De Graef S - Search Results

1

The in-vitro effect of famotidine on sars-cov-2 proteases and virus replication.

Loffredo M, Lucero H, Chen DY, O'Connell A, Bergqvist S, Munawar A, Bandara A, De Graef S, Weeks SD, Douam F, Saeed M, Munawar AH. Loffredo M, et al. Among authors: de graef s. Sci Rep. 2021 Mar 8;11(1):5433. doi: 10.1038/s41598-021-84782-w. Sci Rep. 2021. PMID: 33686143 Free PMC article.

2

Comparative analysis of pyrimidine substituted aminoacyl-sulfamoyl nucleosides as potential inhibitors targeting class I aminoacyl-tRNA synthetases.

Nautiyal M, De Graef S, Pang L, Gadakh B, Strelkov SV, Weeks SD, Van Aerschot A. Nautiyal M, et al. Among authors: de graef s. Eur J Med Chem. 2019 Jul 1;173:154-166. doi: 10.1016/j.ejmech.2019.04.003. Epub 2019 Apr 5. Eur J Med Chem. 2019. PMID: 30995568

3

Synthesis and Biological Evaluation of 1,3-Dideazapurine-Like 7-Amino-5-Hydroxymethyl-Benzimidazole Ribonucleoside Analogues as Aminoacyl-tRNA Synthetase Inhibitors.

Zhang B, Pang L, Nautiyal M, De Graef S, Gadakh B, Lescrinier E, Rozenski J, Strelkov SV, Weeks SD, Van Aerschot A. Zhang B, et al. Among authors: de graef s. Molecules. 2020 Oct 16;25(20):4751. doi: 10.3390/molecules25204751. Molecules. 2020. PMID: 33081246 Free PMC article.

4

Synthesis and structural insights into the binding mode of the albomycin δ1 core and its analogues in complex with their target aminoacyl-tRNA synthetase.

Gadakh B, Vondenhoff G, Pang L, Nautiyal M, De Graef S, Strelkov SV, Weeks SD, Van Aerschot A. Gadakh B, et al. Among authors: de graef s. Bioorg Med Chem. 2020 Sep 1;28(17):115645. doi: 10.1016/j.bmc.2020.115645. Epub 2020 Jul 13. Bioorg Med Chem. 2020. PMID: 32773091

5

Phenyltriazole-functionalized sulfamate inhibitors targeting tyrosyl- or isoleucyl-tRNA synthetase.

De Ruysscher D, Pang L, Mattelaer CA, Nautiyal M, De Graef S, Rozenski J, Strelkov SV, Lescrinier E, Weeks SD, Van Aerschot A. De Ruysscher D, et al. Among authors: de graef s. Bioorg Med Chem. 2020 Aug 1;28(15):115580. doi: 10.1016/j.bmc.2020.115580. Epub 2020 Jun 5. Bioorg Med Chem. 2020. PMID: 32631562

6

Structural Insights into the Binding of Natural Pyrimidine-Based Inhibitors of Class II Aminoacyl-tRNA Synthetases.

Pang L, Nautiyal M, De Graef S, Gadakh B, Zorzini V, Economou A, Strelkov SV, Van Aerschot A, Weeks SD. Pang L, et al. Among authors: de graef s. ACS Chem Biol. 2020 Feb 21;15(2):407-415. doi: 10.1021/acschembio.9b00887. Epub 2020 Jan 8. ACS Chem Biol. 2020. PMID: 31869198

7

Family-wide analysis of aminoacyl-sulfamoyl-3-deazaadenosine analogues as inhibitors of aminoacyl-tRNA synthetases.

Zhang B, De Graef S, Nautiyal M, Pang L, Gadakh B, Froeyen M, Van Mellaert L, Strelkov SV, Weeks SD, Van Aerschot A. Zhang B, et al. Among authors: de graef s. Eur J Med Chem. 2018 Mar 25;148:384-396. doi: 10.1016/j.ejmech.2018.02.013. Epub 2018 Feb 14. Eur J Med Chem. 2018. PMID: 29477072

8

Acylated sulfonamide adenosines as potent inhibitors of the adenylate-forming enzyme superfamily.

De Ruysscher D, Pang L, De Graef S, Nautiyal M, De Borggraeve WM, Rozenski J, Strelkov SV, Weeks SD, Van Aerschot A. De Ruysscher D, et al. Among authors: de graef s. Eur J Med Chem. 2019 Jul 15;174:252-264. doi: 10.1016/j.ejmech.2019.04.045. Epub 2019 Apr 17. Eur J Med Chem. 2019. PMID: 31048140

9

Synthesis and Biological Evaluation of Lipophilic Nucleoside Analogues as Inhibitors of Aminoacyl-tRNA Synthetases.

Nautiyal M, Gadakh B, De Graef S, Pang L, Khan M, Xun Y, Rozenski J, Van Aerschot A. Nautiyal M, et al. Among authors: de graef s. Antibiotics (Basel). 2019 Oct 9;8(4):180. doi: 10.3390/antibiotics8040180. Antibiotics (Basel). 2019. PMID: 31600972 Free PMC article.

10

Prognostic indicators in breast cancer--morphometric methods.

Baak JP, Kurver PH, De Snoo-Niewlaat AJ, De Graef S, Makkink B, Boon ME. Baak JP, et al. Among authors: de graef s. Histopathology. 1982 May;6(3):327-39. doi: 10.1111/j.1365-2559.1982.tb02727.x. Histopathology. 1982. PMID: 7095760

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