García-Mera X - Search Results

1

3,4-Dihydropyrimidin-2(1H)-ones as Antagonists of the Human A_2B Adenosine Receptor: Optimization, Structure-Activity Relationship Studies, and Enantiospecific Recognition.

Majellaro M, Jespers W, Crespo A, Núñez MJ, Novio S, Azuaje J, Prieto-Díaz R, Gioé C, Alispahic B, Brea J, Loza MI, Freire-Garabal M, Garcia-Santiago C, Rodríguez-García C, García-Mera X, Caamaño O, Fernandez-Masaguer C, Sardina JF, Stefanachi A, El Maatougui A, Mallo-Abreu A, Åqvist J, Gutiérrez-de-Terán H, Sotelo E. Majellaro M, et al. J Med Chem. 2021 Jan 14;64(1):458-480. doi: 10.1021/acs.jmedchem.0c01431. Epub 2020 Dec 29. J Med Chem. 2021. PMID: 33372800

2

Synthesis, antiviral and cytostatic activities of carbocyclic nucleosides incorporating a modified cyclopentane ring. Part 2: Adenosine and uridine analogues.

Nieto MI, Blanco JM, Caamaño O, Fernández F, García-Mera X, Balzarini J, Padalko E, Neyts J, De Clercq E. Nieto MI, et al. Nucleosides Nucleotides. 1998 Jul;17(7):1255-66. doi: 10.1080/07328319808004237. Nucleosides Nucleotides. 1998. PMID: 9708318

3

Synthesis and antiviral and antineoplastic activities of some novel carbocyclic guanosine analogues with a cyclobutane ring.

Blanco JM, Caamaño O, Fernández F, García-Mera X, Hergueta AR, López C, Rodríguez-borges JE, Balzarini J, De Clercq E. Blanco JM, et al. Chem Pharm Bull (Tokyo). 1999 Sep;47(9):1314-7. doi: 10.1248/cpb.47.1314. Chem Pharm Bull (Tokyo). 1999. PMID: 10517011

4

Synthesis and antiviral and cytostatic activities of carbocyclic nucleosides incorporating a modified cyclobutane ring. Part 1: Guanosine analogues.

Figueira MJ, Blanco JM, Caamaño O, Fernández F, García-Mera X, López C. Figueira MJ, et al. Arch Pharm (Weinheim). 1999 Oct;332(10):348-52. doi: 10.1002/(sici)1521-4184(199910)332:10<348::aid-ardp348>3.0.co;2-h. Arch Pharm (Weinheim). 1999. PMID: 10575367

5

Synthesis and antiviral activity of carbocyclic nucleosides incorporating a modified cyclopentane ring. Part 3: Adenosine and uridine analogues.

Isabel Nieto M, Manuel Blanco J, Caamaño O, Fernández F, García-Mera X, López C, Balzarini J, De Clercq E. Isabel Nieto M, et al. Nucleosides Nucleotides. 1999 Oct;18(10):2253-63. doi: 10.1080/07328319908044879. Nucleosides Nucleotides. 1999. PMID: 10616729

6

2-Substituted 4-, 5-, and 6-[(1E)-3-oxo-3-phenylprop-1-en-1-yl]pyridazin-3(2H)-ones and 2-substituted 4,5-bis[(1E)-3-oxo-3-phenylprop-1-en-1-yl]pyridazin-3(2H)-ones as potent platelet aggregation inhibitors: design, synthesis, and SAR studies.

Meyers C, Yáñez M, Elmaatougi A, Verhelst T, Coelho A, Fraiz N, Lemière GL, García-Mera X, Laguna R, Cano E, Maes BU, Sotelo E. Meyers C, et al. Bioorg Med Chem Lett. 2008 Jan 15;18(2):793-7. doi: 10.1016/j.bmcl.2007.11.034. Epub 2007 Nov 17. Bioorg Med Chem Lett. 2008. PMID: 18053717

7

Click chemistry approach to assembly proline mimetic libraries containing 1,4-substituted 1,2,3-triazoles.

Rodríguez-Borges JE, Gonçalves S, do Vale ML, García-Mera X, Coelho A, Sotelo E. Rodríguez-Borges JE, et al. J Comb Chem. 2008 May-Jun;10(3):372-5. doi: 10.1021/cc800035z. Epub 2008 Apr 30. J Comb Chem. 2008. PMID: 18444684 No abstract available.

8

Synthesis of novel purinyl-1'-homocarbanucleosides based on a cyclopenta[b]pyrazine system.

Balo C, López C, Caamaño O, Fernández F, García-Mera X, Rodríguez-Borges JE. Balo C, et al. Chem Pharm Bull (Tokyo). 2008 May;56(5):654-8. doi: 10.1248/cpb.56.654. Chem Pharm Bull (Tokyo). 2008. PMID: 18451552 Free article.

9

1,3-dialkyl-8-N-substituted benzyloxycarbonylamino-9-deazaxanthines as potent adenosine receptor ligands: Design, synthesis, structure-affinity and structure-selectivity relationships.

Fernández F, Caamaño O, Isabel Nieto M, López C, García-Mera X, Stefanachi A, Nicolotti O, Isabel Loza M, Brea J, Esteve C, Segarra V, Vidal B, Carotti A. Fernández F, et al. Bioorg Med Chem. 2009 May 15;17(10):3618-29. doi: 10.1016/j.bmc.2009.03.062. Epub 2009 Apr 5. Bioorg Med Chem. 2009. PMID: 19398343

10

Divergent solution-phase synthesis of diarylpyrimidine libraries as selective A3 adenosine receptor antagonists.

Yaziji V, Coelho A, El Maatougui A, Brea J, Loza MI, Garcia-Mera X, Sotelo E. Yaziji V, et al. J Comb Chem. 2009 Jul-Aug;11(4):519-22. doi: 10.1021/cc900044k. J Comb Chem. 2009. PMID: 19472983

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