Nikulin V - Search Results

1

Discovery of Orally Active Hydroxyethylamine Based SPPL2a Inhibitors.

Velcicky J, Mathison CJN, Nikulin V, Pflieger D, Epple R, Azimioara M, Cow C, Michellys PY, Rigollier P, Beisner DR, Bodendorf U, Guerini D, Liu B, Wen B, Zaharevitz S, Brandl T. Velcicky J, et al. Among authors: nikulin v. ACS Med Chem Lett. 2019 May 23;10(6):887-892. doi: 10.1021/acsmedchemlett.9b00044. eCollection 2019 Jun 13. ACS Med Chem Lett. 2019. PMID: 31223443 Free PMC article.

2

Discovery of structurally novel, potent and orally efficacious GPR119 agonists.

Alper P, Azimioara M, Cow C, Mutnick D, Nikulin V, Michellys PY, Wang Z, Reding E, Paliotti M, Li J, Bao D, Zoll J, Kim Y, Zimmerman M, Groessel T, Tuntland T, Joseph SB, McNamara P, Seidel HM, Epple R. Alper P, et al. Among authors: nikulin v. Bioorg Med Chem Lett. 2014 May 15;24(10):2383-7. doi: 10.1016/j.bmcl.2014.03.023. Epub 2014 Mar 27. Bioorg Med Chem Lett. 2014. PMID: 24751443

3

Novel tricyclic pyrazolopyrimidines as potent and selective GPR119 agonists.

Azimioara M, Alper P, Cow C, Mutnick D, Nikulin V, Lelais G, Mecom J, McNeill M, Michellys PY, Wang Z, Reding E, Paliotti M, Li J, Bao D, Zoll J, Kim Y, Zimmerman M, Groessl T, Tuntland T, Joseph SB, McNamara P, Seidel HM, Epple R. Azimioara M, et al. Among authors: nikulin v. Bioorg Med Chem Lett. 2014 Dec 1;24(23):5478-83. doi: 10.1016/j.bmcl.2014.10.010. Epub 2014 Oct 13. Bioorg Med Chem Lett. 2014. PMID: 25455488

4

Structure-Based Design of Selective LONP1 Inhibitors for Probing In Vitro Biology.

Kingsley LJ, He X, McNeill M, Nelson J, Nikulin V, Ma Z, Lu W, Zhou VW, Manuia M, Kreusch A, Gao MY, Witmer D, Vaillancourt MT, Lu M, Greenblatt S, Lee C, Vashisht A, Bender S, Spraggon G, Michellys PY, Jia Y, Haling JR, Lelais G. Kingsley LJ, et al. Among authors: nikulin v. J Med Chem. 2021 Apr 22;64(8):4857-4869. doi: 10.1021/acs.jmedchem.0c02152. Epub 2021 Apr 6. J Med Chem. 2021. PMID: 33821636

5

Structure-based design, synthesis, and antimicrobial activity of indazole-derived SAH/MTA nucleosidase inhibitors.

Li X, Chu S, Feher VA, Khalili M, Nie Z, Margosiak S, Nikulin V, Levin J, Sprankle KG, Tedder ME, Almassy R, Appelt K, Yager KM. Li X, et al. Among authors: nikulin v. J Med Chem. 2003 Dec 18;46(26):5663-73. doi: 10.1021/jm0302039. J Med Chem. 2003. PMID: 14667220

6

Structure-based design, synthesis, and study of potent inhibitors of beta-ketoacyl-acyl carrier protein synthase III as potential antimicrobial agents.

Nie Z, Perretta C, Lu J, Su Y, Margosiak S, Gajiwala KS, Cortez J, Nikulin V, Yager KM, Appelt K, Chu S. Nie Z, et al. Among authors: nikulin v. J Med Chem. 2005 Mar 10;48(5):1596-609. doi: 10.1021/jm049141s. J Med Chem. 2005. PMID: 15743201

7

Iodinated analogs of trimetoquinol as highly potent and selective beta 2-adrenoceptor ligands.

De Los Angeles JE, Nikulin VI, Shams G, Konkar AA, Mehta R, Feller DR, Miller DD. De Los Angeles JE, et al. Among authors: nikulin vi. J Med Chem. 1996 Sep 13;39(19):3701-11. doi: 10.1021/jm960208o. J Med Chem. 1996. PMID: 8809159

8

2-Amino-4-benzyl-4,5,6,7-tetrahydrothiazolo[5,4-c]pyridines: novel selective beta3-adrenoceptor agonists.

Zheng W, Nikulin VI, Konkar AA, Vansal SS, Shams G, Feller DR, Miller DD. Zheng W, et al. Among authors: nikulin vi. J Med Chem. 1999 Jun 17;42(12):2287-94. doi: 10.1021/jm990012z. J Med Chem. 1999. PMID: 10377236

9

1-Benzyl-1,2,3,4-tetrahydroisoquinoline-6,7-diols as novel affinity and photoaffinity probes for beta-adrenoceptor subtypes.

Nikulin VI, Rakov IM, De Los Angeles JE, Mehta RC, Boyd LY, Feller DR, Miller DD. Nikulin VI, et al. Bioorg Med Chem. 2006 Mar 15;14(6):1684-97. doi: 10.1016/j.bmc.2005.12.027. Epub 2006 Jan 20. Bioorg Med Chem. 2006. PMID: 16431119

10

Synthesis and human beta-adrenoceptor activity of 1-(3,5-diiodo-4- methoxybenzyl)-1,2,3,4-tetrahydroisoquinolin-6-ol derivatives in vitro.

He Y, Nikulin VI, Vansal SS, Feller DR, Miller DD. He Y, et al. Among authors: nikulin vi. J Med Chem. 2000 Feb 24;43(4):591-8. doi: 10.1021/jm990463j. J Med Chem. 2000. PMID: 10691685

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