Kulkarni SS - Search Results

1

Fragment-based discovery of new highly substituted 1H-pyrrolo[2,3-b]- and 3H-imidazolo[4,5-b]-pyridines as focal adhesion kinase inhibitors.

Heinrich T, Seenisamy J, Emmanuvel L, Kulkarni SS, Bomke J, Rohdich F, Greiner H, Esdar C, Krier M, Grädler U, Musil D. Heinrich T, et al. Among authors: kulkarni ss. J Med Chem. 2013 Feb 14;56(3):1160-70. doi: 10.1021/jm3016014. Epub 2013 Jan 22. J Med Chem. 2013. PMID: 23294348

2

Structure-activity relationships comparing N-(6-methylpyridin-yl)-substituted aryl amides to 2-methyl-6-(substituted-arylethynyl)pyridines or 2-methyl-4-(substituted-arylethynyl)thiazoles as novel metabotropic glutamate receptor subtype 5 antagonists.

Kulkarni SS, Zou MF, Cao J, Deschamps JR, Rodriguez AL, Conn PJ, Newman AH. Kulkarni SS, et al. J Med Chem. 2009 Jun 11;52(11):3563-75. doi: 10.1021/jm900172f. J Med Chem. 2009. PMID: 19445453 Free PMC article.

3

Discovery of heterobicyclic templates for novel metabotropic glutamate receptor subtype 5 antagonists.

Kulkarni SS, Newman AH. Kulkarni SS, et al. Bioorg Med Chem Lett. 2007 Jun 1;17(11):2987-91. doi: 10.1016/j.bmcl.2007.03.066. Epub 2007 Mar 24. Bioorg Med Chem Lett. 2007. PMID: 17446071 Free PMC article.

4

Structure-activity relationships at monoamine transporters for a series of N-substituted 3alpha-(bis[4-fluorophenyl]methoxy)tropanes: comparative molecular field analysis, synthesis, and pharmacological evaluation.

Kulkarni SS, Grundt P, Kopajtic T, Katz JL, Newman AH. Kulkarni SS, et al. J Med Chem. 2004 Jun 17;47(13):3388-98. doi: 10.1021/jm030646c. J Med Chem. 2004. PMID: 15189035

5

Novel anticholinesterases based on the molecular skeletons of furobenzofuran and methanobenzodioxepine.

Luo W, Yu QS, Zhan M, Parrish D, Deschamps JR, Kulkarni SS, Holloway HW, Alley GM, Lahiri DK, Brossi A, Greig NH. Luo W, et al. Among authors: kulkarni ss. J Med Chem. 2005 Feb 24;48(4):986-94. doi: 10.1021/jm049309+. J Med Chem. 2005. PMID: 15715468

6

Comparative structure-activity relationships of benztropine analogues at the dopamine transporter and histamine H(1) receptors.

Kulkarni SS, Kopajtic TA, Katz JL, Newman AH. Kulkarni SS, et al. Bioorg Med Chem. 2006 Jun 1;14(11):3625-34. doi: 10.1016/j.bmc.2006.01.017. Epub 2006 Feb 3. Bioorg Med Chem. 2006. PMID: 16460947 Free PMC article.

7

Inhibition of human acetyl- and butyrylcholinesterase by novel carbamates of (-)- and (+)-tetrahydrofurobenzofuran and methanobenzodioxepine.

Luo W, Yu QS, Kulkarni SS, Parrish DA, Holloway HW, Tweedie D, Shafferman A, Lahiri DK, Brossi A, Greig NH. Luo W, et al. Among authors: kulkarni ss. J Med Chem. 2006 Apr 6;49(7):2174-85. doi: 10.1021/jm050578p. J Med Chem. 2006. PMID: 16570913 Free PMC article.

8

Synthesis and evaluation of a novel series of 2-chloro-5-((1-methyl-2-(S)-pyrrolidinyl)methoxy)-3-(2-(4-pyridinyl)vinyl)pyridine analogues as potential positron emission tomography imaging agents for nicotinic acetylcholine receptors.

Brown LL, Kulkarni S, Pavlova OA, Koren AO, Mukhin AG, Newman AH, Horti AG. Brown LL, et al. J Med Chem. 2002 Jun 20;45(13):2841-9. doi: 10.1021/jm010550n. J Med Chem. 2002. PMID: 12061886

9

Three-dimensional quantitative structure-activity relationships of mazindol analogues at the dopamine transporter.

Kulkarni SS, Newman AH, Houlihan WJ. Kulkarni SS, et al. J Med Chem. 2002 Sep 12;45(19):4119-27. doi: 10.1021/jm0102093. J Med Chem. 2002. PMID: 12213055

10

Orally Bioavailable Enzymatic Inhibitor of CD38, MK-0159, Protects against Ischemia/Reperfusion Injury in the Murine Heart.

Lagu B, Wu X, Kulkarni S, Paul R, Becherer JD, Olson L, Ravani S, Chatzianastasiou A, Papapetropoulos A, Andrzejewski S. Lagu B, et al. J Med Chem. 2022 Jul 14;65(13):9418-9446. doi: 10.1021/acs.jmedchem.2c00688. Epub 2022 Jun 28. J Med Chem. 2022. PMID: 35762533

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