Baell JB - Search Results

1

Discovery of Acylsulfonohydrazide-Derived Inhibitors of the Lysine Acetyltransferase, KAT6A, as Potent Senescence-Inducing Anti-Cancer Agents.

Priebbenow DL, Leaver DJ, Nguyen N, Cleary B, Lagiakos HR, Sanchez J, Xue L, Huang F, Sun Y, Mujumdar P, Mudududdla R, Varghese S, Teguh S, Charman SA, White KL, Shackleford DM, Katneni K, Cuellar M, Strasser JM, Dahlin JL, Walters MA, Street IP, Monahan BJ, Jarman KE, Jousset Sabroux H, Falk H, Chung MC, Hermans SJ, Downer NL, Parker MW, Voss AK, Thomas T, Baell JB. Priebbenow DL, et al. Among authors: baell jb. J Med Chem. 2020 May 14;63(9):4655-4684. doi: 10.1021/acs.jmedchem.9b02071. Epub 2020 Mar 19. J Med Chem. 2020. PMID: 32118427

2

Khellinone derivatives as blockers of the voltage-gated potassium channel Kv1.3: synthesis and immunosuppressive activity.

Baell JB, Gable RW, Harvey AJ, Toovey N, Herzog T, Hänsel W, Wulff H. Baell JB, et al. J Med Chem. 2004 Apr 22;47(9):2326-36. doi: 10.1021/jm030523s. J Med Chem. 2004. PMID: 15084131

3

Synthesis and biological evaluation of nonpeptide mimetics of omega-conotoxin GVIA.

Baell JB, Duggan PJ, Forsyth SA, Lewis RJ, Lok YP, Schroeder CI. Baell JB, et al. Bioorg Med Chem. 2004 Aug 1;12(15):4025-37. doi: 10.1016/j.bmc.2004.05.040. Bioorg Med Chem. 2004. PMID: 15246080

4

Phosphate isosteres in medicinal chemistry.

Rye CS, Baell JB. Rye CS, et al. Among authors: baell jb. Curr Med Chem. 2005;12(26):3127-41. doi: 10.2174/092986705774933452. Curr Med Chem. 2005. PMID: 16375706 Review.

5

A new class of blockers of the voltage-gated potassium channel Kv1.3 via modification of the 4- or 7-position of khellinone.

Harvey AJ, Baell JB, Toovey N, Homerick D, Wulff H. Harvey AJ, et al. Among authors: baell jb. J Med Chem. 2006 Feb 23;49(4):1433-41. doi: 10.1021/jm050839v. J Med Chem. 2006. PMID: 16480279

6

Discovery of 2-iminobenzimidazoles as a new class of trypanothione reductase inhibitor by high-throughput screening.

Holloway GA, Baell JB, Fairlamb AH, Novello PM, Parisot JP, Richardson J, Watson KG, Street IP. Holloway GA, et al. Among authors: baell jb. Bioorg Med Chem Lett. 2007 Mar 1;17(5):1422-7. doi: 10.1016/j.bmcl.2006.11.090. Epub 2006 Dec 3. Bioorg Med Chem Lett. 2007. PMID: 17194585 Free PMC article.

7

Synthesis and biological evaluation of chalcones as inhibitors of the voltage-gated potassium channel Kv1.3.

Cianci J, Baell JB, Flynn BL, Gable RW, Mould JA, Paul D, Harvey AJ. Cianci J, et al. Among authors: baell jb. Bioorg Med Chem Lett. 2008 Mar 15;18(6):2055-61. doi: 10.1016/j.bmcl.2008.01.099. Epub 2008 Jan 31. Bioorg Med Chem Lett. 2008. PMID: 18289849

8

Trypanothione reductase high-throughput screening campaign identifies novel classes of inhibitors with antiparasitic activity.

Holloway GA, Charman WN, Fairlamb AH, Brun R, Kaiser M, Kostewicz E, Novello PM, Parisot JP, Richardson J, Street IP, Watson KG, Baell JB. Holloway GA, et al. Among authors: baell jb. Antimicrob Agents Chemother. 2009 Jul;53(7):2824-33. doi: 10.1128/AAC.01568-08. Epub 2009 Apr 13. Antimicrob Agents Chemother. 2009. PMID: 19364854 Free PMC article.

9

New substructure filters for removal of pan assay interference compounds (PAINS) from screening libraries and for their exclusion in bioassays.

Baell JB, Holloway GA. Baell JB, et al. J Med Chem. 2010 Apr 8;53(7):2719-40. doi: 10.1021/jm901137j. J Med Chem. 2010. PMID: 20131845

10

Inhibitors of Leishmania GDP-mannose pyrophosphorylase identified by high-throughput screening of small-molecule chemical library.

Lackovic K, Parisot JP, Sleebs N, Baell JB, Debien L, Watson KG, Curtis JM, Handman E, Street IP, Kedzierski L. Lackovic K, et al. Among authors: baell jb. Antimicrob Agents Chemother. 2010 May;54(5):1712-9. doi: 10.1128/AAC.01634-09. Epub 2010 Feb 16. Antimicrob Agents Chemother. 2010. PMID: 20160053 Free PMC article.

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