Perrone R - Search Results

1

Synthesis, radiolabeling and in vivo evaluation of [(11)C](R)-1-[4-[2-(4-methoxyphenyl)phenyl]piperazin-1-yl]-3-(2-pyrazinyloxy)-2-propanol, a potential PET radioligand for the 5-HT(7) receptor.

Hansen HD, Lacivita E, Di Pilato P, Herth MM, Lehel S, Ettrup A, Andersen VL, Dyssegaard A, De Giorgio P, Perrone R, Berardi F, Colabufo NA, Niso M, Knudsen GM, Leopoldo M. Hansen HD, et al. Among authors: perrone r. Eur J Med Chem. 2014 May 22;79:152-63. doi: 10.1016/j.ejmech.2014.03.066. Epub 2014 Mar 29. Eur J Med Chem. 2014. PMID: 24732791

2

Structure-affinity relationship study on N-[4-(4-arylpiperazin-1-yl)butyl]arylcarboxamides as potent and selective dopamine D(3) receptor ligands.

Leopoldo M, Berardi F, Colabufo NA, De Giorgio P, Lacivita E, Perrone R, Tortorella V. Leopoldo M, et al. Among authors: perrone r. J Med Chem. 2002 Dec 19;45(26):5727-35. doi: 10.1021/jm020952a. J Med Chem. 2002. PMID: 12477356

3

Synthesis and structure-affinity relationships of 1-[omega-(4-aryl-1-piperazinyl)alkyl]-1-aryl ketones as 5-HT(7) receptor ligands.

Perrone R, Berardi F, Colabufo NA, Lacivita E, Leopoldo M, Tortorella V. Perrone R, et al. J Med Chem. 2003 Feb 13;46(4):646-9. doi: 10.1021/jm020994z. J Med Chem. 2003. PMID: 12570387

4

Synthesis of chiral 1-[omega-(4-chlorophenoxy)alkyl]-4-methylpiperidines and their biological evaluation at sigma1, sigma2, and sterol delta8-delta7 isomerase sites.

Berardi F, Loiodice F, Fracchiolla G, Colabufo NA, Perrone R, Tortorella V. Berardi F, et al. Among authors: perrone r. J Med Chem. 2003 May 22;46(11):2117-24. doi: 10.1021/jm021014d. J Med Chem. 2003. PMID: 12747784

5

4-(tetralin-1-yl)- and 4-(naphthalen-1-yl)alkyl derivatives of 1-cyclohexylpiperazine as sigma receptor ligands with agonist sigma2 activity.

Berardi F, Ferorelli S, Abate C, Colabufo NA, Contino M, Perrone R, Tortorella V. Berardi F, et al. Among authors: perrone r. J Med Chem. 2004 Apr 22;47(9):2308-17. doi: 10.1021/jm031026e. J Med Chem. 2004. PMID: 15084129

6

Structure-affinity relationship study on N-(1,2,3,4-tetrahydronaphthalen-1-yl)-4-aryl-1-piperazinealkylamides, a new class of 5-hydroxytryptamine7 receptor agents.

Leopoldo M, Berardi F, Colabufo NA, Contino M, Lacivita E, Niso M, Perrone R, Tortorella V. Leopoldo M, et al. Among authors: perrone r. J Med Chem. 2004 Dec 16;47(26):6616-24. doi: 10.1021/jm049702f. J Med Chem. 2004. PMID: 15588097

7

11C-labeling of n-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]arylcarboxamide derivatives and evaluation as potential radioligands for PET imaging of dopamine D3 receptors.

Turolla EA, Matarrese M, Belloli S, Moresco RM, Simonelli P, Todde S, Fazio F, Magni F, Kienle MG, Leopoldo M, Berardi F, Colabufo NA, Lacivita E, Perrone R. Turolla EA, et al. Among authors: perrone r. J Med Chem. 2005 Nov 3;48(22):7018-23. doi: 10.1021/jm050171k. J Med Chem. 2005. PMID: 16250661

8

First structure-activity relationship study on dopamine D3 receptor agents with N-[4-(4-arylpiperazin-1-yl)butyl]arylcarboxamide structure.

Leopoldo M, Lacivita E, Colabufo NA, Contino M, Berardi F, Perrone R. Leopoldo M, et al. Among authors: perrone r. J Med Chem. 2005 Dec 15;48(25):7919-22. doi: 10.1021/jm050729o. J Med Chem. 2005. PMID: 16335915

9

Methyl substitution on the piperidine ring of N-[omega-(6-methoxynaphthalen-1-yl)alkyl] derivatives as a probe for selective binding and activity at the sigma(1) receptor.

Berardi F, Ferorelli S, Abate C, Pedone MP, Colabufo NA, Contino M, Perrone R. Berardi F, et al. Among authors: perrone r. J Med Chem. 2005 Dec 29;48(26):8237-44. doi: 10.1021/jm050654o. J Med Chem. 2005. PMID: 16366605

10

Design, synthesis, and binding affinities of potential positron emission tomography (PET) ligands for visualization of brain dopamine D3 receptors.

Leopoldo M, Lacivita E, De Giorgio P, Colabufo NA, Niso M, Berardi F, Perrone R. Leopoldo M, et al. Among authors: perrone r. J Med Chem. 2006 Jan 12;49(1):358-65. doi: 10.1021/jm050734s. J Med Chem. 2006. PMID: 16392820

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