Marsault É - Search Results

1

Unraveling the structure-activity relationship of tomatidine, a steroid alkaloid with unique antibiotic properties against persistent forms of Staphylococcus aureus.

Chagnon F, Guay I, Bonin MA, Mitchell G, Bouarab K, Malouin F, Marsault É. Chagnon F, et al. Among authors: marsault e. Eur J Med Chem. 2014 Jun 10;80:605-20. doi: 10.1016/j.ejmech.2013.11.019. Eur J Med Chem. 2014. PMID: 24877760

2

Discovery of a new class of macrocyclic antagonists to the human motilin receptor.

Marsault E, Hoveyda HR, Peterson ML, Saint-Louis C, Landry A, Vézina M, Ouellet L, Wang Z, Ramaseshan M, Beaubien S, Benakli K, Beauchemin S, Déziel R, Peeters T, Fraser GL. Marsault E, et al. J Med Chem. 2006 Nov 30;49(24):7190-7. doi: 10.1021/jm0606600. J Med Chem. 2006. PMID: 17125271

3

Tomatidine inhibits replication of Staphylococcus aureus small-colony variants in cystic fibrosis airway epithelial cells.

Mitchell G, Gattuso M, Grondin G, Marsault É, Bouarab K, Malouin F. Mitchell G, et al. Among authors: marsault e. Antimicrob Agents Chemother. 2011 May;55(5):1937-45. doi: 10.1128/AAC.01468-10. Epub 2011 Feb 28. Antimicrob Agents Chemother. 2011. PMID: 21357296 Free PMC article.

4

Macrocycles are great cycles: applications, opportunities, and challenges of synthetic macrocycles in drug discovery.

Marsault E, Peterson ML. Marsault E, et al. J Med Chem. 2011 Apr 14;54(7):1961-2004. doi: 10.1021/jm1012374. Epub 2011 Mar 7. J Med Chem. 2011. PMID: 21381769 Review. No abstract available.

5

Optimization of the potency and pharmacokinetic properties of a macrocyclic ghrelin receptor agonist (Part I): Development of ulimorelin (TZP-101) from hit to clinic.

Hoveyda HR, Marsault E, Gagnon R, Mathieu AP, Vézina M, Landry A, Wang Z, Benakli K, Beaubien S, Saint-Louis C, Brassard M, Pinault JF, Ouellet L, Bhat S, Ramaseshan M, Peng X, Foucher L, Beauchemin S, Bhérer P, Veber DF, Peterson ML, Fraser GL. Hoveyda HR, et al. Among authors: marsault e. J Med Chem. 2011 Dec 22;54(24):8305-20. doi: 10.1021/jm2007062. Epub 2011 Nov 22. J Med Chem. 2011. PMID: 22106937

6

Tomatidine acts in synergy with aminoglycoside antibiotics against multiresistant Staphylococcus aureus and prevents virulence gene expression.

Mitchell G, Lafrance M, Boulanger S, Séguin DL, Guay I, Gattuso M, Marsault E, Bouarab K, Malouin F. Mitchell G, et al. Among authors: marsault e. J Antimicrob Chemother. 2012 Mar;67(3):559-68. doi: 10.1093/jac/dkr510. Epub 2011 Nov 30. J Antimicrob Chemother. 2012. PMID: 22129590

7

Experimental treatment of Staphylococcus aureus bovine intramammary infection using a guanine riboswitch ligand analog.

Ster C, Allard M, Boulanger S, Lamontagne Boulet M, Mulhbacher J, Lafontaine DA, Marsault E, Lacasse P, Malouin F. Ster C, et al. Among authors: marsault e. J Dairy Sci. 2013 Feb;96(2):1000-8. doi: 10.3168/jds.2012-5890. Epub 2012 Dec 14. J Dairy Sci. 2013. PMID: 23245959 Free article.

8

Design and synthesis of potent, selective inhibitors of matriptase.

Colombo E, Désilets A, Duchêne D, Chagnon F, Najmanovich R, Leduc R, Marsault E. Colombo E, et al. Among authors: marsault e. ACS Med Chem Lett. 2012 Apr 11;3(7):530-4. doi: 10.1021/ml3000534. eCollection 2012 Jul 12. ACS Med Chem Lett. 2012. PMID: 24900505 Free PMC article.

9

Analysis of subpocket selectivity and identification of potent selective inhibitors for matriptase and matriptase-2.

Duchêne D, Colombo E, Désilets A, Boudreault PL, Leduc R, Marsault E, Najmanovich R. Duchêne D, et al. Among authors: marsault e. J Med Chem. 2014 Dec 11;57(23):10198-204. doi: 10.1021/jm5015633. Epub 2014 Nov 21. J Med Chem. 2014. PMID: 25387268

10

One-pot synthesis of polyunsaturated fatty acid amides with anti-proliferative properties.

Tremblay H, St-Georges C, Legault MA, Morin C, Fortin S, Marsault E. Tremblay H, et al. Among authors: marsault e. Bioorg Med Chem Lett. 2014 Dec 15;24(24):5635-5638. doi: 10.1016/j.bmcl.2014.10.084. Epub 2014 Nov 1. Bioorg Med Chem Lett. 2014. PMID: 25466189

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