Van Calenbergh S - Search Results

1

Revisiting tubercidin against kinetoplastid parasites: Aromatic substitutions at position 7 improve activity and reduce toxicity.

Hulpia F, Campagnaro GD, Scortichini M, Van Hecke K, Maes L, de Koning HP, Caljon G, Van Calenbergh S. Hulpia F, et al. Among authors: van hecke k, van calenbergh s. Eur J Med Chem. 2019 Feb 15;164:689-705. doi: 10.1016/j.ejmech.2018.12.050. Epub 2018 Dec 21. Eur J Med Chem. 2019. PMID: 30677668

2

Synthesis and structure-activity relationships of analogs of 2'-deoxy-2'-(3-methoxybenzamido)adenosine, a selective inhibitor of trypanosomal glycosomal glyceraldehyde-3-phosphate dehydrogenase.

Van Calenbergh S, Verlinde CL, Soenens J, De Bruyn A, Callens M, Blaton NM, Peeters OM, Rozenski J, Hol WG, Herdewijn P. Van Calenbergh S, et al. J Med Chem. 1995 Sep 15;38(19):3838-49. doi: 10.1021/jm00019a014. J Med Chem. 1995. PMID: 7562915

3

Effect of aromatic short-chain analogues of ceramide on axonal growth in hippocampal neurons.

Van Overmeire I, Boldin SA, Dumont F, Van Calenbergh S, Slegers G, De Keukeleire D, Futerman AH, Herdewijn P. Van Overmeire I, et al. Among authors: van calenbergh s. J Med Chem. 1999 Jul 15;42(14):2697-705. doi: 10.1021/jm990091e. J Med Chem. 1999. PMID: 10411490

4

Synthesis and biological evaluation of ceramide analogues with substituted aromatic rings or an allylic fluoride in the sphingoid moiety.

Van Overmeire I, Boldin SA, Venkataraman K, Zisling R, De Jonghe S, Van Calenbergh S, De Keukeleire D, Futerman AH, Herdewijn P. Van Overmeire I, et al. Among authors: van calenbergh s. J Med Chem. 2000 Nov 2;43(22):4189-99. doi: 10.1021/jm000939v. J Med Chem. 2000. PMID: 11063615

5

5'-Deoxy congeners of 9-(3-amido-3-deoxy-beta-D-xylofuranosyl)-N(6)-cyclopentyladenine: new adenosine A(1) receptor antagonists and inverse agonists.

Van Calenbergh S, Link A, Fujikawa S, de Ligt RA, Vanheusden V, Golisade A, Blaton NM, Rozenski J, IJzerman AP, Herdewijn P. Van Calenbergh S, et al. J Med Chem. 2002 Apr 25;45(9):1845-52. doi: 10.1021/jm0110439. J Med Chem. 2002. PMID: 11960496

6

3'-C-branched-chain-substituted nucleosides and nucleotides as potent inhibitors of Mycobacterium tuberculosis thymidine monophosphate kinase.

Vanheusden V, Munier-Lehmann H, Froeyen M, Dugué L, Heyerick A, De Keukeleire D, Pochet S, Busson R, Herdewijn P, Van Calenbergh S. Vanheusden V, et al. Among authors: van calenbergh s. J Med Chem. 2003 Aug 28;46(18):3811-21. doi: 10.1021/jm021108n. J Med Chem. 2003. PMID: 12930144 Free article.

7

Discovery of bicyclic thymidine analogues as selective and high-affinity inhibitors of Mycobacterium tuberculosis thymidine monophosphate kinase.

Vanheusden V, Munier-Lehmann H, Froeyen M, Busson R, Rozenski J, Herdewijn P, Van Calenbergh S. Vanheusden V, et al. Among authors: van calenbergh s. J Med Chem. 2004 Dec 2;47(25):6187-94. doi: 10.1021/jm040847w. J Med Chem. 2004. PMID: 15566289

8

Synthesis and biological evaluation of cyclopropyl analogues of fosmidomycin as potent Plasmodium falciparum growth inhibitors.

Devreux V, Wiesner J, Goeman JL, Van der Eycken J, Jomaa H, Van Calenbergh S. Devreux V, et al. Among authors: van der eycken j, van calenbergh s. J Med Chem. 2006 Apr 20;49(8):2656-60. doi: 10.1021/jm051177c. J Med Chem. 2006. PMID: 16610809 Free article.

9

Synthesis and biological evaluation of novel PDMP analogues.

Hillaert U, Boldin-Adamsky S, Rozenski J, Busson R, Futerman AH, Van Calenbergh S. Hillaert U, et al. Among authors: van calenbergh s. Bioorg Med Chem. 2006 Aug 1;14(15):5273-84. doi: 10.1016/j.bmc.2006.03.048. Epub 2006 Apr 18. Bioorg Med Chem. 2006. PMID: 16621573 Free article.

10

Rational design of 5'-thiourea-substituted alpha-thymidine analogues as thymidine monophosphate kinase inhibitors capable of inhibiting mycobacterial growth.

Van Daele I, Munier-Lehmann H, Froeyen M, Balzarini J, Van Calenbergh S. Van Daele I, et al. Among authors: van calenbergh s. J Med Chem. 2007 Nov 1;50(22):5281-92. doi: 10.1021/jm0706158. Epub 2007 Oct 2. J Med Chem. 2007. PMID: 17910427

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