Thurkauf A - Search Results

1

Synthesis and anticonvulsant activity of 1-phenylcyclohexylamine analogues.

Thurkauf A, de Costa B, Yamaguchi S, Mattson MV, Jacobson AE, Rice KC, Rogawski MA. Thurkauf A, et al. J Med Chem. 1990 May;33(5):1452-8. doi: 10.1021/jm00167a027. J Med Chem. 1990. PMID: 2329567

2

Analogues of the dioxolanes dexoxadrol and etoxadrol as potential phencyclidine-like agents. Synthesis and structure-activity relationships.

Thurkauf A, Mattson MV, Richardson S, Mirsadeghi S, Ornstein PL, Harrison EA Jr, Rice KC, Jacobson AE, Monn JA. Thurkauf A, et al. J Med Chem. 1992 Apr 17;35(8):1323-9. doi: 10.1021/jm00086a001. J Med Chem. 1992. PMID: 1349351

3

Anticonvulsant activity of the low-affinity uncompetitive N-methyl-D- aspartate antagonist (+-)-5-aminocarbonyl-10,11-dihydro-5H- dibenzo[a,d]cyclohepten-5,10-imine (ADCI): comparison with the structural analogs dizocilpine (MK-801) and carbamazepine.

Rogawski MA, Yamaguchi S, Jones SM, Rice KC, Thurkauf A, Monn JA. Rogawski MA, et al. Among authors: thurkauf a. J Pharmacol Exp Ther. 1991 Oct;259(1):30-7. J Pharmacol Exp Ther. 1991. PMID: 1920122

4

Specificity of phencyclidine-like drugs and benzomorphan opiates for two high affinity phencyclidine binding sites in guinea pig brain.

Reid AA, Mattson MV, de Costa BR, Thurkauf A, Jacobson AE, Monn JA, Rice KC, Rothman RB. Reid AA, et al. Among authors: thurkauf a. Neuropharmacology. 1990 Sep;29(9):811-7. doi: 10.1016/0028-3908(90)90154-j. Neuropharmacology. 1990. PMID: 1963480

5

Synthesis and structure-activity relationship of C5-substituted analogues of (+-)-10,11-dihydro-5H-dibenzo[a,d]cyclohepten-5,10-imine [(+-)-desmethyl-MK801]: ligands for the NMDA receptor-coupled phencyclidine binding site.

Monn JA, Thurkauf A, Mattson MV, Jacobson AE, Rice KC. Monn JA, et al. Among authors: thurkauf a. J Med Chem. 1990 Mar;33(3):1069-76. doi: 10.1021/jm00165a029. J Med Chem. 1990. PMID: 2155320

6

Synthesis and evaluation of N-substituted cis-N-methyl-2-(1-pyrrolidinyl)cyclohexylamines as high affinity sigma receptor ligands. Identification of a new class of highly potent and selective sigma receptor probes.

de Costa BR, Rice KC, Bowen WD, Thurkauf A, Rothman RB, Band L, Jacobson AE, Radesca L, Contreras PC, Gray NM, et al. de Costa BR, et al. Among authors: thurkauf a. J Med Chem. 1990 Nov;33(11):3100-10. doi: 10.1021/jm00173a030. J Med Chem. 1990. PMID: 2172538

7

Synthesis, phencyclidine-like pharmacology, and antiischemic potential of meta-substituted 1-(1-phenylcyclohexyl)-1,2,3,6-tetrahydropyridines.

Thurkauf A, de Costa B, Mattson MV, France CP, Price MT, Olney JW, Woods JH, Jacobson AE, Rice KC. Thurkauf A, et al. J Med Chem. 1990 Aug;33(8):2211-5. doi: 10.1021/jm00170a027. J Med Chem. 1990. PMID: 2374147

8

Synthesis and evaluation of optically pure [3H]-(+)-pentazocine, a highly potent and selective radioligand for sigma receptors.

de Costa BR, Bowen WD, Hellewell SB, Walker JM, Thurkauf A, Jacobson AE, Rice KC. de Costa BR, et al. Among authors: thurkauf a. FEBS Lett. 1989 Jul 17;251(1-2):53-8. doi: 10.1016/0014-5793(89)81427-9. FEBS Lett. 1989. PMID: 2568952 Free article.

9

Anticonvulsant activities of 1-phenylcyclohexylamine and its conformationally restricted analog 1,1-pentamethylenetetrahydroisoquinoline.

Rogawski MA, Thurkauf A, Yamaguchi S, Rice KC, Jacobson AE, Mattson MV. Rogawski MA, et al. Among authors: thurkauf a. J Pharmacol Exp Ther. 1989 Jun;249(3):708-12. J Pharmacol Exp Ther. 1989. PMID: 2659775

10

Synthesis, pharmacological action, and receptor binding affinity of the enantiomeric 1-(1-phenyl-3-methylcyclohexyl)piperidines.

Thurkauf A, Hillery P, Mattson MV, Jacobson AE, Rice KC. Thurkauf A, et al. J Med Chem. 1988 Aug;31(8):1625-8. doi: 10.1021/jm00403a023. J Med Chem. 1988. PMID: 2840502

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