Lucarini S, Spadoni G, Tarzia G, Scaglione F, Dugnani S, Pannacci M, Lucini V, Carmi C, Pala D, Rivara S, Mor M. Bedini A, et al. Among authors: lucarini s. J Med Chem. 2011 Dec 22;54(24):8362-72. doi: 10.1021/jm200790v. Epub 2011 Nov 18. J Med Chem. 2011. PMID: 22047556

6

Highly Potent and Selective MT2 Melatonin Receptor Full Agonists from Conformational Analysis of 1-Benzyl-2-acylaminomethyl-tetrahydroquinolines.

Spadoni G, Bedini A, Lucarini S, Mari M, Caignard DH, Boutin JA, Delagrange P, Lucini V, Scaglione F, Lodola A, Zanardi F, Pala D, Mor M, Rivara S. Spadoni G, et al. Among authors: lucarini s. J Med Chem. 2015 Sep 24;58(18):7512-25. doi: 10.1021/acs.jmedchem.5b01066. J Med Chem. 2015. PMID: 26334942

7

Tetrahydroquinoline Ring as a Versatile Bioisostere of Tetralin for Melatonin Receptor Ligands.

Rivara S, Scalvini L, Lodola A, Mor M, Caignard DH, Delagrange P, Collina S, Lucini V, Scaglione F, Furiassi L, Mari M, Lucarini S, Bedini A, Spadoni G. Rivara S, et al. Among authors: lucarini s. J Med Chem. 2018 Apr 26;61(8):3726-3737. doi: 10.1021/acs.jmedchem.8b00359. Epub 2018 Apr 4. J Med Chem. 2018. PMID: 29595267

8

Potent, Metabolically Stable 2-Alkyl-8-(2H-1,2,3-triazol-2-yl)-9H-adenines as Adenosine A2A Receptor Ligands.

Pace S, Brogin G, Stasi MA, Riccioni T, Borsini F, Capocasa F, Manera F, Tallarico C, Grossi P, Vacondio F, Bassi M, Bartoccini F, Lucarini S, Piersanti G, Tarzia G, Cabri W, Minetti P. Pace S, et al. Among authors: lucarini s. ChemMedChem. 2015 Jul;10(7):1149-52. doi: 10.1002/cmdc.201500113. Epub 2015 May 7. ChemMedChem. 2015. PMID: 25951302

9

Pharmacokinetic and pharmacodynamic evaluation of ramelteon : an insomnia therapy.

Spadoni G, Bedini A, Lucarini S, Mor M, Rivara S. Spadoni G, et al. Among authors: lucarini s. Expert Opin Drug Metab Toxicol. 2015 Jul;11(7):1145-56. doi: 10.1517/17425255.2015.1045487. Epub 2015 May 8. Expert Opin Drug Metab Toxicol. 2015. PMID: 25956235 Review.

10

2-Arylmelatonin analogues: Probing the 2-phenyl binding pocket of melatonin MT₁ and MT₂ receptors.

Mari M, Elisi GM, Bedini A, Lucarini S, Retini M, Lucini V, Scaglione F, Vincenzi F, Varani K, Castelli R, Mor M, Rivara S, Spadoni G. Mari M, et al. Among authors: lucarini s. Eur J Med Chem. 2022 Dec 5;243:114762. doi: 10.1016/j.ejmech.2022.114762. Epub 2022 Sep 14. Eur J Med Chem. 2022. PMID: 36150258

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