Discovery of BMS-986251: A Clinically Viable, Potent, and Selective RORγt Inverse Agonist.
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Cherney RJ, et al. Among authors: zhao q.
ACS Med Chem Lett. 2020 Mar 31;11(6):1221-1227. doi: 10.1021/acsmedchemlett.0c00063. eCollection 2020 Jun 11.
ACS Med Chem Lett. 2020.
PMID: 32551004
Free PMC article.