Van Calenbergh S - Search Results

1

Structure Guided Lead Generation toward Nonchiral M. tuberculosis Thymidylate Kinase Inhibitors.

Song L, Merceron R, Gracia B, Quintana AL, Risseeuw MDP, Hulpia F, Cos P, Aínsa JA, Munier-Lehmann H, Savvides SN, Van Calenbergh S. Song L, et al. Among authors: van calenbergh s. J Med Chem. 2018 Apr 12;61(7):2753-2775. doi: 10.1021/acs.jmedchem.7b01570. Epub 2018 Mar 15. J Med Chem. 2018. PMID: 29510037

2

Synthesis and structure-activity relationships of analogs of 2'-deoxy-2'-(3-methoxybenzamido)adenosine, a selective inhibitor of trypanosomal glycosomal glyceraldehyde-3-phosphate dehydrogenase.

Van Calenbergh S, Verlinde CL, Soenens J, De Bruyn A, Callens M, Blaton NM, Peeters OM, Rozenski J, Hol WG, Herdewijn P. Van Calenbergh S, et al. J Med Chem. 1995 Sep 15;38(19):3838-49. doi: 10.1021/jm00019a014. J Med Chem. 1995. PMID: 7562915

3

N6-cyclopentyl-3'-substituted-xylofuranosyladenosines: a new class of non-xanthine adenosine A1 receptor antagonists.

Van Calenbergh S, von Frijtag Drabbe Künzel JK, Blaton NM, Peeters OM, Rozenski J, Van Aerschot A, De Bruyn A, De Keukeleire D, IJzerman AP, Herdewijn P. Van Calenbergh S, et al. Among authors: van aerschot a. J Med Chem. 1997 Nov 7;40(23):3765-72. doi: 10.1021/jm970176k. J Med Chem. 1997. PMID: 9371242

4

Effect of aromatic short-chain analogues of ceramide on axonal growth in hippocampal neurons.

Van Overmeire I, Boldin SA, Dumont F, Van Calenbergh S, Slegers G, De Keukeleire D, Futerman AH, Herdewijn P. Van Overmeire I, et al. Among authors: van calenbergh s. J Med Chem. 1999 Jul 15;42(14):2697-705. doi: 10.1021/jm990091e. J Med Chem. 1999. PMID: 10411490

5

Structure-activity relationship of short-chain sphingoid bases as inhibitors of sphingosine kinase.

De Jonghe S, Van Overmeire I, Poulton S, Hendrix C, Busson R, Van Calenbergh S, De Keukeleire D, Spiegel S, Herdewijn P. De Jonghe S, et al. Among authors: van overmeire i, van calenbergh s. Bioorg Med Chem Lett. 1999 Nov 1;9(21):3175-80. doi: 10.1016/s0960-894x(99)00554-5. Bioorg Med Chem Lett. 1999. PMID: 10560747

6

Synthesis and biological evaluation of ceramide analogues with substituted aromatic rings or an allylic fluoride in the sphingoid moiety.

Van Overmeire I, Boldin SA, Venkataraman K, Zisling R, De Jonghe S, Van Calenbergh S, De Keukeleire D, Futerman AH, Herdewijn P. Van Overmeire I, et al. Among authors: van calenbergh s. J Med Chem. 2000 Nov 2;43(22):4189-99. doi: 10.1021/jm000939v. J Med Chem. 2000. PMID: 11063615

7

5'-Deoxy congeners of 9-(3-amido-3-deoxy-beta-D-xylofuranosyl)-N(6)-cyclopentyladenine: new adenosine A(1) receptor antagonists and inverse agonists.

Van Calenbergh S, Link A, Fujikawa S, de Ligt RA, Vanheusden V, Golisade A, Blaton NM, Rozenski J, IJzerman AP, Herdewijn P. Van Calenbergh S, et al. J Med Chem. 2002 Apr 25;45(9):1845-52. doi: 10.1021/jm0110439. J Med Chem. 2002. PMID: 11960496

8

Synthesis and evaluation of thymidine-5'-O-monophosphate analogues as inhibitors of Mycobacterium tuberculosis thymidylate kinase.

Vanheusden V, Munier-Lehmann H, Pochet S, Herdewijn P, Van Calenbergh S. Vanheusden V, et al. Among authors: van calenbergh s. Bioorg Med Chem Lett. 2002 Oct 7;12(19):2695-8. doi: 10.1016/s0960-894x(02)00551-6. Bioorg Med Chem Lett. 2002. PMID: 12217356

9

Enzymatic and structural analysis of inhibitors designed against Mycobacterium tuberculosis thymidylate kinase. New insights into the phosphoryl transfer mechanism.

Haouz A, Vanheusden V, Munier-Lehmann H, Froeyen M, Herdewijn P, Van Calenbergh S, Delarue M. Haouz A, et al. Among authors: van calenbergh s. J Biol Chem. 2003 Feb 14;278(7):4963-71. doi: 10.1074/jbc.M209630200. Epub 2002 Nov 25. J Biol Chem. 2003. PMID: 12454011 Free article.

10

3'-C-branched-chain-substituted nucleosides and nucleotides as potent inhibitors of Mycobacterium tuberculosis thymidine monophosphate kinase.

Vanheusden V, Munier-Lehmann H, Froeyen M, Dugué L, Heyerick A, De Keukeleire D, Pochet S, Busson R, Herdewijn P, Van Calenbergh S. Vanheusden V, et al. Among authors: van calenbergh s. J Med Chem. 2003 Aug 28;46(18):3811-21. doi: 10.1021/jm021108n. J Med Chem. 2003. PMID: 12930144 Free article.

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