Dubowchik GM - Search Results

1

The synthesis and SAR of calcitonin gene-related peptide (CGRP) receptor antagonists derived from tyrosine surrogates. Part 2.

Han X, Civiello RL, Conway CM, Cook DA, Davis CD, Degnan AP, Jiang XJ, Macci R, Mathias NR, Moench P, Pin SS, Schartman R, Signor LJ, Thalody G, Tora G, Whiterock V, Xu C, Macor JE, Dubowchik GM. Han X, et al. Among authors: dubowchik gm. Bioorg Med Chem Lett. 2013 Mar 15;23(6):1870-3. doi: 10.1016/j.bmcl.2013.01.011. Epub 2013 Jan 24. Bioorg Med Chem Lett. 2013. PMID: 23402880

2

Cathepsin B-sensitive dipeptide prodrugs. 1. A model study of structural requirements for efficient release of doxorubicin.

Dubowchik GM, Firestone RA. Dubowchik GM, et al. Bioorg Med Chem Lett. 1998 Dec 1;8(23):3341-6. doi: 10.1016/s0960-894x(98)00609-x. Bioorg Med Chem Lett. 1998. PMID: 9873731

3

Cathepsin B-sensitive dipeptide prodrugs. 2. Models of anticancer drugs paclitaxel (Taxol), mitomycin C and doxorubicin.

Dubowchik GM, Mosure K, Knipe JO, Firestone RA. Dubowchik GM, et al. Bioorg Med Chem Lett. 1998 Dec 1;8(23):3347-52. doi: 10.1016/s0960-894x(98)00610-6. Bioorg Med Chem Lett. 1998. PMID: 9873732

4

Fluoresceinated FKBP12 ligands for a high-throughput fluorescence polarization assay.

Dubowchik GM, Ditta JL, Herbst JJ, Bollini S, Vinitsky A. Dubowchik GM, et al. Bioorg Med Chem Lett. 2000 Mar 20;10(6):559-62. doi: 10.1016/s0960-894x(00)00045-7. Bioorg Med Chem Lett. 2000. PMID: 10741553

5

Synthesis of an immunoconjugate of camptothecin.

Walker MA, Dubowchik GM, Hofstead SJ, Trail PA, Firestone RA. Walker MA, et al. Among authors: dubowchik gm. Bioorg Med Chem Lett. 2002 Jan 21;12(2):217-9. doi: 10.1016/s0960-894x(01)00707-7. Bioorg Med Chem Lett. 2002. PMID: 11755358

6

Doxorubicin immunoconjugates containing bivalent, lysosomally-cleavable dipeptide linkages.

Dubowchik GM, Radia S, Mastalerz H, Walker MA, Firestone RA, Dalton King H, Hofstead SJ, Willner D, Lasch SJ, Trail PA. Dubowchik GM, et al. Bioorg Med Chem Lett. 2002 Jun 3;12(11):1529-32. doi: 10.1016/s0960-894x(02)00194-4. Bioorg Med Chem Lett. 2002. PMID: 12031335

7

Cephalosporin prodrugs of paclitaxel for immunologically specific activation by L-49-sFv-beta-lactamase fusion protein.

Vrudhula VM, Kerr DE, Siemers NO, Dubowchik GM, Senter PD. Vrudhula VM, et al. Among authors: dubowchik gm. Bioorg Med Chem Lett. 2003 Feb 10;13(3):539-42. doi: 10.1016/s0960-894x(02)00935-6. Bioorg Med Chem Lett. 2003. PMID: 12565967

8

2-arylaminothiazoles as high-affinity corticotropin-releasing factor 1 receptor (CRF1R) antagonists: synthesis, binding studies and behavioral efficacy.

Dubowchik GM, Michne JA, Zuev D, Schwartz W, Scola PM, James CA, Ruediger EH, Pin SS, Burris KD, Balanda LA, Gao Q, Wu D, Fung L, Fiedler T, Browman KE, Taber MT, Zhang J. Dubowchik GM, et al. Bioorg Med Chem Lett. 2003 Nov 17;13(22):3997-4000. doi: 10.1016/j.bmcl.2003.08.055. Bioorg Med Chem Lett. 2003. PMID: 14592493

9

An efficient sequence for the preparation of small secondary amine hydrochloride salts for focused library generation without need for distillation or chromatographic purification.

Dubowchik GM, Michne JA, Zuev D. Dubowchik GM, et al. Bioorg Med Chem Lett. 2004 Jun 21;14(12):3147-9. doi: 10.1016/j.bmcl.2004.04.014. Bioorg Med Chem Lett. 2004. PMID: 15149663

10

Tetrahydroisoquinoline derivatives as melatonin MT2 receptor antagonists.

Karageorge GN, Bertenshaw S, Iben L, Xu C, Sarbin N, Gentile A, Dubowchik GM. Karageorge GN, et al. Among authors: dubowchik gm. Bioorg Med Chem Lett. 2004 Dec 6;14(23):5881-4. doi: 10.1016/j.bmcl.2004.09.024. Bioorg Med Chem Lett. 2004. PMID: 15501061

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

56 results

Search Page

Filters