Harris DL - Search Results

1

Substituted tetrahydroisoquinolines as selective antagonists for the orexin 1 receptor.

Perrey DA, German NA, Gilmour BP, Li JX, Harris DL, Thomas BF, Zhang Y. Perrey DA, et al. Among authors: harris dl. J Med Chem. 2013 Sep 12;56(17):6901-16. doi: 10.1021/jm400720h. Epub 2013 Aug 26. J Med Chem. 2013. PMID: 23941044 Free PMC article.

2

Identifying structural determinants of potency for analogs of apelin-13: integration of C-terminal truncation with structure-activity.

Zhang Y, Maitra R, Harris DL, Dhungana S, Snyder R, Runyon SP. Zhang Y, et al. Among authors: harris dl. Bioorg Med Chem. 2014 Jun 1;22(11):2992-7. doi: 10.1016/j.bmc.2014.04.001. Epub 2014 Apr 13. Bioorg Med Chem. 2014. PMID: 24755525

3

Identification of N-{[6-chloro-4-(2,6-dimethoxyphenyl)quinazolin-2-yl]carbonyl}-l-leucine (NTRC-808), a novel nonpeptide chemotype selective for the neurotensin receptor type 2.

Thomas JB, Giddings AM, Olepu S, Wiethe RW, Harris DL, Narayanan S, Warner KR, Sarret P, Longpre JM, Runyon SP, Gilmour BP. Thomas JB, et al. Among authors: harris dl. Bioorg Med Chem Lett. 2015 Jan 15;25(2):292-6. doi: 10.1016/j.bmcl.2014.11.047. Epub 2014 Nov 24. Bioorg Med Chem Lett. 2015. PMID: 25499438 Free PMC article.

4

Effect of 1-substitution on tetrahydroisoquinolines as selective antagonists for the orexin-1 receptor.

Perrey DA, German NA, Decker AM, Thorn D, Li JX, Gilmour BP, Thomas BF, Harris DL, Runyon SP, Zhang Y. Perrey DA, et al. Among authors: harris dl. ACS Chem Neurosci. 2015 Apr 15;6(4):599-614. doi: 10.1021/cn500330v. Epub 2015 Feb 12. ACS Chem Neurosci. 2015. PMID: 25643283 Free PMC article.

5

Regulation of the Apelinergic System and Its Potential in Cardiovascular Disease: Peptides and Small Molecules as Tools for Discovery.

Narayanan S, Harris DL, Maitra R, Runyon SP. Narayanan S, et al. Among authors: harris dl. J Med Chem. 2015 Oct 22;58(20):7913-27. doi: 10.1021/acs.jmedchem.5b00527. Epub 2015 Jul 10. J Med Chem. 2015. PMID: 26102594 Free PMC article. Review.

6

The importance of the 6- and 7-positions of tetrahydroisoquinolines as selective antagonists for the orexin 1 receptor.

Perrey DA, Decker AM, Li JX, Gilmour BP, Thomas BF, Harris DL, Runyon SP, Zhang Y. Perrey DA, et al. Among authors: harris dl. Bioorg Med Chem. 2015 Sep 1;23(17):5709-24. doi: 10.1016/j.bmc.2015.07.013. Epub 2015 Jul 16. Bioorg Med Chem. 2015. PMID: 26216017 Free PMC article.

7

Discovery of Novel Proline-Based Neuropeptide FF Receptor Antagonists.

Nguyen T, Decker AM, Langston TL, Mathews KM, Siemian JN, Li JX, Harris DL, Runyon SP, Zhang Y. Nguyen T, et al. Among authors: harris dl. ACS Chem Neurosci. 2017 Oct 18;8(10):2290-2308. doi: 10.1021/acschemneuro.7b00219. Epub 2017 Aug 9. ACS Chem Neurosci. 2017. PMID: 28737888 Free PMC article.

8

Blocking Alcoholic Steatosis in Mice with a Peripherally Restricted Purine Antagonist of the Type 1 Cannabinoid Receptor.

Amato GS, Manke A, Harris DL, Wiethe RW, Vasukuttan V, Snyder RW, Lefever TW, Cortes R, Zhang Y, Wang S, Runyon SP, Maitra R. Amato GS, et al. Among authors: harris dl. J Med Chem. 2018 May 24;61(10):4370-4385. doi: 10.1021/acs.jmedchem.7b01820. Epub 2018 May 10. J Med Chem. 2018. PMID: 29688015 Free PMC article.

9

Rational design of cannabinoid type-1 receptor allosteric modulators: Org27569 and PSNCBAM-1 hybrids.

Nguyen T, Gamage TF, Decker AM, Finlay DB, Langston TL, Barrus D, Glass M, Harris DL, Zhang Y. Nguyen T, et al. Among authors: harris dl. Bioorg Med Chem. 2021 Jul 1;41:116215. doi: 10.1016/j.bmc.2021.116215. Epub 2021 May 12. Bioorg Med Chem. 2021. PMID: 34015703 Free PMC article.

10

Discovery of Arylsulfonamides as Dual Orexin Receptor Agonists.

Zhang D, Perrey DA, Decker AM, Langston TL, Mavanji V, Harris DL, Kotz CM, Zhang Y. Zhang D, et al. Among authors: harris dl. J Med Chem. 2021 Jun 24;64(12):8806-8825. doi: 10.1021/acs.jmedchem.1c00841. Epub 2021 Jun 8. J Med Chem. 2021. PMID: 34101446 Free PMC article.

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