Sbardella G - Search Results

1

Identification of structural features of 2-alkylidene-1,3-dicarbonyl derivatives that induce inhibition and/or activation of histone acetyltransferases KAT3B/p300 and KAT2B/PCAF.

Castellano S, Milite C, Feoli A, Viviano M, Mai A, Novellino E, Tosco A, Sbardella G. Castellano S, et al. Among authors: sbardella g. ChemMedChem. 2015 Jan;10(1):144-57. doi: 10.1002/cmdc.201402371. Epub 2014 Oct 21. ChemMedChem. 2015. PMID: 25333655

2

Synthesis and anti-HIV-1 activity of thio analogues of dihydroalkoxybenzyloxopyrimidines.

Mai A, Artico M, Sbardella G, Massa S, Loi AG, Tramontano E, Scano P, La Colla P. Mai A, et al. Among authors: sbardella g. J Med Chem. 1995 Aug 18;38(17):3258-63. doi: 10.1021/jm00017a010. J Med Chem. 1995. PMID: 7650679

3

Dihydro(alkylthio)(naphthylmethyl)oxopyrimidines: novel non-nucleoside reverse transcriptase inhibitors of the S-DABO series.

Mai A, Artico M, Sbardella G, Quartarone S, Massa S, Loi AG, De Montis A, Scintu F, Putzolu M, La Colla P. Mai A, et al. Among authors: sbardella g. J Med Chem. 1997 May 9;40(10):1447-54. doi: 10.1021/jm960802y. J Med Chem. 1997. PMID: 9154967

4

N-[4-(1,1'-biphenyl)methyl]-4-(4-thiomorpholinylmethyl) benzenamines as non-oxazolidinone analogues of antimycobacterial U-100480.

Artico M, Mai A, Sbardella G, Massa S, Lampis G, Deidda D, Pompei R. Artico M, et al. Among authors: sbardella g. Bioorg Med Chem Lett. 1998 Jun 16;8(12):1493-8. doi: 10.1016/s0960-894x(98)00248-0. Bioorg Med Chem Lett. 1998. PMID: 9873376

5

5-Alkyl-2-(alkylthio)-6-(2,6-dihalophenylmethyl)-3, 4-dihydropyrimidin-4(3H)-ones: novel potent and selective dihydro-alkoxy-benzyl-oxopyrimidine derivatives.

Mai A, Artico M, Sbardella G, Massa S, Novellino E, Greco G, Loi AG, Tramontano E, Marongiu ME, La Colla P. Mai A, et al. Among authors: sbardella g. J Med Chem. 1999 Feb 25;42(4):619-27. doi: 10.1021/jm980260f. J Med Chem. 1999. PMID: 10052969

6

Nitroquinolones with broad-spectrum antimycobacterial activity in vitro.

Artico M, Mai A, Sbardella G, Massa S, Musiu C, Lostia S, Demontis F, La Colla P. Artico M, et al. Among authors: sbardella g. Bioorg Med Chem Lett. 1999 Jun 21;9(12):1651-6. doi: 10.1016/s0960-894x(99)00251-6. Bioorg Med Chem Lett. 1999. PMID: 10397494

7

Chiral resolution and molecular modeling investigation of rac-2-cyclopentylthio-6-[1-(2,6-difluorophenyl)ethyl]-3,4-dihydro-5-methylpyrimidin-4(3H)-one (MC-1047), a potent anti-HIV-1 reverse transcriptase agent of the DABO class.

Quaglia M, Mai A, Sbardella G, Artico M, Ragno R, Massa S, del Piano D, Setzu G, Doratiotto S, Cotichini V. Quaglia M, et al. Among authors: sbardella g. Chirality. 2001 Feb;13(2):75-80. doi: 10.1002/1520-636X(2001)13:2<75::AID-CHIR1001>3.0.CO;2-W. Chirality. 2001. PMID: 11170249

8

3-(4-aroyl-1H-pyrrol-2-yl)-N-hydroxy-2-propenamides, a new class of synthetic histone deacetylase inhibitors.

Massa S, Mai A, Sbardella G, Esposito M, Ragno R, Loidl P, Brosch G. Massa S, et al. Among authors: sbardella g. J Med Chem. 2001 Jun 21;44(13):2069-72. doi: 10.1021/jm015515v. J Med Chem. 2001. PMID: 11405644

9

Structure-activity relationship studies on new DABOS: effect of substitutions at pyrimidine C-5 and C-6 positions on anti-HIV-1 activity.

Sbardella G, Mai A, Artico M, Chimenti P, Massa S, Loddo R, Marongiu ME, La Collat P, Pani A. Sbardella G, et al. Antivir Chem Chemother. 2001 Jan;12(1):37-50. doi: 10.1177/095632020101200102. Antivir Chem Chemother. 2001. PMID: 11437321 Free article.

10

Structure-based design, synthesis, and biological evaluation of conformationally restricted novel 2-alkylthio-6-[1-(2,6-difluorophenyl)alkyl]-3,4-dihydro-5-alkylpyrimidin-4(3H)-ones as non-nucleoside inhibitors of HIV-1 reverse transcriptase.

Mai A, Sbardella G, Artico M, Ragno R, Massa S, Novellino E, Greco G, Lavecchia A, Musiu C, La Colla M, Murgioni C, La Colla P, Loddo R. Mai A, et al. Among authors: sbardella g. J Med Chem. 2001 Aug 2;44(16):2544-54. doi: 10.1021/jm010853h. J Med Chem. 2001. PMID: 11472208

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

95 results

Search Page

Filters