Pinard E - Search Results

1

3-Amido-3-aryl-piperidines: A Novel Class of Potent, Selective, and Orally Active GlyT1 Inhibitors.

Pinard E, Alberati D, Alvarez-Sanchez R, Brom V, Burner S, Fischer H, Hauser N, Kolczewski S, Lengyel J, Mory R, Saladin C, Schulz-Gasch T, Stalder H. Pinard E, et al. ACS Med Chem Lett. 2014 Feb 4;5(4):428-33. doi: 10.1021/ml500005m. eCollection 2014 Apr 10. ACS Med Chem Lett. 2014. PMID: 24900853 Free PMC article.

2

Discovery of (R)-1-[2-hydroxy-3-(4-hydroxy-phenyl)-propyl]-4-(4-methyl-benzyl)-piperidin-4-ol: a novel NR1/2B subtype selective NMDA receptor antagonist.

Pinard E, Alanine A, Bourson A, Büttelmann B, Gill R, Heitz M, Jaeschke G, Mutel V, Trube G, Wyler R. Pinard E, et al. Bioorg Med Chem Lett. 2001 Aug 20;11(16):2173-6. doi: 10.1016/s0960-894x(01)00392-4. Bioorg Med Chem Lett. 2001. PMID: 11514163

3

4-Aminoquinolines as a novel class of NR1/2B subtype selective NMDA receptor antagonists.

Pinard E, Alanine A, Bourson A, Büttelmann B, Heitz M, Mutela Ramanjit Gill V, Trube G, Wyler R. Pinard E, et al. Bioorg Med Chem Lett. 2002 Sep 16;12(18):2615-9. doi: 10.1016/s0960-894x(02)00470-5. Bioorg Med Chem Lett. 2002. PMID: 12182873

4

2-(3,4-Dihydro-1H-isoquinolin-2yl)-pyridines as a novel class of NR1/2B subtype selective NMDA receptor antagonists.

Büttelmann B, Alanine A, Bourson A, Gill R, Heitz MP, Mutel V, Pinard E, Trube G, Wyler R. Büttelmann B, et al. Among authors: pinard e. Bioorg Med Chem Lett. 2003 Mar 10;13(5):829-32. doi: 10.1016/s0960-894x(03)00007-6. Bioorg Med Chem Lett. 2003. PMID: 12617901

5

4-(3,4-dihydro-1H-isoquinolin-2yl)-pyridines and 4-(3,4-dihydro-1H-isoquinolin-2-yl)-quinolines as potent NR1/2B subtype selective NMDA receptor antagonists.

Büttelmann B, Alanine A, Bourson A, Gill R, Heitz MP, Mutel V, Pinard E, Trube G, Wyler R. Büttelmann B, et al. Among authors: pinard e. Bioorg Med Chem Lett. 2003 May 19;13(10):1759-62. doi: 10.1016/s0960-894x(03)00232-4. Bioorg Med Chem Lett. 2003. PMID: 12729659

6

1-Benzyloxy-4,5-dihydro-1H-imidazol-2-yl-amines, a novel class of NR1/2B subtype selective NMDA receptor antagonists.

Alanine A, Bourson A, Büttelmann B, Gill R, Heitz MP, Mutel V, Pinard E, Trube G, Wyler R. Alanine A, et al. Among authors: pinard e. Bioorg Med Chem Lett. 2003 Oct 6;13(19):3155-9. doi: 10.1016/s0960-894x(03)00713-3. Bioorg Med Chem Lett. 2003. PMID: 12951084

7

Discovery of N-(2-aryl-cyclohexyl) substituted spiropiperidines as a novel class of GlyT1 inhibitors.

Pinard E, Ceccarelli SM, Stalder H, Alberati D. Pinard E, et al. Bioorg Med Chem Lett. 2006 Jan 15;16(2):349-53. doi: 10.1016/j.bmcl.2005.09.075. Epub 2005 Oct 21. Bioorg Med Chem Lett. 2006. PMID: 16246557

8

Discovery of N-(2-hydroxy-2-aryl-cyclohexyl) substituted spiropiperidines as GlyT1 antagonists with improved pharmacological profile.

Ceccarelli SM, Pinard E, Stalder H, Alberati D. Ceccarelli SM, et al. Among authors: pinard e. Bioorg Med Chem Lett. 2006 Jan 15;16(2):354-7. doi: 10.1016/j.bmcl.2005.09.067. Epub 2005 Oct 21. Bioorg Med Chem Lett. 2006. PMID: 16246561

9

Discovery of 4-substituted-8-(2-hydroxy-2-phenyl-cyclohexyl)-2,8-diaza-spiro[4.5]decan-1-one as a novel class of highly selective GlyT1 inhibitors with improved metabolic stability.

Alberati D, Hainzl D, Jolidon S, Krafft EA, Kurt A, Maier A, Pinard E, Thomas AW, Zimmerli D. Alberati D, et al. Among authors: pinard e. Bioorg Med Chem Lett. 2006 Aug 15;16(16):4311-5. doi: 10.1016/j.bmcl.2006.05.058. Epub 2006 Jun 6. Bioorg Med Chem Lett. 2006. PMID: 16757170

10

Design and synthesis of 4-substituted-8-(2-phenyl-cyclohexyl)-2,8-diaza-spiro[4.5]decan-1-one as a novel class of GlyT1 inhibitors: achieving selectivity against the mu opioid and nociceptin/orphanin FQ peptide (NOP) receptors.

Alberati D, Ceccarelli SM, Jolidon S, Krafft EA, Kurt A, Maier A, Pinard E, Stalder H, Studer D, Thomas AW, Zimmerli D. Alberati D, et al. Among authors: pinard e. Bioorg Med Chem Lett. 2006 Aug 15;16(16):4305-10. doi: 10.1016/j.bmcl.2006.05.064. Epub 2006 Jun 9. Bioorg Med Chem Lett. 2006. PMID: 16762548

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