Sparling BA - Search Results

1

Pharmacological Assessment of Sepiapterin Reductase Inhibition on Tactile Response in the Rat.

Meyer JT, Sparling BA, McCarty WJ, Zhang M, Soto M, Schneider S, Chen H, Roberts J, Tan H, Kornecook T, Andrews PS, Knutson CG. Meyer JT, et al. Among authors: sparling ba. J Pharmacol Exp Ther. 2019 Nov;371(2):476-486. doi: 10.1124/jpet.119.257105. Epub 2019 May 20. J Pharmacol Exp Ther. 2019. PMID: 31110114

2

Virtual screening to identify potent sepiapterin reductase inhibitors.

Gao H, Schneider S, Andrews P, Wang K, Huang X, Sparling BA. Gao H, et al. Among authors: sparling ba. Bioorg Med Chem Lett. 2020 Jan 15;30(2):126793. doi: 10.1016/j.bmcl.2019.126793. Epub 2019 Nov 9. Bioorg Med Chem Lett. 2020. PMID: 31740247

3

Sulfonamides as Selective Na_V1.7 Inhibitors: Optimizing Potency, Pharmacokinetics, and Metabolic Properties to Obtain Atropisomeric Quinolinone (AM-0466) that Affords Robust in Vivo Activity.

Graceffa RF, Boezio AA, Able J, Altmann S, Berry LM, Boezio C, Butler JR, Chu-Moyer M, Cooke M, DiMauro EF, Dineen TA, Feric Bojic E, Foti RS, Fremeau RT Jr, Guzman-Perez A, Gao H, Gunaydin H, Huang H, Huang L, Ilch C, Jarosh M, Kornecook T, Kreiman CR, La DS, Ligutti J, Milgram BC, Lin MJ, Marx IE, Nguyen HN, Peterson EA, Rescourio G, Roberts J, Schenkel L, Shimanovich R, Sparling BA, Stellwagen J, Taborn K, Vaida KR, Wang J, Yeoman J, Yu V, Zhu D, Moyer BD, Weiss MM. Graceffa RF, et al. Among authors: sparling ba. J Med Chem. 2017 Jul 27;60(14):5990-6017. doi: 10.1021/acs.jmedchem.6b01850. Epub 2017 Apr 20. J Med Chem. 2017. PMID: 28324649

4

Discovery and hit-to-lead evaluation of piperazine amides as selective, state-dependent Na_V1.7 inhibitors.

Sparling BA, Yi S, Able J, Bregman H, DiMauro EF, Foti RS, Gao H, Guzman-Perez A, Huang H, Jarosh M, Kornecook T, Ligutti J, Milgram BC, Moyer BD, Youngblood B, Yu VL, Weiss MM. Sparling BA, et al. Medchemcomm. 2016 Dec 2;8(4):744-754. doi: 10.1039/c6md00578k. eCollection 2017 Apr 1. Medchemcomm. 2016. PMID: 30108793 Free PMC article.

5

Progress in the discovery of small molecule modulators of the Cys-loop superfamily receptors.

Sparling BA, DiMauro EF. Sparling BA, et al. Bioorg Med Chem Lett. 2017 Aug 1;27(15):3207-3218. doi: 10.1016/j.bmcl.2017.04.073. Epub 2017 May 4. Bioorg Med Chem Lett. 2017. PMID: 28606760 Review.

6

Sustainable Practices in Medicinal Chemistry Part 2: Green by Design.

Aliagas I, Berger R, Goldberg K, Nishimura RT, Reilly J, Richardson P, Richter D, Sherer EC, Sparling BA, Bryan MC. Aliagas I, et al. Among authors: sparling ba. J Med Chem. 2017 Jul 27;60(14):5955-5968. doi: 10.1021/acs.jmedchem.6b01837. Epub 2017 Apr 12. J Med Chem. 2017. PMID: 28375009 Review.

7

High-Throughput Implementation of the NanoBRET Target Engagement Intracellular Kinase Assay to Reveal Differential Compound Engagement by SIK2/3 Isoforms.

Jin HY, Tudor Y, Choi K, Shao Z, Sparling BA, McGivern JG, Symons A. Jin HY, et al. Among authors: sparling ba. SLAS Discov. 2020 Feb;25(2):215-222. doi: 10.1177/2472555219893277. Epub 2019 Dec 18. SLAS Discov. 2020. PMID: 31849250 Free article.

8

Decarboxylative Anti-Michael Addition to Olefins Mediated by Photoredox Catalysis.

Lovett GH, Sparling BA. Lovett GH, et al. Among authors: sparling ba. Org Lett. 2016 Jul 15;18(14):3494-7. doi: 10.1021/acs.orglett.6b01712. Epub 2016 Jul 1. Org Lett. 2016. PMID: 27364853

9

Total Synthesis of (-)-Nemorosone and (+)-Secohyperforin.

Sparling BA, Tucker JK, Moebius DC, Shair MD. Sparling BA, et al. Org Lett. 2015 Jul 17;17(14):3398-401. doi: 10.1021/acs.orglett.5b01121. Epub 2015 Jun 30. Org Lett. 2015. PMID: 26125288

10

Enantioselective total synthesis of hyperforin.

Sparling BA, Moebius DC, Shair MD. Sparling BA, et al. J Am Chem Soc. 2013 Jan 16;135(2):644-7. doi: 10.1021/ja312150d. Epub 2012 Dec 31. J Am Chem Soc. 2013. PMID: 23270309

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My Custom Filters

Publication date

Text availability

Article attribute

Article type

Article Language

Species

Sex

Age

Other

15 results

Search Page

Filters