Cronk LA - Search Results

1

A novel series of selective leukotriene antagonists: exploration and optimization of the acidic region in 1,6-disubstituted indoles and indazoles.

Yee YK, Bernstein PR, Adams EJ, Brown FJ, Cronk LA, Hebbel KC, Vacek EP, Krell RD, Snyder DW. Yee YK, et al. Among authors: cronk la. J Med Chem. 1990 Sep;33(9):2437-51. doi: 10.1021/jm00171a018. J Med Chem. 1990. PMID: 2391686

2

1,3,6-trisubstituted indoles as peptidoleukotriene antagonists: benefits of a second, polar, pyrrole substituent.

Brown FJ, Cronk LA, Aharony D, Snyder DW. Brown FJ, et al. Among authors: cronk la. J Med Chem. 1992 Jun 26;35(13):2419-39. doi: 10.1021/jm00091a010. J Med Chem. 1992. PMID: 1320123

3

Synthesis and in vitro LTD4 antagonist activity of bicyclic and monocyclic cyclopentylurethane and cyclopentylacetamide N-arylsulfonyl amides.

Matassa VG, Brown FJ, Bernstein PR, Shapiro HS, Maduskuie TP Jr, Cronk LA, Vacek EP, Yee YK, Snyder DW, Krell RD, et al. Matassa VG, et al. Among authors: cronk la. J Med Chem. 1990 Sep;33(9):2621-9. doi: 10.1021/jm00171a043. J Med Chem. 1990. PMID: 2167983

4

Evolution of a series of peptidoleukotriene antagonists: synthesis and structure-activity relationships of 1,6-disubstituted indoles and indazoles.

Brown FJ, Yee YK, Cronk LA, Hebbel KC, Krell RD, Snyder DW. Brown FJ, et al. Among authors: cronk la. J Med Chem. 1990 Jun;33(6):1771-81. doi: 10.1021/jm00168a036. J Med Chem. 1990. PMID: 2342071

5

Hydroxyacetophenone-derived antagonists of the peptidoleukotrienes.

Brown FJ, Bernstein PR, Cronk LA, Dosset DL, Hebbel KC, Maduskuie TP Jr, Shapiro HS, Vacek EP, Yee YK, Willard AK, et al. Brown FJ, et al. Among authors: cronk la. J Med Chem. 1989 Apr;32(4):807-26. doi: 10.1021/jm00124a014. J Med Chem. 1989. PMID: 2704027

6

Synthesis, structure-activity relationships, and pharmacological evaluation of a series of fluorinated 3-benzyl-5-indolecarboxamides: identification of 4-[[5-[((2R)-2-methyl-4,4,4-trifluorobutyl)carbamoyl]-1-methyl indol- 3-yl]methyl]-3-methoxy-N-[(2-methylphenyl)sulfonyl]benzamide, a potent, orally active antagonist of leukotrienes D4 and E4.

Jacobs RT, Bernstein PR, Cronk LA, Vacek EP, Newcomb LF, Aharony D, Buckner CK, Kusner EJ. Jacobs RT, et al. Among authors: cronk la. J Med Chem. 1994 Apr 29;37(9):1282-97. doi: 10.1021/jm00035a008. J Med Chem. 1994. PMID: 8176706

7

Substituted 3-(phenylmethyl)-1H-indole-5-carboxamides and 1-(phenylmethyl)indole-6-carboxamides as potent, selective, orally active antagonists of the peptidoleukotrienes.

Jacobs RT, Brown FJ, Cronk LA, Aharony D, Buckner CK, Kusner EJ, Kirkland KM, Neilson KL. Jacobs RT, et al. Among authors: cronk la. J Med Chem. 1993 Feb 5;36(3):394-409. doi: 10.1021/jm00055a011. J Med Chem. 1993. PMID: 8381184

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