Dombrowski A - Search Results

1

Development of Orally Efficacious Allosteric Inhibitors of TNFα via Fragment-Based Drug Design.

Dietrich JD, Longenecker KL, Wilson NS, Goess C, Panchal SC, Swann SL, Petros AM, Hobson AD, Ihle D, Song D, Richardson P, Comess KM, Cox PB, Dombrowski A, Sarris K, Donnelly-Roberts DL, Duignan DB, Gomtsyan A, Jung P, Krueger AC, Mathieu S, McClure A, Stoll VS, Wetter J, Mankovich JA, Hajduk PJ, Vasudevan A, Stoffel RH, Sun C. Dietrich JD, et al. Among authors: dombrowski a. J Med Chem. 2021 Jan 14;64(1):417-429. doi: 10.1021/acs.jmedchem.0c01280. Epub 2020 Dec 30. J Med Chem. 2021. PMID: 33378180

2

Emerging Trends in Flow Chemistry and Applications to the Pharmaceutical Industry.

Bogdan AR, Dombrowski AW. Bogdan AR, et al. J Med Chem. 2019 Jul 25;62(14):6422-6468. doi: 10.1021/acs.jmedchem.8b01760. Epub 2019 Mar 8. J Med Chem. 2019. PMID: 30794752

3

High-Throughput Reaction Screening with Nanomoles of Solid Reagents Coated on Glass Beads.

Tu NP, Dombrowski AW, Goshu GM, Vasudevan A, Djuric SW, Wang Y. Tu NP, et al. Among authors: dombrowski aw. Angew Chem Int Ed Engl. 2019 Jun 11;58(24):7987-7991. doi: 10.1002/anie.201900536. Epub 2019 May 7. Angew Chem Int Ed Engl. 2019. PMID: 30891860

4

The Chosen Few: Parallel Library Reaction Methodologies for Drug Discovery.

Dombrowski AW, Aguirre AL, Shrestha A, Sarris KA, Wang Y. Dombrowski AW, et al. J Org Chem. 2022 Feb 18;87(4):1880-1897. doi: 10.1021/acs.joc.1c01427. Epub 2021 Nov 15. J Org Chem. 2022. PMID: 34780177

5

[No title available]

[No authors listed] [No authors listed] PMID: 39291026

6

Expanding the Medicinal Chemist Toolbox: Comparing Seven C(sp²)-C(sp³) Cross-Coupling Methods by Library Synthesis.

Dombrowski AW, Gesmundo NJ, Aguirre AL, Sarris KA, Young JM, Bogdan AR, Martin MC, Gedeon S, Wang Y. Dombrowski AW, et al. ACS Med Chem Lett. 2020 Mar 23;11(4):597-604. doi: 10.1021/acsmedchemlett.0c00093. eCollection 2020 Apr 9. ACS Med Chem Lett. 2020. PMID: 32292569 Free PMC article.

7

Rearrangement of 3-Hydroxyazetidines into 2-Oxazolines.

Ruggeri M, Dombrowski AW, Djuric SW, Baxendale IR. Ruggeri M, et al. J Org Chem. 2020 Jun 5;85(11):7276-7286. doi: 10.1021/acs.joc.0c00656. Epub 2020 May 12. J Org Chem. 2020. PMID: 32369365

8

Di(2-picolyl)amines as Modular and Robust Ligands for Nickel-Catalyzed C(sp²)-C(sp³) Cross-Electrophile Coupling.

Rago AJ, Vasilopoulos A, Dombrowski AW, Wang Y. Rago AJ, et al. Among authors: dombrowski aw. Org Lett. 2022 Nov 25;24(46):8487-8492. doi: 10.1021/acs.orglett.2c03346. Epub 2022 Nov 15. Org Lett. 2022. PMID: 36377969

9

Incorporating Synthetic Accessibility in Drug Design: Predicting Reaction Yields of Suzuki Cross-Couplings by Leveraging AbbVie's 15-Year Parallel Library Data Set.

Raghavan P, Rago AJ, Verma P, Hassan MM, Goshu GM, Dombrowski AW, Pandey A, Coley CW, Wang Y. Raghavan P, et al. Among authors: dombrowski aw. J Am Chem Soc. 2024 Jun 5;146(22):15070-15084. doi: 10.1021/jacs.4c00098. Epub 2024 May 20. J Am Chem Soc. 2024. PMID: 38768950 Free PMC article.

10

High-Temperature Boc Deprotection in Flow and Its Application in Multistep Reaction Sequences.

Bogdan AR, Charaschanya M, Dombrowski AW, Wang Y, Djuric SW. Bogdan AR, et al. Org Lett. 2016 Apr 15;18(8):1732-5. doi: 10.1021/acs.orglett.6b00378. Epub 2016 Apr 5. Org Lett. 2016. PMID: 27046640

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