Akdemir A - Search Results

1

Selective inhibition of human carbonic anhydrases by novel amide derivatives of probenecid: synthesis, biological evaluation and molecular modelling studies.

D'Ascenzio M, Carradori S, Secci D, Vullo D, Ceruso M, Akdemir A, Supuran CT. D'Ascenzio M, et al. Among authors: akdemir a. Bioorg Med Chem. 2014 Aug 1;22(15):3982-8. doi: 10.1016/j.bmc.2014.06.003. Epub 2014 Jun 26. Bioorg Med Chem. 2014. PMID: 25027802

2

Identification of novel α7 nicotinic receptor ligands by in silico screening against the crystal structure of a chimeric α7 receptor ligand binding domain.

Akdemir A, Edink E, Thompson AJ, Lummis SC, Kooistra AJ, de Graaf C, de Esch IJ. Akdemir A, et al. Bioorg Med Chem. 2012 Oct 1;20(19):5992-6002. doi: 10.1016/j.bmc.2012.06.054. Epub 2012 Jul 11. Bioorg Med Chem. 2012. PMID: 22959526 Free PMC article.

3

The extremo-α-carbonic anhydrase (CA) from Sulfurihydrogenibium azorense, the fastest CA known, is highly activated by amino acids and amines.

Akdemir A, Vullo D, De Luca V, Scozzafava A, Carginale V, Rossi M, Supuran CT, Capasso C. Akdemir A, et al. Bioorg Med Chem Lett. 2013 Feb 15;23(4):1087-90. doi: 10.1016/j.bmcl.2012.12.009. Epub 2012 Dec 20. Bioorg Med Chem Lett. 2013. PMID: 23294703

4

o-Benzenedisulfonimido-sulfonamides are potent inhibitors of the tumor-associated carbonic anhydrase isoforms CA IX and CA XII.

Güzel-Akdemir Ö, Akdemir A, Isik S, Vullo D, Supuran CT. Güzel-Akdemir Ö, et al. Among authors: akdemir a. Bioorg Med Chem. 2013 Mar 15;21(6):1386-91. doi: 10.1016/j.bmc.2012.12.037. Epub 2013 Jan 4. Bioorg Med Chem. 2013. PMID: 23352754

5

Xanthates and trithiocarbonates strongly inhibit carbonic anhydrases and show antiglaucoma effects in vivo.

Carta F, Akdemir A, Scozzafava A, Masini E, Supuran CT. Carta F, et al. Among authors: akdemir a. J Med Chem. 2013 Jun 13;56(11):4691-700. doi: 10.1021/jm400414j. Epub 2013 May 16. J Med Chem. 2013. PMID: 23647428

6

A class of sulfonamides with strong inhibitory action against the α-carbonic anhydrase from Trypanosoma cruzi.

Güzel-Akdemir Ö, Akdemir A, Pan P, Vermelho AB, Parkkila S, Scozzafava A, Capasso C, Supuran CT. Güzel-Akdemir Ö, et al. Among authors: akdemir a. J Med Chem. 2013 Jul 25;56(14):5773-81. doi: 10.1021/jm400418p. Epub 2013 Jul 10. J Med Chem. 2013. PMID: 23815159

7

Inhibition of tumor-associated human carbonic anhydrase isozymes IX and XII by a new class of substituted-phenylacetamido aromatic sulfonamides.

Akdemir A, Güzel-Akdemir O, Scozzafava A, Capasso C, Supuran CT. Akdemir A, et al. Bioorg Med Chem. 2013 Sep 1;21(17):5228-32. doi: 10.1016/j.bmc.2013.06.029. Epub 2013 Jun 20. Bioorg Med Chem. 2013. PMID: 23842519

8

Computational investigation of the selectivity of salen and tetrahydrosalen compounds towards the tumor-associated hCA XII isozyme.

Akdemir A, De Monte C, Carradori S, Supuran CT. Akdemir A, et al. J Enzyme Inhib Med Chem. 2015 Feb;30(1):114-8. doi: 10.3109/14756366.2014.892936. Epub 2014 Mar 25. J Enzyme Inhib Med Chem. 2015. PMID: 24666302 Free article.

9

Synthesis of a new series of dithiocarbamates with effective human carbonic anhydrase inhibitory activity and antiglaucoma action.

Bozdag M, Carta F, Vullo D, Akdemir A, Isik S, Lanzi C, Scozzafava A, Masini E, Supuran CT. Bozdag M, et al. Among authors: akdemir a. Bioorg Med Chem. 2015 May 15;23(10):2368-76. doi: 10.1016/j.bmc.2015.03.068. Epub 2015 Mar 31. Bioorg Med Chem. 2015. PMID: 25846066

10

Discovery of novel isatin-based sulfonamides with potent and selective inhibition of the tumor-associated carbonic anhydrase isoforms IX and XII.

Güzel-Akdemir Ö, Akdemir A, Karalı N, Supuran CT. Güzel-Akdemir Ö, et al. Among authors: akdemir a. Org Biomol Chem. 2015 Jun 21;13(23):6493-9. doi: 10.1039/c5ob00688k. Epub 2015 May 13. Org Biomol Chem. 2015. PMID: 25967275

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