Mackay SP - Search Results

1

Topographical Mapping of Isoform-Selectivity Determinants for J-Channel-Binding Inhibitors of Sphingosine Kinases 1 and 2.

Adams DR, Tawati S, Berretta G, Rivas PL, Baiget J, Jiang Z, Alsfouk A, Mackay SP, Pyne NJ, Pyne S. Adams DR, et al. Among authors: mackay sp. J Med Chem. 2019 Apr 11;62(7):3658-3676. doi: 10.1021/acs.jmedchem.9b00162. Epub 2019 Mar 27. J Med Chem. 2019. PMID: 30889352 Free article.

2

Exploring DNA topoisomerase I inhibition by the benzo[c]phenanthridines fagaronine and ethoxidine using steered molecular dynamics.

Clark RL, Deane FM, Anthony NG, Johnston BF, McCarthy FO, Mackay SP. Clark RL, et al. Among authors: mackay sp. Bioorg Med Chem. 2007 Jul 15;15(14):4741-52. doi: 10.1016/j.bmc.2007.05.002. Epub 2007 May 6. Bioorg Med Chem. 2007. PMID: 17517513

3

2-Aryl-3,3,3-trifluoro-2-hydroxypropionic acids: a new class of protein tyrosine phosphatase 1B inhibitors.

Adams DR, Abraham A, Asano J, Breslin C, Dick CA, Ixkes U, Johnston BF, Johnston D, Kewnay J, Mackay SP, MacKenzie SJ, McFarlane M, Mitchell L, Spinks D, Takano Y. Adams DR, et al. Among authors: mackay sp. Bioorg Med Chem Lett. 2007 Dec 1;17(23):6579-83. doi: 10.1016/j.bmcl.2007.09.069. Epub 2007 Sep 25. Bioorg Med Chem Lett. 2007. PMID: 17931864

4

Manganese dioxide mediated one-pot synthesis of methyl 9H-pyrido[3,4-b]indole-1-carboxylate: Concise synthesis of alangiobussinine.

Baiget J, Llona-Minguez S, Lang S, Mackay SP, Suckling CJ, Sutcliffe OB. Baiget J, et al. Among authors: mackay sp. Beilstein J Org Chem. 2011;7:1407-11. doi: 10.3762/bjoc.7.164. Epub 2011 Oct 12. Beilstein J Org Chem. 2011. PMID: 22043251 Free PMC article.

5

Doing the methylene shuffle--further insights into the inhibition of mitotic kinesin Eg5 with S-trityl L-cysteine.

Abualhasan MN, Good JA, Wittayanarakul K, Anthony NG, Berretta G, Rath O, Kozielski F, Sutcliffe OB, Mackay SP. Abualhasan MN, et al. Among authors: mackay sp. Eur J Med Chem. 2012 Aug;54:483-98. doi: 10.1016/j.ejmech.2012.05.034. Epub 2012 Jun 7. Eur J Med Chem. 2012. PMID: 22749640

6

Identification and development of the 1,4-benzodiazepin-2-one and quinazoline-2,4-dione scaffolds as submicromolar inhibitors of HAT.

Clark RL, Clements CJ, Barrett MP, Mackay SP, Rathnam RP, Owusu-Dapaah G, Spencer J, Huggan JK. Clark RL, et al. Among authors: mackay sp. Bioorg Med Chem. 2012 Oct 15;20(20):6019-33. doi: 10.1016/j.bmc.2012.08.049. Epub 2012 Aug 31. Bioorg Med Chem. 2012. PMID: 22985960

7

Structure-activity relationships and molecular modeling of sphingosine kinase inhibitors.

Baek DJ, MacRitchie N, Anthony NG, Mackay SP, Pyne S, Pyne NJ, Bittman R. Baek DJ, et al. Among authors: mackay sp. J Med Chem. 2013 Nov 27;56(22):9310-27. doi: 10.1021/jm401399c. Epub 2013 Nov 14. J Med Chem. 2013. PMID: 24164513 Free PMC article.

8

Small-molecule inhibitors of IκB kinase (IKK) and IKK-related kinases.

Llona-Minguez S, Baiget J, Mackay SP. Llona-Minguez S, et al. Among authors: mackay sp. Pharm Pat Anal. 2013 Jul;2(4):481-98. doi: 10.4155/ppa.13.31. Pharm Pat Anal. 2013. PMID: 24237125 Review.

9

Resveratrol and its oligomers: modulation of sphingolipid metabolism and signaling in disease.

Lim KG, Gray AI, Anthony NG, Mackay SP, Pyne S, Pyne NJ. Lim KG, et al. Among authors: mackay sp. Arch Toxicol. 2014 Dec;88(12):2213-32. doi: 10.1007/s00204-014-1386-4. Epub 2014 Oct 25. Arch Toxicol. 2014. PMID: 25344023 Free article. Review.

10

Inhibitory Kappa B Kinase α (IKKα) Inhibitors That Recapitulate Their Selectivity in Cells against Isoform-Related Biomarkers.

Anthony NG, Baiget J, Berretta G, Boyd M, Breen D, Edwards J, Gamble C, Gray AI, Harvey AL, Hatziieremia S, Ho KH, Huggan JK, Lang S, Llona-Minguez S, Luo JL, McIntosh K, Paul A, Plevin RJ, Robertson MN, Scott R, Suckling CJ, Sutcliffe OB, Young LC, Mackay SP. Anthony NG, et al. Among authors: mackay sp. J Med Chem. 2017 Aug 24;60(16):7043-7066. doi: 10.1021/acs.jmedchem.7b00484. Epub 2017 Aug 15. J Med Chem. 2017. PMID: 28737909 Free PMC article.

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